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Strategic Partners

Celtarys Research

Filter by topic or event to instantly explore talks, courses, and sessions from across Dr. GPCR University.

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Strategic Project Management for scientists

Lecture 4: Unconventional GPCR Ligands as Drugs

Lecture 2: Drug Disposition in Physiological Tissues as a Therapeutic Variable

Lecture 5: Unique Exploitable GPCR-Ligand Behaviors for Therapeutic Benefit

Lecture 3: The Application of GPCR Ligand Kinetics to Candidate Design

Lecture 1: The Eyes to See- The Importance of Pharmacologic Assays

Lecture 4: Allosteric Modulators: NAMs, PAMs, Special Properties, Methods to quantify the allosteric effect

Lecture 3: Agonists and Efficacy: A New World of GPCR Efficacies / Biased Signaling

Lecture 2: Drug Affinity: Measurement of Antagonism (Binding and Function) / Classifying Antagonists

Lecture 1: GPCR Project Initiation and Design for Discovery of New Molecules

Class 4 - New dimensions of activity: Allosteric modulators and kinetics

Class 3 - Antagonist pharmacology and binding assay analysis

Class 2 - Quantifying agonist pharmacology and biased agonism

Class 1 - Concentration-response analysis: Become a CRC super-user

Class 4 - Characterizing Allosteric Modulators

Class 3 - Characterizing Antagonists

Class 2 - Characterizing Agonists

Class 1 - Fundamentals of Pharmacology

Molecular determinants of ligand efficacy and potency in GPCR signaling

Agonist bias at the Adenosine A1 Receptor: The story of BnOCPA

Neuropeptide recognition and GPCR activation using the expanded receptor repertoire of nematodes – Insights into molecular signatures in vivo

Location bias of GRKs and Arrestins

Gz-Enhanced Signal Transduction assaY (GzESTY) for GPCR deorphanization

Ligand-biased signalling and location bias; two faces of functional selectivity

Accurate Mechanistic Calculation of μ Opioid Receptor Signaling Efficacy - Poster Presentation

Panel Discussion on Publishing in Academia

Roundtable Discussion

The Serotonergic Psychedelic N, N-Dipropyltryptamine Prevents Seizures in a Mouse Model of Fragile X Syndrome

The Good, the Bad, and the Ugly

Using small protein analogs to target challenging GPCRs

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