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GPCR Weekly News

October 22, 2025

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October 2, 2025

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September 18, 2025

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Contributors Articles

Kiyan Afzali

The Perils and Guardrails of Modifying Signalling Proteins in Bioassays

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John Teye Azietaku

Reflections on My PhD Journey: Lessons Learned

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Cam Sinh Lu

Harnessing Deep Mutational Scanning for Enhanced Drug Discovery

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GPCR Industry News

April 17, 2025

Lilly's oral GLP-1, orforglipron, demonstrated statistically significant efficacy results and a safety profile consistent with injectable GLP-1 medicines in successful Phase 3 trial

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April 14, 2025

Pfizer Provides Update on Oral GLP-1 Receptor Agonist Danuglipron

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April 22, 2025

Collaboration between Nostrum Biodiscovery and Celtarys Research: a strategic alliance

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Call for GPCR Papers

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Special Issue on Adhesion GPCRs

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November 1, 2024

Emerging Voices in GPCR Biology in Special Issue of Molecular Pharmacology

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September 27, 2023

opnMe GPCR Route 66+ project

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Adhesion GPCRs

March 25, 2025

Identification of a GPCR as a tip link-independent equilibrioceptor

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March 26, 2025

Spatiotemporal profiling of adhesion G protein-coupled receptors in developing mouse and human pancreas reveals a role for GPR56 in islet development

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February 18, 2025

A force-sensitive adhesion GPCR is required for equilibrioception

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GPCR Activation and Signaling

April 16, 2025

Insights Into the Cellular and Molecular Mechanisms Behind the Antifibrotic Effects of Nerandomilast

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April 18, 2025

Challenging activity and signaling bias in tachykinin NK1 and NK2 receptors by truncated neuropeptides

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April 16, 2025

Intercellular sphingolipid signaling mediates aversive learning in C. elegans

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GPCR Binders, Drugs, and more

April 1, 2025

Identification of anti-resorptive GPCRs by high-content imaging in human osteoclasts

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April 7, 2025

Synthesis and Characterization of Photoswitchable Covalent Ligands for the β2-Adrenoceptor

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April 4, 2025

Minimal Structural Variation of GPR84 Full Agonist Causes Functional Switch to Inverse Agonism

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GPCRs in Cardiology, Endocrinology, and Taste 

April 8, 2025

The DNA repair factor ku80 binds and activates the adhesion receptor ELTD1/ADGRL4

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April 1, 2025

DRD2-Mediated AMPK Ubiquitination Regulates the Occurrence of Hepatic Steatosis

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March 29, 2025

Genomic insights into ORs gene family of G protein-coupled receptors expansion driving omnivorous feeding in Spotted knifejaw (Oplegnathus punctatus)

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GPCRs in Neuroscience 

March 31, 2025

Neurokinin 3 receptor agonist senktide stimulates GnRH release in isolated hypogonadotropic hypogonadism mice

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April 1, 2025

Evidence for Bxy-npr-21 on controlling juveniles' growth and modulating male sexual arousal: from molecules to behaviors

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April 1, 2025

Characterization of Anthozoan-Specific Opsins from a Reef-Building Coral, Acropora tenuis, as Gq-Coupled Opsins

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GPCRs in Oncology and Immunology

April 10, 2025

SIGMAR1 screened by a GPCR-related classifier regulates endoplasmic reticulum stress in bladder cancer

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April 7, 2025

G-protein coupled receptors in metabolic reprogramming and cancer

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April 4, 2025

Unveiling the Role of DPYS: A New Prognostic Biomarker in Sarcoma

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Methods & Updates in GPCR Research 

April 18, 2025

Structural Systems Biology Toolkit (SSBtoolkit): From Molecular Structure to Subcellular Signaling Pathways

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April 7, 2025

Topology-Driven Negative Sampling Enhances Generalizability in Protein-Protein Interaction Prediction

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April 7, 2025

A new approach to psoriasis therapy: photoswitchable A3 adenosine receptor activation

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Reviews, GPCRs, and more

April 18, 2025

Discovery of Feeding Regulatory Peptides and The Importance of Peptide Discovery Research

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April 9, 2025

Where are we now? Biased signalling of Class B G protein-coupled receptor-targeted therapeutics

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April 1, 2025

Opioid Analgesics: Rise and Fall of Ligand Biased Signaling and Future Perspectives in the Quest for the Holy Grail

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Structural and molecular insights into GPCR function

April 17, 2025

Structural dynamics of olfactory receptors: implications for odorant binding and activation mechanisms

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April 15, 2025

Distinct activation mechanisms of CXCR4 and ACKR3 revealed by single-molecule analysis of their conformational landscapes

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April 3, 2025

Proton perception and activation of a proton-sensing GPCR

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