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Stay at the Forefront of GPCR Drug Discovery

 

Gain insider methods from the pioneers shaping biased signaling, assay design, and pharmacology—skills you won't find in any textbook or paper.

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⧖ Hours of Expert Training

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◕ New Courses added regularly ​

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Explore the Masterclasses

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Terry Kenakin

Decoding Drug Action
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Terry Kenakin

Seeing is Believing: Assaying Drug Action
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Terry Kenakin

The Allosteric Advantage
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Sam Hoare

CRC Super-User: Your Data Advantage
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Terry Kenakin

The Art of Antagonism
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Sam Hoare

The Agonist Effect: A Story of Bias
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Terry Kenakin

Unlocking Agonist Behavior
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Sam Hoare

The Antagonist's Grip
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Sam Hoare

The Dynamic Allosteric Effect

Learn directly from world leaders in GPCR research

Access exclusive training from the scientists shaping the future of GPCR drug discovery

Dr. Kenneth Jacobson

Dr. Kenneth Jacobson

NIH

Medicinal chemist leading purinergic GPCR drug discovery at the NIH, focused on adenosine and nucleotide receptors and their pharmacology. Recipient of major honors including the ACS Smissman Award and the ASPET Goodman and Gilman Award for Drug Receptor Pharmacology.

Dr. Sam Hoare

Dr. Sam Hoare

Pharmechanics

GPCR signaling & biased agonism expert regularly consulted by top pharma companies for assay design strategies. Pioneer in quantitative pharmacology methods.

Dr. Yamina Berchiche

Dr. Yamina Berchiche

Dr. GPCR & Yamina's Corner

Community builder for scientists with expertise in GPCR project strategy and translational applications.

Dr. Matteo Pavan

Dr. Matteo Pavan

NIH

Computational Chemist Driving Structure-Based Drug Discovery | Molecular Modeling | AI / Machine Learning

Dr. Terry Kenakin

Dr. Terry Kenakin

Terry's Corner

Author of 'A Pharmacology Primer', the definitive GPCR reference used by labs worldwide. Former GSK principal research investigator with 40+ years of experience.

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The GPCR Field Is Advancing Fast – Don't Fall Behind

Stay ahead in drug discovery with insights from the world's top GPCR experts.

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