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MRGPRs), a subfamily of GPCRs, are largely expressed by sensory neurons and known to modulate itch and pain

and Taste Orphan GPCR GPRC5C Facilitates Angiotensin II-Induced Smooth Muscle Contraction GPCRs in Neuroscience

Patients With Multiple Myeloma and Lymphoma Undergoing Chimeric Antigen Receptor T-Cell Therapy GPCRs in Neuroscience

Photoaffinity Probe that Captures the Active Conformation of the Cannabinoid CB2 Receptor GPCRs in Neuroscience

β-adrenergic receptor signaling mediated by β-arrestins and its potential role in heart failure GPCRs in Neuroscience

GPCRs in Neuroscience CGRP physiology, pharmacology, and therapeutic targets: Migraine and beyond.

ENDO 2024 Highlighting Therapeutic Potential of its GPCR Drug Discovery Platform GPCRs and Emotional Pain

Interactions Using BRET Biosensors Reveals Functional Differences among Receptor Paralogs GPCRs in Neuroscience

Neurosci. 2, 727–733. https://doi.org/10.1038/35094577.

Eur J of Neuroscience   2017 , 45  (1), 2–19. https://doi.org/10.1111/ejn.13390 . (3)         Borovac Neuroscience Letters   2001 , 302  (1), 5–8. https://doi.org/10.1016/S0304-3940(01)01568-3 . (15)      An Order of Magnitude Faster DNA-PAINT Imaging by Optimized Sequence Design and Buffer Conditions.

In addition to its function about weight gain and appetite control mechanisms of MC3R, recent studies In this review paper, we aimed to point out the importance of the MC3R regulations in three main concepts

and Gαi1, respectively (Figure 2B), as well as different coupling preferences between specific Gβγ pairs ACS Chem Neurosci. 2010;1(6):435-49. 3.            Kola I, Landis J. delta opioid receptors is an endogenous mechanism and therapeutic target for relief from inflammatory pain

Some studies have also reported GPR84 involvement in pain, atherosclerosis, and even metabolic disorders

receptor type 2 (CB2R) has emerged as a compelling target across inflammation, immune modulation, and pain

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transcriptional responses and contribute to physiological processes such as meiosis in ovarian follicles and pain

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