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Stay at the Forefront of GPCR Drug Discovery

 

Gain insider methods from the pioneers shaping biased signaling, assay design, and pharmacology—skills you won't find in any textbook or paper.

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⧖ Hours of Expert Training

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◕ New Courses added regularly ​

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Explore the Masterclasses

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Terry Kenakin

GPCR Projects: From Idea to Molecule
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Terry Kenakin

GPCR Efficacy: The Biased Signal
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Terry Kenakin

From Body to Benefit: Drug Disposition
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Terry Kenakin

Antagonism: Affinity & Function
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Terry Kenakin

Designing with Time: GPCR Ligand Kinetics
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Terry Kenakin

Unconventional GPCR Ligands
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Terry Kenakin

Assessing Bias: The Practical Approach
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Terry Kenakin

NAMs & PAMs: Quantifying the Impact
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Terry Kenakin

The New Frontier of GPCR Therapeutics

Learn directly from world leaders in GPCR research

Access exclusive training from the scientists shaping the future of GPCR drug discovery

Dr. Kenneth Jacobson

Dr. Kenneth Jacobson

NIH

Medicinal chemist leading purinergic GPCR drug discovery at the NIH, focused on adenosine and nucleotide receptors and their pharmacology. Recipient of major honors including the ACS Smissman Award and the ASPET Goodman and Gilman Award for Drug Receptor Pharmacology.

Dr. Sam Hoare

Dr. Sam Hoare

Pharmechanics

GPCR signaling & biased agonism expert regularly consulted by top pharma companies for assay design strategies. Pioneer in quantitative pharmacology methods.

Dr. Yamina Berchiche

Dr. Yamina Berchiche

Dr. GPCR & Yamina's Corner

Community builder for scientists with expertise in GPCR project strategy and translational applications.

Dr. Matteo Pavan

Dr. Matteo Pavan

NIH

Computational Chemist Driving Structure-Based Drug Discovery | Molecular Modeling | AI / Machine Learning

Dr. Terry Kenakin

Dr. Terry Kenakin

Terry's Corner

Author of 'A Pharmacology Primer', the definitive GPCR reference used by labs worldwide. Former GSK principal research investigator with 40+ years of experience.

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The GPCR Field Is Advancing Fast – Don't Fall Behind

Stay ahead in drug discovery with insights from the world's top GPCR experts.

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