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Results found for "Druggable GPCR"
- How do GPCRs sense pH changes? New cryo-EM structures of GPR4 and GPR68 reveal how extracellular histidines act as proton sensors-trigger activation and biased G protein coupling! Did you know that we work hard to bring you the most recent GPCR News, weekly? Catch up today in the Ecosystem using your free site membership! ➡️https://www.ecosystem.drgpcr.com/structural-and-molecular-insights-into-gpcr-function/structural-basis-and-biased-signaling-of-proton-sensation-by-gpcrs-mediated-by-extracellular-histidine-rearrangement #gpcr#drgpcr | Dr. GPCR Ecosystem
Home → Flash News → How do GPCRs sense pH changes? Did you know that we work hard to bring you the most recent GPCR News, weekly? #gpcr#drgpcr Published on May 26, 2025 Category GPCR Weekly News How do GPCRs sense pH changes? Did you know that we work hard to bring you the most recent GPCR News, weekly? #gpcr#drgpcr Previous Next Recent Articles
- Affiliate Policy | Dr. GPCR Ecosystem
GPCR Ecosystem. GPCR Ambassador Program Dr. GPCR, Corp., (“Dr. GPCR”, "DrGPCR", "Doctor GPCR", "Ecosystem Dr. GPCR", "EcosystemDrGPCR". Dr. GPCR”, "DrGPCR", "Doctor GPCR", "Ecosystem Dr. GPCR", "EcosystemDrGPCR". Dr. GPCR”, "DrGPCR", "Doctor GPCR", "Ecosystem Dr. GPCR", "EcosystemDrGPCR". Dr.
- 220 GPCRs. One platform. Endless questions. In Ep.167 of the Dr. GPCR Podcast, Tom Sakmar and Ilana Kotliar reveal a full GPCR-RAMP interaction map—powered by Luminex, dual-tagged constructs, and open science. Big win for the GPCR community. ✳️ Listen now: Ep 167 with Drs. Tom Sakmar & Ilana Kotliar #GPCRresearch #DrGPCR #GPCRpodcast #GPCRtools #OpenScience | Dr. GPCR Ecosystem
GPCR Podcast, Tom Sakmar and Ilana Kotliar reveal a full GPCR-RAMP interaction map—powered by Luminex Big win for the GPCR community. ✳️ Listen now: Ep 167 with Drs. GPCR Podcast 220 GPCRs. One platform. Endless questions. In Ep.167 of the Dr. GPCR Podcast, Tom Sakmar and Ilana Kotliar reveal a full GPCR-RAMP interaction map—powered by Luminex Big win for the GPCR community. ✳️ Listen now: Ep 167 with Drs.
- Check out the latest GPCR news in the Ecosystem today! You’ll need to register but don’t worry, it’s Free! Cutting-edge cryo-EM reveals how LYCHOS, a lysosomal protein, senses cholesterol to regulate metabolism and cell growth ➡️https://www.ecosystem.drgpcr.com/structural-and-molecular-insights-into-gpcr-function/cryo-em-reveals-cholesterol-binding-in-the-lysosomal-gpcr-like-protein-lychos #gpcr #drgpcr | Dr. GPCR Ecosystem
Home → Flash News → Check out the latest GPCR news in the Ecosystem today! metabolism and cell growth ➡️https://www.ecosystem.drgpcr.com/structural-and-molecular-insights-into-gpcr-function /cryo-em-reveals-cholesterol-binding-in-the-lysosomal-gpcr-like-protein-lychos #gpcr #drgpcr Published on February 4, 2025 Category GPCR Weekly News Check out the latest GPCR news in the Ecosystem today! /cryo-em-reveals-cholesterol-binding-in-the-lysosomal-gpcr-like-protein-lychos #gpcr #drgpcr Previous
- Inês Pinheiro, Monserrat Avila Zozaya & Yamina Berchiche | Dr. GPCR Ecosystem
GPCR Ecosystem About Monserrat Avila Zozaya I am a cell biologist interested in studying GPCRs, especially adhesion GPCRs. GPCR is to accelerate GPCR drug discovery by sharing the latest research and technology advances in the GPCR podcast. Dr. GPCR Ecosystem Enjoying the Dr. GPCR Podcast? Leave a Review.
- Check out our #SpotifyWrapped 🚀! In 2024, Dr. GPCR reached listeners worldwide, sparking conversations about GPCRs with top experts. Thank you for tuning in! 📊🎙️ ✳️Check out our top episode: https://www.ecosystem.drgpcr.com/dr-gpcr-podcast/ep-148-with-dr-arthur-christopoulos #gpcr #drgpcr | Dr. GPCR Ecosystem
GPCR reached listeners worldwide, sparking conversations about GPCRs with top experts. 📊🎙️ ✳️Check out our top episode: https://www.ecosystem.drgpcr.com/dr-gpcr-podcast/ep-148-with-dr-arthur-christopoulos #gpcr #drgpcr Published on January 29, 2025 Category Check out our #SpotifyWrapped 🚀! GPCR reached listeners worldwide, sparking conversations about GPCRs with top experts. #gpcr #drgpcr Previous Next Recent Articles
- Who We Are | Dr. GPCR Ecosystem
GPCR Ecosystem: uniting scientists, biotech, and innovators to advance GPCR research worldwide. GPCR Ecosystem We unite the GPCR Community to advance drug discovery Where GPCR Experts Move Science GPCR began as a podcast. GPCR Symposium with over 100 attendees 2024 GPCR University Launched comprehensive courses and expert The GPCR Challenge Scientists waste an average of 12 hours per week searching for relevant GPCR research
- What if you could map GPCR-RAMP interactions across the entire superfamily in a single experiment? That’s precisely what Dr. Kotliar from the Sakmar lab made possible! In Ep.167 of the Dr. GPCR Podcast, we chat with Drs. Tom Sakmar and Ilana Kotliar about how their lab developed: A multiplexed Luminex assay to screen hundreds of interactions at once A 220-clone DUET-tagged GPCR library, available on Addgene An online interface to search GPCR-RAMP data and antibody validations This is open-access science at its best, built for the GPCR research community. ✳️ Listen to the episode: Ep 167 with Drs. Tom Sakmar & Ilana Kotliar #GPCRresearch #DrGPCRecosystem #GPCRdrugdiscovery #GPCRtrainingprogram #GPCRpodcast | Dr. GPCR Ecosystem
Home → Flash News → What if you could map GPCR-RAMP interactions across the entire superfamily in a single GPCR Podcast, we chat with Drs. library, available on Addgene An online interface to search GPCR-RAMP data and antibody validations GPCR Podcast What if you could map GPCR-RAMP interactions across the entire superfamily in a single experiment GPCR Podcast, we chat with Drs.
- A new study from the Hudson Lab at the University of Glasgow shows that the FFA receptor antagonist AH7614 is actually an inverse agonist - suppressing fat cell formation, boosting lipolysis and reducing glucose uptake. Explore how targeting FFA4 could help fight metabolic disorders. Catch up with the latest research conducted in the Hudson lab in Ep. 161 of the Dr. GPCR Podcast. Subscribe to the Dr. GPCR Newsletter 📰 and get the latest GPCR News delivered to your inbox ➡️https://www.ecosystem.drgpcr.com/gpcrs-in-cardiology-endocrinology-and-taste/inverse-agonism-of-the-ffa4-free-fatty-acid-receptor-controls-both-adipogenesis-and-mature-adipocyte-function #GPCR #drGPCR #FFA4 #metabolism #adipocytes” | Dr. GPCR Ecosystem
GPCR Podcast. Subscribe to the Dr. GPCR Newsletter 📰 and get the latest GPCR News delivered to your inbox ➡️https://www.ecosystem.drgpcr.com #GPCR #drGPCR #FFA4 #metabolism #adipocytes” Published on April 7, 2025 Category GPCR Weekly News A GPCR Podcast. Subscribe to the Dr. GPCR Newsletter 📰 and get the latest GPCR News delivered to your inbox ➡️ https:// www.ecosystem.drgpcr.com
- Register for Adhesion GPCR Workshop 2024 | Dr. GPCR Ecosystem
Register now for the Adhesion GPCR Workshop 2024. Secure your spot to connect with leading GPCR researchers, attend sessions, and explore the latest in GPCR science. Home Registration Full Agenda Venue Travel Tips Sponsors Special Issue on Adhesion GPCRs Registrations Join the AGPCR24 group How to register for the Adhesion GPCR workshop 2024? If you're a Dr.
- Hacking GPCRs: Tools, Tech & Drug Discovery with Tom Sakmar & Ilana Kotliar | Dr. GPCR Ecosystem
GPCR signaling in disease. << Back to podcast list Strategic Partner(s) Hacking GPCRs: Tools, Tech & Beyond GPCR-RAMP: New Avenues “What if your favorite scaffold protein interacts with GPCRs?” Keyword Cloud GPCR-RAMP interactions , multiplex assays , GPCR research community , Dr. GPCR ecosystem , GPCR data platform , GPCR autoantibodies , Addgene GPCR library , GPCR training program GPCR Podcast? Leave a Review.
- Our History | Dr. GPCR Ecosystem
of GPCR science. GPCR Podcast episode premiered, featuring Dr. May 2022 — Media Partner at GPCR Retreat . Jul 2022 — Media Partner at GPCR ECI Transatlantic . GPCR University with the first GPCR Course led by Dr. Terry Kenakin , enrolling 30+ students . GPCR Team . May 16, 2024 — Episode #151 featured the Dr. GPCR Board .
- Dr. Yamina Berchiche | Dr. GPCR Ecosystem
GPCR podcast , your host and founder, Dr. Yamina Berchiche introduces the very first podcast dedicated to GPCRs researcher and their work. GPCR Ecosystem, with the goal is to bring together GPCR scientists, biotech, and pharma leaders as well , grow, and thrive together to accelerate GPCR drug discovery and improve human health. GPCR Ecosystem Enjoying the Dr. GPCR Podcast? Leave a Review.
- From Pipettes to Platforms The Evolution of GPCR Research | Dr. GPCR Ecosystem
Discover the evolution of GPCR research — from single pipettes to automated platforms shaping precision : The Evolution of GPCR Research Published on November 13, 2025 Category Dr. GPCR Podcast Back when GPCR assays were performed with single channel pipettes, failure wasn’t cheap. GPCR Premium for deeper tools and insights: https://www.ecosystem.drgpcr.com/gpcr-university-pricing #GPCR #DrGPCR #DrugDiscovery #Pharmacology #Biotech Previous Next Recent Articles
- About Dr. GPCR Ecosystem | Uniting the GPCR Community to Advance Drug Discovery
GPCR unites researchers, industry, and partners to accelerate GPCR science and drug discovery—through GPCR Ecosystem We unite the GPCR community to advance drug discovery. We bring the GPCR community together to fuel GPCR drug discovery—one receptor at a time. across the global GPCR ecosystem. : We verify GPCR relevance during onboarding to preserve focus and quality.
- Let’s connect the dots! Update your Dr. GPCR profile to make meaningful connections in the global GPCR network 🌐 ✳️Visit https://www.ecosystem.drgpcr.com/account/my-account and fill out the boxes with your most updated information. #gpcr #drgpcr | Dr. GPCR Ecosystem
GPCR profile to make meaningful connections in the global GPCR network 🌐 ✳️Visit https://www.ecosystem.drgpcr.com #gpcr #drgpcr Published on January 8, 2025 Category Dr. GPCR Profiles Let’s connect the dots! GPCR profile to make meaningful connections in the global GPCR network 🌐 ✳️Visit https://www.ecosystem.drgpcr.com #gpcr #drgpcr Previous Next Recent Articles
- Stay ahead in the GPCR field 💼 Updating your profile ensures you’re ready for the next opportunity. ✳️Go to https://www.ecosystem.drgpcr.com/account/my-account and let our GPCR-exclusive community know what you’re up to #gpcr #drgpcr | Dr. GPCR Ecosystem
Home → Flash News → Stay ahead in the GPCR field 💼 Updating your profile ensures you’re ready for the ✳️Go to https://www.ecosystem.drgpcr.com/account/my-account and let our GPCR-exclusive community know what you’re up to #gpcr #drgpcr Published on January 29, 2025 Category Dr. GPCR Profiles Stay ahead in the GPCR field 💼 Updating your profile ensures you’re ready for the next community know what you’re up to #gpcr #drgpcr Previous Next Recent Articles
- This study adds a key piece to the puzzle of adhesion GPCR signaling. Understanding receptor-specific nuances, like the role of NTF cleavage, is crucial for decoding their functional outcomes. Did you know that we work hard to bring you the most recent GPCR News, weekly? Catch up today in the Ecosystem using your free site membership! ➡️https://www.ecosystem.drgpcr.com/adhesion-gpcrs/n-terminal-fragment-shedding-contributes-to-signaling-of-the-full-length-adhesion-receptor-adgrl3 #gpcr #drgpcr | Dr. GPCR Ecosystem
Home → Flash News → This study adds a key piece to the puzzle of adhesion GPCR signaling. Did you know that we work hard to bring you the most recent GPCR News, weekly? #gpcr #drgpcr Published on January 28, 2025 Category GPCR Weekly News This study adds a key piece to the puzzle of adhesion GPCR signaling. #gpcr #drgpcr Previous Next Recent Articles
- Every receptor tells a story | Dr. GPCR Ecosystem
Every receptor tells a story but GPCRs speak a language of organization. Dr. Michelle Halls unpacks how GPCR signaling isn’t just about ligand–receptor interaction. a story Published on November 11, 2025 Category Dr.GPCR Podcast Every receptor tells a story — but GPCRs Michelle Halls unpacks how GPCR signaling isn’t just about ligand–receptor interaction. signaling: 👉 https://www.ecosystem.drgpcr.com/dr-gpcr-podcast/leadership-luck-and-gpcr-signaling #GPCR
- 🚀 Ready to dive into the world of GPCR drug development? Join Dr. Terry Kenakin for the 4-week course “Development of GPCR Ligands as Therapeutic Drugs”! Get exclusive access to expert lectures, recordings, reading materials, and even a private call with Dr. Kenakin himself! Don’t miss this chance to level up your knowledge. 🔹 Spots are limited—save yours now! 👉 https://www.ecosystem.drgpcr.com/event-details-registration/development-of-gpcr-ligands-as-therapeutic-drugs #gpcr #drgpcr #pharmacolgy #drugdiscovery #research | Dr. GPCR Ecosystem
Home → Flash News → 🚀 Ready to dive into the world of GPCR drug development? Join Dr. Terry Kenakin for the 4-week course “Development of GPCR Ligands as Therapeutic Drugs”! GPCR Courses 🚀 Ready to dive into the world of GPCR drug development? Join Dr. Terry Kenakin for the 4-week course “Development of GPCR Ligands as Therapeutic Drugs”! #gpcr #drgpcr #pharmacolgy #drugdiscovery #research Previous Next Recent Articles
- University | Dr. GPCR Ecosystem
Advance your GPCR research career with Dr. GPCR University. GPCR University A nonprofit created by scientists, for scientists—bringing the global GPCR community GPCR University? Dr. G protein-coupled receptors (GPCRs). GPCR University Masterclasses?
- Dr. Yamina Berchiche | Dr. GPCR Ecosystem
GPCR, an ecosystem designed to bring together stakeholders interested in using G-Protein Coupled Receptors (GPCRs) that control virtually everything in the body as drug targets. GPCR is to accelerate GPCR drug discovery by sharing the latest research and technology advances in the GPCR podcast. Dr. GPCR Ecosystem Enjoying the Dr. GPCR Podcast? Leave a Review.
- This new study reveals how the conformation of parathyroid hormone (PTH) and the C-terminal helix α5 of Gα regulate the selective coupling of PTH1R to Gs or Gq. Through Cryo-EM and single-cell experiments, the authors show differences in binding affinity, duration, and strength. Subscribe to the Dr. GPCR Newsletter 📰 and get the latest GPCR News delivered to your inbox ➡️ https://www.ecosystem.drgpcr.com/structural-and-molecular-insights-into-gpcr-function/allosteric-mechanism-in-the-distinctive-coupling-of-gq-and-gs-to-the-parathyroid-hormone-type-1-receptor #gpcr #drgpcr | Dr. GPCR Ecosystem
GPCR Newsletter 📰 and get the latest GPCR News delivered to your inbox ➡️ https://www.ecosystem.drgpcr.com /structural-and-molecular-insights-into-gpcr-function/allosteric-mechanism-in-the-distinctive-coupling-of-gq-and-gs-to-the-parathyroid-hormone-type -1-receptor #gpcr #drgpcr Published on April 28, 2025 Category GPCR Weekly News This new study reveals GPCR Newsletter 📰 and get the latest GPCR News delivered to your inbox ➡️ https://www.ecosystem.drgpcr.com -1-receptor #gpcr #drgpcr Previous Next Recent Articles
- Class B GPCR drugs are reshaping treatment for migraine, diabetes, and obesity- but did you know ligand bias plays a key role in their success? This new review explores how tweaking peptide drugs can boost efficacy, reduce side effects, and unlock next-gen therapies. Subscribe to the Dr. GPCR Newsletter 📰 and get the latest GPCR News delivered to your inbox ➡️https://www.ecosystem.drgpcr.com/reviews/where-are-we-now%3F-biased-signalling-of-class-b-g-protein-coupled-receptor-targeted-therapeutics #gpcr#drgpcr | Dr. GPCR Ecosystem
Home → Flash News → Class B GPCR drugs are reshaping treatment for migraine, diabetes, and obesity- but GPCR Newsletter 📰 and get the latest GPCR News delivered to your inbox ➡️https://www.ecosystem.drgpcr.com /where-are-we-now%3F-biased-signalling-of-class-b-g-protein-coupled-receptor-targeted-therapeutics #gpcr #drgpcr Published on June 2, 2025 Category GPCR Weekly News Class B GPCR drugs are reshaping treatment GPCR Newsletter 📰 and get the latest GPCR News delivered to your inbox ➡️ https://www.ecosystem.drgpcr.com
- where signaling happens inside a cell | Dr. GPCR Ecosystem
Michelle describes how reading those early papers on lipid-rich domains and GPCR–G protein compartmentalization This moment cuts straight to the heart of how many of us fell in love with GPCR biology — that realization If you work with GPCRs, this perspective changes how you design experiments and interpret data. 🎧 Watch /leadership-luck-and-gpcr-signaling ✨ Join Premium: https://www.ecosystem.drgpcr.com/gpcr-university-pricing #GPCR #DrGPCR Previous Next Recent Articles
- Dr. Juan José Fung | Dr. GPCR Ecosystem
Juan José Fung is a Principal Scientist at GPCR Therapeutics, Inc , a drug discovery company focused on targeting GPCR heteromers in cancer, headquartered in Seoul, Korea, with an R&D facility in the SF Brian Kobilka , studying the dimerization of GPCRs. Dr. Juan José Fung on the web LinkedIn GPCR Therapeutics Dr. GPCR Ecosystem Enjoying the Dr. GPCR Podcast? Leave a Review.
- What are your thoughts on β2AR? Listen to Ep.163 of the @DrGPCR Podcast, where @DVeprintsev shares his thoughts and experiences about working with GPCRs, tips on framing your research correctly, and other insightful topics. Don’t miss out! ✳️https://www.ecosystem.drgpcr.com/dr-gpcr-podcast/ep-163-with-dr.-dmitry- #GPCRs #SciencePodcast #DrugDiscovery #Biotech #DrGPCR | Dr. GPCR Ecosystem
.163 of the @DrGPCR Podcast, where @DVeprintsev shares his thoughts and experiences about working with GPCRs ✳️https://www.ecosystem.drgpcr.com/dr-gpcr-podcast/ep-163-with-dr. GPCR Podcast What are your thoughts on β2AR? ✳️ https://www.ecosystem.drgpcr.com/dr-gpcr-podcast/ep-163-with-dr. -dmitry- #GPCRs #SciencePodcast #DrugDiscovery #Biotech #DrGPCR Previous Next Recent Articles
- Science isn't always about eureka moments—sometimes it's about steady progress. In our latest Dr. GPCR Podcast episode, Ian Chronis shares his top aha moments, from learning the hard way about gel electrophoresis to discovering the hidden complexities of GPCR signaling. ✅ https://buff.ly/FTB69y9 #GPCR #DrGPCR #SciencePodcast #Pharmacology | Dr. GPCR Ecosystem
GPCR Podcast episode, Ian Chronis shares his top aha moments, from learning the hard way about gel electrophoresis to discovering the hidden complexities of GPCR signaling. ✅ https://buff.ly/FTB69y9 #GPCR #DrGPCR #SciencePodcast GPCR Podcast Science isn't always about eureka moments—sometimes it's about steady progress. GPCR Podcast episode, Ian Chronis shares his top aha moments, from learning the hard way about gel electrophoresis to discovering the hidden complexities of GPCR signaling. ✅ https://buff.ly/FTB69y9 #GPCR #DrGPCR #SciencePodcast
- Flash News: Your Hub for GPCR Insights and Scientific Conference Programs
GPCR blog breaks down the moment Dr. #GPCR #DrGPCR #GPCRimaging #biotech #drugdiscovery A GPCR imaging breakthrough that didn’t start in signaling: 👉 https://www.ecosystem.drgpcr.com/dr-gpcr-podcast/leadership-luck-and-gpcr-signaling #GPCR GPCR Premium → https://www.ecosystem.drgpcr.com/gpcr-university #GPCR #DrGPCR #pharmacology #drugdiscovery GPCR Podcast : https://www.ecosystem.drgpcr.com/dr-gpcr-podcast/model-predict-discover #DrGPCR #GPCR
- Dr. Simone Prömel & Dr. Ines Liebscher | Dr. GPCR Ecosystem
of the Adhesion GPCR Latrophilin-1. There she focused on the different modes of action of Adhesion GPCRs and found that they do not only GPCR Ecosystem About Dr. Ines Liebscher Dr. Her postdoctoral work leads her to investigate a whole family of orphan receptors: adhesion GPCRs. GPCR Ecosystem Enjoying the Dr. GPCR Podcast? Leave a Review.
