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- pharmacology at your fingertips terrys corner launches | Dr. GPCR Ecosystem
Flash News → pharmacology at your fingertips terrys corner launches Published on July 4, 2025 Category GPCR Weekly News Stronger pharmacology drives smarter decisions in GPCR discovery. GPCR Weekly: ♦️ Yamina’s Corner—GPCR consulting to de-risk and accelerate your pipeline ♦️ Celtarys’ validated TR-FRET assay for CB1/CB2 ♦️ Chemokine-GPCR selectivity decoded ♦️ PTH1R structures reveal https://www.ecosystem.drgpcr.com/post/pharmacology-at-your-fingertips-terry-s-corner-launches #DrGPCR #GPCR
- Did you know registrations are already open for all our 2025 Dr.GPCR University Courses? Check out what you can learn this year from the master, Dr. Terry Kenakin 😉and save your spot soon! Remember Premium Members get a 25% discount 🙌 ✳️Click here and start your next learning experience https://www.ecosystem.drgpcr.com/gpcr-courses #gpcr #drgpcr | Dr. GPCR Ecosystem
25% discount 🙌 ✳️Click here and start your next learning experience https://www.ecosystem.drgpcr.com/gpcr-courses #gpcr #drgpcr Published on February 18, 2025 Category GPCR Weekly News Did you know registrations are discount 🙌 ✳️ Click here and start your next learning experience https://www.ecosystem.drgpcr.com/gpcr-courses #gpcr #drgpcr Previous Next Recent Articles
- New insights into FPR2 signaling! GRK5 drives FPR2 endocytosis, but β-arrestin plays a pivotal role in postendocytic trafficking, plasma membrane recycling, and regulating signal transduction. Check out the latest GPCR news in the Ecosystem today! You’ll need to register but don’t worry, it’s Free! ➡️https://www.ecosystem.drgpcr.com/receptor-activation-and-signaling/grk5-regulates-endocytosis-of-fpr2-independent-of-%CE%B2-arrestins #gpcr #drgpcr | Dr. GPCR Ecosystem
Check out the latest GPCR news in the Ecosystem today! receptor-activation-and-signaling/grk5-regulates-endocytosis-of-fpr2-independent-of-%CE%B2-arrestins #gpcr #drgpcr Published on January 30, 2025 Category GPCR Weekly News New insights into FPR2 signaling! Check out the latest GPCR news in the Ecosystem today! receptor-activation-and-signaling/grk5-regulates-endocytosis-of-fpr2-independent-of-%CE%B2-arrestins #gpcr
- Check out the new optical BRET-based biosensor, Gαi bONE-GO! In neuronal cell lines, the use of Gαi bONE-GO revealed that several natural opioid neuropeptides act as partial agonists, contrary to their previous characterization as full agonists. Check out the latest GPCR news in the Ecosystem today! You’ll need to register but don’t worry, it’s Free! ➡️https://buff.ly/e6gAlBv #gpcr#drgpcr | Dr. GPCR Ecosystem
Check out the latest GPCR news in the Ecosystem today! ➡️https://buff.ly/e6gAlBv #gpcr#drgpcr Published on April 21, 2025 Category GPCR Weekly News Check out Check out the latest GPCR news in the Ecosystem today! ➡️ https:// buff.ly/e6gAlBv #gpcr#drgpcr Previous Next Recent Articles
- Xylazine, Fentanyl, and the Fight for Breath with Catherine Demery | Dr. GPCR Ecosystem
academia, building translational experiments, and using real-world data to drive impactful science in the GPCR GPCR Podcast Strategic Partners Xylazine, Fentanyl, and the Fight for Breath with Catherine Demery Two How GPCR pharmacology connects molecular insights to real-world interventions. GPCR ecosystem , GPCR training program , GPCR podcast , opioid pharmacology , xylazine research , mu GPCR Podcast? Leave a Review.
- Jacob Lee & Jin Choe | Dr. GPCR Ecosystem
GPCR Podcast Strategic Partners Jacob Lee & Jin Choe About this episode In this special episode of the GPCR Ecosystem Jin Choe on LinkedIn Jin Choe on Dr. GPCR Ecosystem Enjoying the Dr. GPCR Podcast? Review on Apple Podcasts ★ Rate on Spotify ✉️ Send feedback to the team Recent Podcast Articles How GPCR Collaboration Built an Innovation Engine From Pipettes to Platforms: The Evolution of GPCR Research How GPCR Spatial Signaling Sparked a Scientific Journey Thanks for listening to this podcast episode
- Dr. Paul Insel | Dr. GPCR Ecosystem
GPCR Podcast Strategic Partners Dr. Paul Insel About this episode In 1975, Dr. GPCR Ecosystem Enjoying the Dr. GPCR Podcast? Leave a Review. Review on Apple Podcasts ★ Rate on Spotify ✉️ Send feedback to the team Recent Podcast Articles How GPCR Collaboration Built an Innovation Engine From Pipettes to Platforms: The Evolution of GPCR Research How GPCR Spatial Signaling Sparked a Scientific Journey Thanks for listening to this podcast episode
- Annabelle Milner | Dr. GPCR Ecosystem
GPCR Podcast Strategic Partners Annabelle Milner About Annabelle Milner Annabelle completed her undergraduate Annabelle’s Ph.D. work focuses on microbial-derived metabolites that signal through GPCRs expressed in GPCR Enjoying the Dr. GPCR Podcast? Leave a Review. Collaboration Built an Innovation Engine From Pipettes to Platforms: The Evolution of GPCR Research How GPCR Spatial Signaling Sparked a Scientific Journey Thanks for listening to this podcast episode
- Dr. Ilana Kotliar | Dr. GPCR Ecosystem
GPCR Podcast Strategic Partners Dr. Ilana Kotliar About Dr. Ilana uses chemical biology-based methods to study the regulation and protein-protein interactions of GPCRs GPCR Enjoying the Dr. GPCR Podcast? Leave a Review. Collaboration Built an Innovation Engine From Pipettes to Platforms: The Evolution of GPCR Research How GPCR Spatial Signaling Sparked a Scientific Journey Thanks for listening to this podcast episode
- Dr. Alexander S. Hauser | Dr. GPCR Ecosystem
GPCR Podcast Strategic Partners Dr. Alexander S. Hauser About Dr. Alexander S. Award” for his work on GPCRs. Dr. Alexander S. GPCR Ecosystem Enjoying the Dr. GPCR Podcast? Leave a Review. Collaboration Built an Innovation Engine From Pipettes to Platforms: The Evolution of GPCR Research How GPCR Spatial Signaling Sparked a Scientific Journey Thanks for listening to this podcast episode
- ep 175 with jens carlsson release picture | Dr. GPCR Ecosystem
Discover how embracing failure turned frustration into a breakthrough career designing GPCR experiments GPCR Podcast. Home → Flash News → ep 175 with jens carlsson release picture Model. Predict. GPCR Podcast What if a failed experiment became the best thing that ever happened to your career? Computational Biochemistry at Uppsala University , where his lab uses structure-based modeling to predict GPCR-ligand GPCR Podcast : https://www.ecosystem.drgpcr.com/dr-gpcr-podcast/model-predict-discover #DrGPCR #GPCR
- Dr. Kevin Pfleger | Dr. GPCR Ecosystem
GPCR Podcast Strategic Partners Dr. Kevin Pfleger About this episode Dr. I sat down with Kevin to chat about GPCRs, pharmacology, and his contributions to the field in both the GPCR Ecosystem Enjoying the Dr. GPCR Podcast? Leave a Review. Collaboration Built an Innovation Engine From Pipettes to Platforms: The Evolution of GPCR Research How GPCR Spatial Signaling Sparked a Scientific Journey Thanks for listening to this podcast episode
- Biochemical Mechanisms Underlying Location Bias in GPCR Signaling
Retreat 2023 About Program Registration Logo Contest Committee Sponsors GPCR Retreat Program < Back to schedule Biochemical Mechanisms Underlying Location Bias in GPCR Signaling Date & Time Saturday, November His lab is also interested in identifying novel signal transduction mechanisms of GPCRs, such as the GPCR Previous Event Next Event Great Lakes GPCR Retreat and Club des Récepteurs à Sept Domaines Transmembranaires 22nd GPCR Retreat Sponsored by
- Dr. Arun Shukla | Dr. GPCR Ecosystem
GPCR Podcast Strategic Partners Dr. Arun first started working on GPCRs and their structural characterization at the Max Planck Institute Fascinated by GPCRs he wrote to Dr. GPCR Ecosystem Enjoying the Dr. GPCR Podcast? Leave a Review. Collaboration Built an Innovation Engine From Pipettes to Platforms: The Evolution of GPCR Research
- Dr. Josephine (Pina) Cardarelli | Dr. GPCR Ecosystem
GPCR Podcast Strategic Partners Dr. Josephine (Pina) Cardarelli About Dr. Pina Cardarelli, CSO for GPCR Therapeutics Inc., based in South Korea, has recently been named President of GPCR Therapeutics, USA, a newly incorporated Biotechnology company in the Bay Area. Additionally, they have a library of target GPCR heteromers for Oncology. Dr. GPCR Ecosystem Enjoying the Dr. GPCR Podcast? Leave a Review.
- Dr. J. Silvio Gutkind | Dr. GPCR Ecosystem
GPCR Podcast Strategic Partners Dr. J. Silvio Gutkind About this episode Dr. J. GPCR Ecosystem Enjoying the Dr. GPCR Podcast? Leave a Review. Review on Apple Podcasts ★ Rate on Spotify ✉️ Send feedback to the team Recent Podcast Articles How GPCR Collaboration Built an Innovation Engine From Pipettes to Platforms: The Evolution of GPCR Research How GPCR Spatial Signaling Sparked a Scientific Journey Thanks for listening to this podcast episode
- Steve McCloskey | Dr. GPCR Ecosystem
GPCR Podcast Strategic Partners Steve McCloskey About Steve McCloskey Steve McCloskey is an Alumni from GPCR Ecosystem Enjoying the Dr. GPCR Podcast? Leave a Review. Review on Apple Podcasts ★ Rate on Spotify ✉️ Send feedback to the team Recent Podcast Articles How GPCR Collaboration Built an Innovation Engine From Pipettes to Platforms: The Evolution of GPCR Research How GPCR Spatial Signaling Sparked a Scientific Journey Thanks for listening to this podcast episode
- Dr. Paul Insel | Dr. GPCR Ecosystem
GPCR Podcast Strategic Partners Dr. Paul Insel About this episode Dr. GPCR Ecosystem Enjoying the Dr. GPCR Podcast? Leave a Review. Review on Apple Podcasts ★ Rate on Spotify ✉️ Send feedback to the team Recent Podcast Articles How GPCR Collaboration Built an Innovation Engine From Pipettes to Platforms: The Evolution of GPCR Research How GPCR Spatial Signaling Sparked a Scientific Journey Thanks for listening to this podcast episode
- How do GRK-specific phosphorylation barcodes influence β-arrestin binding to GPCRs? New cryo-EM structures from Chen et al. (Nature, 2025) reveal that β-arrestin1 and β-arrestin2 form distinct complexes with ACKR3 depending on whether it's phosphorylated by GRK2 or GRK5, shaping arrestin conformation, complex stability, and engagement mode. Surprisingly, arrestin’s finger loop didn’t dive into the receptor core. Instead, it latched onto the micelle surface, breaking canonical expectations. Also, β-arrestin2 lacks a membrane anchor, making it more dynamic — a potential clue to its functional specialization. These findings underscore how barcode location + arrestin isoform = unique signaling outcomes. open book Read the full study: Inside Out: Mapping GPCRs from Membrane Codes to Market Moves #GPCRs #Arrestin #ACKR3 #GRKs #CryoEM #StructuralBiology #SignalingBias #Phosphorylation #DrGPCR | Dr. GPCR Ecosystem
Home → Flash News → How do GRK-specific phosphorylation barcodes influence β-arrestin binding to GPCRs + arrestin isoform = unique signaling outcomes. open book Read the full study: Inside Out: Mapping GPCRs from Membrane Codes to Market Moves #GPCRs #Arrestin #ACKR3 #GRKs #CryoEM #StructuralBiology #SignalingBias barcodes influence β-arrestin binding to GPCRs? Read the full study: Inside Out: Mapping GPCRs from Membrane Codes to Market Moves #GPCRs #Arrestin #
- Dr. Mark Connor | Dr. GPCR Ecosystem
GPCR Podcast Strategic Partners Dr. Mark Connor About Dr. Focus on study of drugs and toxins on GPCR (opioid, cannabinoid receptor) and ion channel (K, Ca, TRP GPCR Ecosystem Enjoying the Dr. GPCR Podcast? Leave a Review. Collaboration Built an Innovation Engine From Pipettes to Platforms: The Evolution of GPCR Research How GPCR Spatial Signaling Sparked a Scientific Journey Thanks for listening to this podcast episode
- The Role of Quantitative Sciences in GPCRs with Dr. Nagarajan Vaidehi | Dr. GPCR Ecosystem
GPCR Podcast Strategic Partners The Role of Quantitative Sciences in GPCRs with Dr. GPCR Enjoying the Dr. GPCR Podcast? Leave a Review. Review on Apple Podcasts ★ Rate on Spotify ✉️ Send feedback to the team Recent Podcast Articles How GPCR Collaboration Built an Innovation Engine From Pipettes to Platforms: The Evolution of GPCR Research How GPCR Spatial Signaling Sparked a Scientific Journey Thanks for listening to this podcast episode
- Dr. Amynah Pradhan | Dr. GPCR Ecosystem
GPCR Podcast Strategic Partners Dr. Amynah Pradhan About this episode In this episode of the Dr. GPCR podcast , we meet with Dr. Amynah Pradhan. GPCR Ecosystem Enjoying the Dr. GPCR Podcast? Leave a Review. Collaboration Built an Innovation Engine From Pipettes to Platforms: The Evolution of GPCR Research How GPCR Spatial Signaling Sparked a Scientific Journey Thanks for listening to this podcast episode
- Dr. Kenneth A. Jacobson | Dr. GPCR Ecosystem
GPCR Podcast Strategic Partners Dr. Kenneth A. Jacobson About Dr. Kenneth A. Jacobson Kenneth A. GPCR Enjoying the Dr. GPCR Podcast? Leave a Review. Review on Apple Podcasts ★ Rate on Spotify ✉️ Send feedback to the team Recent Podcast Articles How GPCR Collaboration Built an Innovation Engine From Pipettes to Platforms: The Evolution of GPCR Research How GPCR Spatial Signaling Sparked a Scientific Journey Thanks for listening to this podcast episode
- Dr. Graeme Milligan | Dr. GPCR Ecosystem
GPCR Podcast Strategic Partners Dr. Graeme Milligan About Dr. main research group centers on the function, structure, and regulation of G protein-coupled receptors (GPCRs GPCR Ecosystem Enjoying the Dr. GPCR Podcast? Leave a Review. Collaboration Built an Innovation Engine From Pipettes to Platforms: The Evolution of GPCR Research How GPCR Spatial Signaling Sparked a Scientific Journey Thanks for listening to this podcast episode
- Dr. Nyla Naim, Dr. Michael Lemieux & Dr. Jason Nasse | Dr. GPCR Ecosystem
GPCR Podcast Strategic Partners Dr. Nyla Naim, Dr. Michael Lemieux & Dr. Jason Nasse About Dr. GPCR Ecosystem About Dr. GPCR Ecosystem About Dr. Jason Nasse Dr. GPCR Ecosystem Enjoying the Dr. GPCR Podcast? Leave a Review. Collaboration Built an Innovation Engine From Pipettes to Platforms: The Evolution of GPCR Research
- Retreat | Dr. GPCR Ecosystem
GPCR Retreat — an immersive event uniting scientists, biotech leaders, and innovators in GPCR research GPCR Retreat - Coming Soon - Please tell us your thoughts about scientific gatherings by filling out
- Dr. Richard Premont | Dr. GPCR Ecosystem
GPCR Podcast Strategic Partners Dr. Richard Premont About Dr. Richard Premont "Dr. to the identification of GRK5 and continued focus on GRKs (particularly GRKs 4,5,6) and arrestins as GPCR an independent faculty position at Duke in Gastroenterology, where he remained until 2018 studying GPCRs GPCR Enjoying the Dr. GPCR Podcast? Leave a Review. Collaboration Built an Innovation Engine From Pipettes to Platforms: The Evolution of GPCR Research
- Dr. Richard Premont | Dr. GPCR Ecosystem
GPCR Podcast Strategic Partners Dr. Richard Premont About Dr. Richard Premont "Dr. to the identification of GRK5 and continued focus on GRKs (particularly GRKs 4,5,6) and arrestins as GPCR an independent faculty position at Duke in Gastroenterology, where he remained until 2018 studying GPCRs GPCR Enjoying the Dr. GPCR Podcast? Leave a Review. Collaboration Built an Innovation Engine From Pipettes to Platforms: The Evolution of GPCR Research
- Dr. Richard Premont | Dr. GPCR Ecosystem
GPCR Podcast Strategic Partners Dr. Richard Premont About Dr. Richard Premont "Dr. to the identification of GRK5 and continued focus on GRKs (particularly GRKs 4,5,6) and arrestins as GPCR an independent faculty position at Duke in Gastroenterology, where he remained until 2018 studying GPCRs GPCR Enjoying the Dr. GPCR Podcast? Leave a Review. Collaboration Built an Innovation Engine From Pipettes to Platforms: The Evolution of GPCR Research
- Dr. Richard Premont | Dr. GPCR Ecosystem
GPCR Podcast Strategic Partners Dr. Richard Premont About Dr. Richard Premont "Dr. to the identification of GRK5 and continued focus on GRKs (particularly GRKs 4,5,6) and arrestins as GPCR an independent faculty position at Duke in Gastroenterology, where he remained until 2018 studying GPCRs GPCR Enjoying the Dr. GPCR Podcast? Leave a Review. Collaboration Built an Innovation Engine From Pipettes to Platforms: The Evolution of GPCR Research
