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  • The Truth About GPCR Product Launches: Years in the Making

    Featuring logos from Dr. GPCR and Revvity. Dr. on Dr. GPCR   Dr. GPCR X Revvity Collaboration ⸻ Want more like this? 👉 Join the Dr. GPCR Premium Ecosystem  for behind-the-scenes access to GPCR innovators, exclusive deep-dives, and practical

  • Understanding Enzyme Inhibition In GPCR Discovery Programs

    2025; Nxera Pharma earns $10m milestone from AbbVie neurological deal. 🔍 This Week in Dr. mutated GPCRs. 🎥 Live AMA with Dr. Kenakin — October 30, 12 PM EST Bring your toughest pharmacology questions and join Dr. Read the roundup ➤ Why Dr.

  • Terry’s Corner, Celtarys' Leap, and the $7B GPCR Horizon

    GPCR Updates Learn Pharmacology That Drives Discovery  – From Dr. Explore Dr. This blog post breaks down Dr. GPCR Podcast appearance. Stay curious,   The Dr. GPCR Team

  • Don't miss the chance to be part of the Dr. GPCR Summit 2022!

    ⚠️Mark your calendar for the Dr. GPCR Summit 2022 held between Oct. 10 - 16, it's FREE! Join the #GPCR movement by signing up now! ➡️ https://bit.ly/3cKMXlw #gpcr #drgpcr

  • How System-Level GPCR Thinking Prevents Discovery Failures

    Dr. GPCR Podcast: Chemical Probes for GPCR Imaging with Dr. In this episode, Dr. I will keep Dr. GPCR and the offered resources in my work sphere." GPCR? Donate : https://www.ecosystem.drgpcr.com/donate Dr.

  • Competitive vs Non-Competitive GPCR Antagonists: How to Interpret Pharmacology Data with Confidence

    Dr. GPCR-Based Drug Discovery conference is where the future of GPCR therapies will be defined. Register and join your colleagues in September ➤ Why Dr. GPCR Premium Membership Gives You an Edge In a world filled with noise, Dr. ” - DrGPCR University Course Attendee Get a competitive advantage—Join Dr.

  • 📰 GPCR Weekly News, June 17 to 23, 2024

    Lefkowitz, Howard Rockman for their review G Protein-Coupled Receptors: A Century of Research and Discovery Dr GPCR University We are excited to announce that Dr. The two back-to-back courses are new and specially tailored to the Dr. GPCR Ecosystem and our community. The classes will be online Thursdays from 10 am EST. GPCR Ecosystem

  • Your GPCR Program Decisions Depend on Good Data Interpretation

    Welcome GPCR Fans,   In GPCR-targeted drug discovery, precision isn’t optional—it’s a requirement. That’s why this week at Dr. I wish Dr. field” — Dr. Get The Full Story ➤ Why Dr. GPCR Premium Membership Gives You an Edge Dr.

  • How Collaboration Drives GPCR Discoveries

    GPCR signaling wasn’t linear. It wasn’t clean. For years, the GPCR community wrestled with unreliable antibodies. Why GPCR Collaboration Is Essential for Modern Science Hodson makes the point bluntly: modern GPCR science Together, they push GPCR science faster. this story resonates with your work or curiosity, go deeper. 🎧 Listen to the full conversation with Dr

  • Better GPCR Drug Discovery Decisions Start With Structured Learning

    Dr. GPCR University — Reorganized for Clarity and Speed The Dr. In this session, Dr. An upcoming live Ask-Me-Anything (AMA) with Dr. Kenakin takes place February 26 at 12:00 PM EST. Submit your work today ➤ Why Dr. classified publications, priority event tracking, curated career opportunities, and full access to Dr

  • GPCR Allosteric Modulation: Why Allostery is the Engine of Drug Discovery

    s latest lecture delivers high-impact insight crafted for teams navigating the complex behaviors of GPCR-targeting As Kenakin explains, all GPCR signaling is allosteric , and pretending otherwise introduces risk at every But without understanding how GPCR state changes  influence that affinity—or vice versa—drug discovery Corner  is your trusted, expert-led guide through the evolving landscape of GPCR science. Subscribers gain access to: Weekly lessons by Dr.

  • 📰 GPCR Weekly News

    Hello Readers👋, Get the latest GPCR News more frequently directly in your inbox and in the Ecosystem , and more Life, death and resurrection of plant GPCRs Structural and Molecular Insights into GPCR Function Papers GPCRs: Signal Transduction. GPCR Events, Meetings, and Webinars 2nd GPCR-Targeted Drug Discovery Summit | February 21-23, Boston. Explore Dr. GPCR Ecosystem

  • Targeting Intracellular Allosteric Sites in GPCRs

    Exploring the intracellular allosteric site GPCRs represent one of the largest and most vital families For this reason, GPCRs have been a focus of drug development for decades due to their role in regulating GPCR activity, enabling greater specificity and fewer side effects. allosteric site common in class A and class B GPCRs, particularly in chemokine receptors. Check the original article at https://pubmed.ncbi.nlm.nih.gov/37852356/ #GPCR #DrGPCR #Ecosystem

  • Time is your enemy, GPCRs are your friend

    Come attend this month's virtual café talk to see the awesome work of Dr. Stuart Maudsley on how an aging physiological context affects #GPCR signaling #drgpcr. Register here (FREE) https://www.ecosystem.drgpcr.com/dr-gpcr-virtual-cafe/ #gpcr #drgpcr #virtualcafe

  • How GPCR Spatial Signaling Sparked a Scientific Journey

    Many GPCR scientists trace their origin story back to a single unexpected spark. Not a grand plan. Luck, Leadership & GPCR Signaling Michelle is clear: luck played a role. But so did choice. . 🎧 Listen to the full conversation with Michelle Halls on  The Dr. GPCR Podcast 🔓 Want to go deeper? Join   Dr. GPCR Premium  for exclusive tools, deep dives, and expert access.

  • Why Kinetics Matter More Than Kd in GPCR Drug Discovery

    Kenakin is a masterful teacher and communicator—and a leading expert in our field.” — Dr. GPCR University Course Attendee Dr. GPCR Podcast : From Personal Pain to Scientific Purpose: Alex Serafini’s Journey We sit down with Dr. Secure your spot ➤ Why Dr. Dr.

  • Automated micro-plate-based methods for quantifying GPCR activation

    Excited to hear Dr. Joe Clayton from BioTek Instruments talk about automated micro-plate-based methods for quantifying #GPCR activation. https://www.ecosystem.drgpcr.com/dr-gpcr-virtual-cafe/ #drgpcr #gpcr #virtualcafe

  • Unlocking the Future of Medicine: Advancements in GPCR Research

    protein-coupled receptor function via membrane-interacting intrinsically disordered C-terminal domains Dr We are pleased to announce the scheduled dates for our highly anticipated courses led by Dr. As of July 31st, early-bird registration for our premium Ecosystem members will begin, allowing you to Scientist; Biochemistry, Cellular and Mechanistic Pharmacology; Lead Discovery and Optimization Join the Dr GPCR Ecosystem

  • 📰 GPCR Weekly News, June 10 to 16, 2024

    This week's highlight includes congrats to: Dr. Levitz for their work on Emerging modes of regulation of neuromodulatory G protein-coupled receptors Dr GPCR University We are thrilled to announce that Dr. Dr. GPCR Podcast Tune into the 156th episode of the Dr. GPCR Podcast, featuring Dr. GPCR Ecosystem

  • Assay Volume Control: Your GPCR Drug Discovery Power Lever

    allosteric site on an orphan GPCR. 🔍 This Week in Dr. In this upcoming episode, Dr. In this behind-the-scenes look, Dr. Read the full story➤ Why Dr. I wish Dr.

  • Dr. Simone Promel

    Do you have your ticket for the Dr. GPCR Virtual Cafe? Join us for another virtual cafe talk to hear about the amazing work that Dr. Simone Promel / Promel Lab is doing on adhesion #GPCRs. Register here (free): https://www.ecosystem.drgpcr.com/dr-gpcr-virtual-cafe/ #gpcr #drgpcr #podcast

  • How Breakthroughs Happen: Eric Trinquet on Innovation, Serendipity & GPCRs

    Dr. Frame your strategy, then let the serendipity occur.” — Dr. on Dr. GPCR   Dr. GPCR X Revvity Collaboration ⸻ Want more like this? 👉 Join the Dr. GPCR Premium Ecosystem  for behind-the-scenes access to GPCR innovators, exclusive deep-dives, and practical

  • Quantifying the kinetics of GPCR signaling

    Join us and learn how to quantify your kinetic GPCR signaling from the expert himself: Dr. https://www.ecosystem.drgpcr.com/dr-gpcr-virtual-cafe/ #gpcr #drgpcr #virtualcafe

  • Exciting GPCR Events for Next Year! + GPCR Weekly Rocket Launch ⦿ Oct 28 - Nov 3, 2024

    Get your space suits on, GPCR cadets! up with a series of cosmic GPCR events for the year ahead. Discounted GPCR courses - because who doesn't love a good deal?  From 2025, only Premium Members will have access to Classified GPCR News. Classified GPCR News  Let’s dive into the   Classified GPCR News from October 28th to November 3rd, 2024

  • How Schild Analysis Protects Your Conclusions in GPCR Research

    In this week’s lesson, Dr. Access this week’s key insight ➤ Dr. Dr. 👉 Access this week’s full Premium Edition here ➤ What Members Say “Dr. See you in the Ecosystem, Dr. GPCR Team

  • Targeting GPCRs in the CNS: Advances in Drug Discovery Strategies

    The central role of GPCRs in Neurological Disorders GPCRs are the largest family of membrane receptors Over 30% of FDA-approved drugs target GPCRs, with many targeting CNS located GPCRs. GPCR Structure, Activation, and Signaling Pathways in the Brain An understanding of GPCR structure is GPCR signaling: (A) an orthosteric ligand (orange) binds an inactive GPCR, the β2 adrenergic receptor Emerging GPCR Therapeutic Targets in CNS Drug Discovery GPCRs have been studied for decades, but there

  • Enzyme Inhibition Pharmacology: The Hidden Gatekeepers of GPCR Drug Discovery

    Before your GPCR ligand ever meets its receptor, it meets the enzymes that determine whether it survives Even the most elegant GPCR ligand can fail if it never reaches its receptor. 🎥  Coming Soon: Live AMA with Dr. Terry Kenakin This Month’s Live AMA — October 30 at 12 PM EST Join Dr. Monthly AMAs  where you can challenge Dr. Kenakin with your own enzyme or GPCR interaction puzzles.

  • Join Us Today!

    🌐Dr. GPCR Ecosystem is under construction and dozens of your colleagues are enjoying its benefits! Catch up with the latest #GPCR news, start a discussion in the forum, and much more today! Join the #GPCR movement by becoming a site member for FREE! ➡️ https://www.ecosystem.drgpcr.com/ #gpcr #drgpcr

  • From Failed Experiments to Predictive GPCR Models

    Watch Episode 175 From failed assays to breakthroughs in GPCR modeling , Dr. At that point, very few GPCR crystal structures had been determined. Hear the full conversation with Jens Carlsson 🎧 Catch the full episode on the Dr. GPCR Podcast 💡 Stay curious. Stay connected. Looking for more insights like this? The Dr. GPCR Premium Ecosystem  gives you exclusive access to thought leaders, technical resources, and deep-dive

  • GPCR Drug Discovery at Discovery on Target: Why This Track Is About More Than Receptors

    Join Dr. . 🌐 Why Dr. GPCR Is in This Conversation At Dr. Kenakin Himself If you’re part of the Dr. . ✨ Be part of Dr. GPCR’s nonprofit mission to connect and empower the global GPCR ecosystem. 📅 September 24, 2025 📍 Pressed

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