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CFTX-1554 is being developed as a non-opioid approach to the treatment of neuropathic pain, a debilitating

Terry Kenakin , a veteran pharmacologist with over 40 years of industry experience. If you're just beginning your pharmacology journey… This is the lesson that will connect the dots. You’ll leave with the language, logic, and big-picture view that underpins all future learning in pharmacology

Gunnar Schulte for his study on the International Union of Basic and Clinical Pharmacology. Jianming Han, Tao Che for their analysis of GPCR-G protein selectivity revealed by structural pharmacology Here’s a sneak peek at what you can expect: Principles of Pharmacology in Drug Discovery I - Techniques Principles of Pharmacology in Drug Discovery II - Advanced Methods for the Optimization of Candidate 2026 GPCR Jobs HIGHLIGHT Principal Scientist, In vitro pharmacology NEW Senior Scientist - Discovery

This new learning hub is your go-to space to revisit core pharmacology concepts, master new ones, and Explore Terry's Corner Better decisions start with better pharmacology.

I We are diving into the second class of our Principles of Pharmacology I course with enthusiasm and you missed out on enrolling in this one, worry not – a spot is reserved just for you in Principles of Pharmacology Seize this opportunity to enhance your expertise and proficiency in pharmacology! Modules: October 31st : The Eyes to See- The Importance of Pharmacologic Assays. Emerging Voices in GPCR Biology in Special Issue of Molecular Pharmacology GPCR Events, Meetings, and

Nb39: This nanobody was identified for the μ-opioid receptor (μOR) and also increased the affinity of Annual review of pharmacology and toxicology, 57, 19–37. https://doi.org/10.1146/annurev-pharmtox-010716

Thrilling beginning to Principles of Pharmacology I We are excited to announce the start of our Principles of Pharmacology I course! Don’t miss this opportunity to advance your knowledge and skills in pharmacology! Modules: October 31st : The Eyes to See- The Importance of Pharmacologic Assays. Emerging Voices in GPCR Biology in Special Issue of Molecular Pharmacology GPCR Events, Meetings, and

Pharmacology isn’t only about ligands, receptors, and downstream G protein signaling—it’s also about The Hidden Lever in GPCR Research In GPCR pharmacology, the conversation often centers on ligand properties—affinity Clarify whether observed effects reflect true pharmacology or assay artifacts . From Bench Insight to Strategic Advantage Terry Kenakin’s decades of pharmacology leadership converge A growing on-demand library  of expert pharmacology lessons to revisit anytime.

Administration (FDA) for use in adults for the management of acute pain severe enough to require an intravenous opioid

and Daniel Isom  for their research on Advances in yeast synthetic biology for human GPCR biology and pharmacology Materials Access to the private group Certificate of participation Learn the essentials: Measuring the pharmacologic genetic disease Advances in yeast synthetic biology for human G protein-coupled receptor biology and pharmacology 7, 2024 | 16th Annual PEGS Europe   July 12 - 17, 2026 | 20th World Congress of Basic and Clinical Pharmacology

Andrew Tobin for an incredible week filled with prestigious events, including receiving the British Pharmacological and TPD Structural Biology Platforms GPCR Events, Meetings, and Webinars December 10 - 12, 2024 | Pharmacology | BIO International Convention 2025 July 12 - 17, 2026 | 20th World Congress of Basic and Clinical Pharmacology Principal Scientist, Medicinal Chemistry PhD fellowship in GPCR mechanosensing Senior Scientist, GPCR Pharmacology Research Associate - Professor Graeme Milligan Postdoc in Molecular Pharmacology - The Hauser Group

Every Thursday at 10 AM EST: Principles of Pharmacology I October 3, 10, 17, 24 (four sessions) Topics : Pharmacologic activity measurement, mechanisms of action, and GPCR discovery strategies. Principles of Pharmacology II October 31, November 7, 14, 21, December 5 (five sessions) (we skipped The Principles of Pharmacology I & II BUNDLE is your key to mastering the field. GPCR Jobs HIGHLIGHT Research Associate - Professor Graeme Milligan HIGHLIGHT Postdoc in Molecular Pharmacology

Allosteric GPCR Binding Sites and Their Ligandability Potential Today, we started the Principles of Pharmacology Emerging Voices in GPCR Biology in Special Issue of Molecular Pharmacology GPCR Events, Meetings, and GPCRs-Targeted Drug Discovery Summit Europe July 12 - 17, 2026 | 20th World Congress of Basic and Clinical Pharmacology I Cell Biology - Tectonic Therapeutic PhD fellowship in GPCR mechanosensing Senior Scientist, GPCR Pharmacology Research Associate - Professor Graeme Milligan Postdoc in Molecular Pharmacology - The Hauser Group

GPCR University workshop on Advanced Data Analysis for GPCR Pharmacology, led by the esteemed Dr. GPCR Matchmaking Read Mark's job spotlight article for a Principal Scientist in In Vitro Pharmacology Mark recently discussed this exciting opportunity with Beth Fleck, Director of In Vitro Pharmacology 2026 GPCR Jobs HIGHLIGHT Principal Scientist, In vitro pharmacology NEW Senior Scientist - Receptor Pharmacology NEW PostDoctoral Scientist Senior Research Associate/Associate Scientist, Protein Science

Tomas , Kyle Sloop , et al. for their outstanding study on Class B1 GPCRs: insights into multireceptor pharmacology November 26 - 28, 2024 | GPCRs-Targeted Drug Discovery Summit Europe NEW December 10 - 12, 2024 | Pharmacology | BIO International Convention 2025 July 12 - 17, 2026 | 20th World Congress of Basic and Clinical Pharmacology I Cell Biology - Tectonic Therapeutic PhD fellowship in GPCR mechanosensing Senior Scientist, GPCR Pharmacology Research Associate - Professor Graeme Milligan Postdoc in Molecular Pharmacology - The Hauser Group

That’s not pharmacology. That’s kinetics. It’s a shift in how expert drug hunters see pharmacology. Unlock “Kinetics: Advanced Applications” Only in Terry’s Corner Why Terry’s Corner Most pharmacology engagement opportunities  through AMAs and topic suggestions Practical insights  distilled from decades of pharmacology

Highlights: Congratulations to our amazing Board Member JoAnn Trejo for being elected to the British Pharmacological Paltusotine for Adult Patients with Acromegaly GPCR Events, Meetings, and Webinars December 10 - 12, 2024 | Pharmacology | BIO International Convention 2025 July 12 - 17, 2026 | 20th World Congress of Basic and Clinical Pharmacology Principal Scientist, Medicinal Chemistry PhD fellowship in GPCR mechanosensing Senior Scientist, GPCR Pharmacology Research Associate - Professor Graeme Milligan Postdoc in Molecular Pharmacology - The Hauser Group

affect signaling pathways in class A dopamine receptors like D1/D2 and D1/D3, which exhibit distinct pharmacological Pharmacol Rev, 2016. 68 (4): p. 954-1013. 6.          Mol Pharmacol, 2012. 81 (3): p. 309-18. 9.         

One of its first pillars, Terry’s Pharmacology Corner , led by Dr. Through Terry’s Pharmacology Corner , he shares decades of expertise in an accessible, on-demand format Terry Kenakin , a pioneer who helped shape modern pharmacology and deepen our understanding of GPCR function Related Links 🔗 Explore Terry’s Pharmacology Corner → TerryKenakin.com 📧 Connect with us →   Hello@

GPCR University course, 'Applying Pharmacology to Drug Discovery,' led by Dr. and more Nanobody-Mediated Dualsteric Engagement of the Angiotensin Receptor Broadens Biased Ligand Pharmacology Pharmacological characterization and radiolabeling of VUF15485, a high-affinity small-molecule agonist Spring in Barcelona GPCR Events, Meetings, and Webinars February 20, 2024 | Career Opportunities in Pharmacology 2026 GPCR Jobs NEW Research Fellow NEW  Postdoctoral Fellow – Molecular Pharmacology of Feeding Behavior

Gunnar Schulte, Lukas Grätz, Pawel Kozielewicz, et al. for their study on Frizzleds act as dynamic pharmacological Samuel Hoare on Advanced data analysis for GPCR pharmacology, which will be held on Thursdays between , 2024 | 11th Adhesion GPCR Workshop July 12 - 17, 2026 | 20th World Congress of Basic and Clinical Pharmacology 2026 GPCR Jobs NEW Principal Scientist, In vitro pharmacology Senior Associate Scientist - Global Research Research Unit Postdoctoral Scholar – Synaptic physiology, optical imaging, substance use disorder, pharmacology

It will bridge foundational receptor theory with today’s most pressing pharmacological questions, from gives you timeless and timely tools to improve selectivity, model efficacy, and design smarter GPCR pharmacology

Kenakin and Hoare on '   Applying Pharmacology to Drug Discovery ' and ' Advanced Data Analysis for GPCR Pharmacology .' Dates:  September 5 to 26, 2024 What You’ll Learn during the four sessions: How to measure pharmacologic s dive into the   Classified GPCR News  from August 5th to 11th, 2024 GPCR Activation and Signaling Pharmacological 7, 2024 | 16th Annual PEGS Europe   July 12 - 17, 2026 | 20th World Congress of Basic and Clinical Pharmacology

, 2024 | 11th Adhesion GPCR Workshop July 12 - 17, 2026 | 20th World Congress of Basic and Clinical Pharmacology 2026 GPCR Jobs NEW Scientist; Biochemistry, Cellular and Mechanistic Pharmacology; Lead Discovery and Director GPCR Drug Discovery Biologist HIGHLIGHT Principal Scientist, In vitro pharmacology Post-Doctoral Scientist- Molecular Pharmacology (FDE) Research Assistant Senior Scientist - Receptor Pharmacology

Terry Kenakin's "Applying Pharmacology to Drug Discovery" course at Dr. pathways and two distinct high-affinity sites for succinate in succinate receptor 1/GPR91 Specific pharmacological , 2024 | 11th Adhesion GPCR Workshop July 12 - 17, 2026 | 20th World Congress of Basic and Clinical Pharmacology Research Unit Postdoctoral Scholar – Synaptic physiology, optical imaging, substance use disorder, pharmacology Research Fellow Postdoctoral Fellow – Molecular Pharmacology of Feeding Behavior Director of Laboratory

This opens up a new pharmacological space—and a reason to revisit “failed” targets with fresh eyes. Persistent binding isn’t just about longer half-lives—it’s about smarter pharmacology. ahead with The Kenakin Brief  — a concise, science‑first email update with the latest insights in GPCR pharmacology

studies, it facilitates the structural context necessary to map receptor localization in defined states (pharmacological Br J Pharmacol. 2023 Dec 12. doi: 10.1111/bph.16297. 

Course Schedule and Details Every Thursday at 10 am EST Principles of Pharmacology in Drug Discovery Candidate Molecules Dates: September 5th to 26th, 2024 Registrants will learn: Essentials of measuring pharmacologic Principles of Pharmacology in Drug Discovery II - Advanced Methods for the Optimization of Candidate , 2024 | 11th Adhesion GPCR Workshop July 12 - 17, 2026 | 20th World Congress of Basic and Clinical Pharmacology Discovery Biotherapeutics Post-Doctoral Fellow/Trainee Scientist; Biochemistry, Cellular and Mechanistic Pharmacology

What emerged wasn’t just another pharmacology group — it became a collaborative engine for GPCR discovery Turning Silos into Systems The early 2000s were not kind to exploratory pharmacology. Why This Matters GPCR research demands integration — pharmacology, structural biology, signaling pathways

In this eye-opening module, Terry Kenakin explores a concept that could change how you interpret pharmacological