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472 results found for "Stefano Moro"
- Structural perspectives on the mechanism of signal activation, ligand selectivity and allosteric...
Thus, we need to know much more about the structures of receptor-ligand complexes at high resolution. Read more at the source #DrGPCR #GPCR #IndustryNews
- 📰 GPCR Weekly News, April 8 to 14, 2024
Stay updated for more details. Do you want to re-watch our recorded events? GPCR Symposiums and much more! relaxation of human coronary arteries: A key role for Gβγ subunit instead of cAMP GPCR Binders, Drugs, and more peptides that are self-secreted by yeast expressing a G-protein-coupled receptor Reviews, GPCRs, and more
- AlphaFold’s Breakthrough in GPCR Research: Revolutionizing Discovery, Yet Awaiting Experimental Proof
striking: AlphaFold2 outperformed homology models, achieving a 60% hit rate for compounds targeting TAAR1, more integration with other computational techniques, could help overcome these limitations, leading to more
- A broad look into the future of systemic sclerosis
angiotensin II receptor subtype 1 (AT1R) and the endothelin receptor type A (ETAR) are discussed in more Read more at the source #DrGPCR #GPCR #IndustryNews
- 📰 GPCR Weekly News, April 1 to 7, 2024
Stay updated for more details. Do you want to re-watch our recorded events? GPCR Symposiums and much more! Intracellular pocket conformations determine signaling through the μ opioid receptor GPCR Binders, Drugs, and more
- Comparative study of neuropeptide signaling systems in Hemiptera
This research provides more knowledge on neuropeptide systems and sets the groundwork for the creation Read more at the source #DrGPCR #GPCR #IndustryNews
- Although the cannabinoid type-2 receptor (CB2) is highly expressed in the immune system, emerging...
While more work is needed to further elucidate the translational value of selectively targeting CB2 receptors Read more at the source #DrGPCR #GPCR #IndustryNews
- Structures of β 1-adrenergic receptor in complex with Gs and ligands of different efficacies
investigations uncover that the intermediate state complex comprising β1-AR and nucleotide-free Gs is more Read more at the source #DrGPCR #GPCR #IndustryNews
- Immerse yourself in the Dr. GPCR Ecosystem!
Catch up with the latest #GPCR news, our monthly Virtual Cafe, and much more!
- Ermium Therapeutics has constituted its SAB
leaders in GPCRs pharmacology, immunology, drug discovery and development for auto-immune diseases" Read more
- Discovery of 3(2-aminoethyl)-thiazolidine-2,4-diones as a novel chemotype of sigma-1 receptor ligand
Six compounds showed more than 50% displacement of the radioligand at 10 µM concentration with compound Read more at the source #DrGPCR #GPCR #IndustryNews
- 🧠Do you want to share your #GPCR knowledge?
GPCR Ecosystem and create a course on your favorite #GPCR research, technique and more… Available for
- 2nd IRN i-GPCRnet, September 30 to October 1st, 2022. University of Wurzburg, Germany
Read more at the source #DrGPCR #GPCR #IndustryNews
- Dr. Ross Bathgate becomes Scientific co-founder of LASEREDD Therapeutics
that I’m starting a new position as Scientific co-founder LASEREDD Therapeutics" Ross Bathgate Read more
- ShouTi Pharma CEO Dr. Raymond Stevens was interviewed by Moira Gunn of the NPR TechNation podcast
April 2022 Read more at the source #DrGPCR #GPCR #IndustryNews
- 📰 GPCR Weekly News, May 20 to 26, 2024
Stay tuned for more details, and be ready to register in July 2024. Dr. drinking GRK5 is required for adipocyte differentiation through ERK activation GPCR Binders, Drugs, and more the plasma membrane and suppresses the Saccharomyces cerevisiae mating pathway Reviews, GPCRs, and more
- Inversago Pharma appoints Glenn S. Vraniak as Chief Financial Officer
Vraniak’s career spans more than 20 years of financial and commercial experience in the life sciences Read more at the source #DrGPCR #GPCR #IndustryNews
- Gαs and Gαq/11 protein coupling bias of two AVPR2 mutants (R68W and V162A) that cause nephrogenic di
receptor and consequently activated signaling pathways, and also may shed light on the development of more Read more at the source #DrGPCR #GPCR #IndustryNews
- In vitro assays for the functional characterization of (psychedelic) substances at the serotonin...
More specifically, this review covers assays to monitor the canonical G protein signaling pathway (e.g Read more at the source #DrGPCR #GPCR #IndustryNews 5-HT2AR, GPCR, hallucinogens, in vitro assay, psychedelics
- 📰 GPCR Weekly News, June 19 to 25, 2023
We will be hosting a career panel (more on our panelists soon)! GPCR Binders, Drugs, and more Molecular Characterization of Two Wamide Neuropeptide Signaling Systems Reviews, GPCRs, and more 7TM domain structures of adhesion GPCRs: what's new and what's missing?
- Join Us Today!
Catch up with the latest #GPCR news, start a discussion in the forum, and much more today!
- Meet Peter McNamara, Ph.D., Tectonic’s SVP, Head of Research
Read more at the source #DrGPCR #GPCR #IndustryNews
- 📰 GPCR Weekly News, October 16 to 22, 2023
You can find more information about them on the Live Talks page and mark your calendar HERE. GPCR Newsletter for more insights! transduction at GPCRs: Allosteric activation of the ERK MAPK by β-arrestin GPCR Binders, Drugs, and more
- GPCR Therapeutics welcomes Dr. Ed Brennan as their new Vice President, Head of Clinical Development
He has led teams that have filed more than 10 Investigational New Drug Applications (IND), as well as #biotech #lifesciences #appointment #GPCR #Oncology" Read more at the source #DrGPCR #GPCR #IndustryNews
- Orion and Peptilogics are pursuing AI-driven drug discovery to explore new functional chemical ...
#ai #drugdiscovery #gpcr" Read more at the source #DrGPCR #GPCR #IndustryNews
- Addex Therapeutics CEO Tim Dyer: There is a $4-bil market opportunity in dyskinesia
Read more at the source #DrGPCR #GPCR #IndustryNews
- 📰 GPCR Weekly News, December 4 to 10, 2023
For more information click HERE, don’t miss out on this exclusive opportunity! the G protein-coupled receptor C3aR1 reveals ligand-mediated biased agonism GPCR Binders, Drugs, and more the impact of different detergents and nanodiscs on the A2A adenosine receptor Reviews, GPCRs, and more
- Intermolecular Interactions in G Protein-Coupled Receptor Allosteric Sites at the Membrane Interface
candidates in G protein-coupled receptor (GPCR) drug development by displaying subtype selectivity and more Read more at the source #DrGPCR #GPCR #IndustryNews