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Fast, clear, live-cell receptor trafficking detection. with TRF plate readers No-wash protocol simplifies workflow Formats available for modified GPCR cell lines TRF detection, which effectively filters out short-lived background signals. This results in high sensitivity and specificity in no-wash, plate-based live-cell assays. pHSense™ Eu Tag-lite® formats.

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Different ligands stabilize distinct receptor states, leading to diverse signaling outcomes. GPCR-Ligand Behaviors for Therapeutic Benefit Terry Kenakin 🔒 Premium Content Watch recording Principles Virtual Café Listen to casual, interactive discussions with experts in the field. Are the masterclasses on-demand or live? Dr. GPCR University offers both on-demand and live classes led by experts in the field.

University Vault: The Ultimate On-Demand GPCR Learning Library Every talk inside the University Vault More Benefits What Scientists Appreciate The most comprehensive library of GPCR knowledge online. Anonymous As a postdoc, my travel budget is limited.

Explore a curated list of GPCR Courses to enhance your knowledge and career. First name Last name Email* Join Our Mailing List Count me in! GPCR Event listings Direct access to members of the GPCR community How do I sign up for a membership Log into your account, go to the Pricing section, and select the option you’d like to choose. You will receive an email with a link to create a new password.

) and the process of characterizing the mechanism of action of ligands to enable the prediction of activity Registrants will learn: Essentials of measuring pharmacologic activity of ligands (affinity, efficacy Application of this knowledge to determine the mechanism of action of new GPCR ligands. Classes will be live from Zoom on Thursdays from 10 am to 11:30 am EST. Sessions will include a 1-hour live lecture plus 30 minutes of Q&A.

Terry Kenakin’s unique course, Development of GPCR Ligands as Therapeutic Drugs , and gain essential elimination 🔹 Safety First – Identifying toxicity risks and drug-drug interactions ⏳ Availability is limited Trial and Plans to Advance Next-Generation Oral Small Molecule PTH1R Agonist Revolutionizing Protein-Ligand Cortical astrocyte activation triggers meningeal nociception and migraine-like pain GPCRs in Oncology and Immunology Spatial analysis of a complete DIPG-infiltrated brainstem reveals novel ligand-receptor

🚀 This workshop will explore how different ligands (compounds) can stabilize unique receptor conformations for better drug design —maximizing efficacy while minimizing side effects The session wraps up with a lively 🧬 Receptor Flexibility : Ligands stabilize different receptor states, creating unique signaling pathways encourages leveraging bias for better therapeutic outcomes. 📌 Receptors are Dynamic Players 🔹 Different ligands BIAS_WORKSHOP_PRINT .pdf Download PDF • 9.11MB BIAS_EXERCISE .pdf Download PDF • 721KB What would you like