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GPCR unites researchers, industry, and partners to accelerate GPCR science and drug discovery—through GPCR Ecosystem We unite the GPCR community to advance drug discovery. We bring the GPCR community together to fuel GPCR drug discovery—one receptor at a time. Contact Us Our Mission Advance GPCR science and drug discovery by connecting people, data, and opportunities across the global GPCR ecosystem.

function The NTF Release Sensor Approach for Drug Discovery for Human Adhesion GPCRs Stephanie Häfner Discovery for Human Adhesion GPCRs Stephanie Häfner Abstract "G Protein-coupled receptors (GPCRs) are common drug targets, yet no approved drugs exist for the Adhesion G Protein-coupled receptors (aGPCRs drug discovery methods. This tailored system aims to expedite the identification of drugs targeting the unique aGPCR receptor

Drugs” closes March 18th! If you’re working on GPCR drug discovery, you know that finding a promising candidate is just the start 👉 Development of GPCR Ligands as Therapeutic Drugs | Dr. If you’re working on GPCR drug discovery , you know that finding a promising candidate is just the start 👉 Development of GPCR Ligands as Therapeutic Drugs | Dr.

Measuring and understanding bias helps design drugs that maximize therapeutic benefits while minimizing Kinetics to Candidate Design Lecture 4: Unconventional GPCR Ligands as Drugs Lecture 5: Unique Exploitable Lecture 1: GPCR Project Initiation and Design for Discovery of New Molecules Lecture 2: Drug Affinity GPCR University Masterclasses designed for? Some classes may require basic knowledge of GPCRs, but many are designed to accommodate beginners as

Home → Flash News → irreversible drugs post 3 Irreversible kinetics = strategic lever in drug design. These lessons bridge molecular pharmacology with real-world design strategy, giving discovery teams the Quantifying irreversible activity (K_inact / K_I) — turning persistent binding into measurable design GPCR Ecosystem #GPCR #DrGPCR #Pharmacology #DrugDiscovery #Kinetics #ReceptorPharmacology #MedicinalChemistry uncomfortable truth: 👉 Your biotech is already running on an operating cadence you didn’t consciously design

GPCR, an ecosystem designed to bring together stakeholders interested in using G-Protein Coupled Receptors (GPCRs) that control virtually everything in the body as drug targets. GPCR is to accelerate GPCR drug discovery by sharing the latest research and technology advances in the GPCR About John Azietaku John Teye Azietaku,PhD is a trained pharmacist, holding a Ph.D. in Drug Discovery virtual drug screening to identify agonists and antagonists targeting Class A GPCRs.

Home → Flash News → 💡 GPCR drug development doesn’t have to be a mystery! Learn from Dr. Sign up today 👉 Development of GPCR Ligands as Therapeutic Drugs | Dr. GPCR Courses 💡 GPCR drug development doesn’t have to be a mystery! Learn from Dr. Sign up today 👉 Development of GPCR Ligands as Therapeutic Drugs | Dr. uncomfortable truth: 👉 Your biotech is already running on an operating cadence you didn’t consciously design

Discover how low-offset kinetics reshape drug efficacy. Home → Flash News → irreversible drugs post 1 Irreversible Drugs – Trailer Published on October 21, 2025 Category Terry's Corner Irreversible drugs change the rules of engagement. GPCR Ecosystem #GPCR #DrGPCR #Pharmacology #DrugDiscovery #MedicinalChemistry #PKPD #ReceptorKinetics uncomfortable truth: 👉 Your biotech is already running on an operating cadence you didn’t consciously design

Applying Pharmacology to Drug Discovery Dr. Terry Kenakin Get Started Premium Members benefits: - Subscribe and save 25% on every GPCR Course - Early-bird access - Recordings will be available < Back to GPCR courses Watch recording Your Instructor Dr.

Terry Kenakin is hosting a 4-week course on GPCR drug development—and registration closes in 3 days! 👉 Development of GPCR Ligands as Therapeutic Drugs | Dr. Terry Kenakin is hosting a 4-week course on GPCR drug development —and registration closes in 3 days! 👉 Development of GPCR Ligands as Therapeutic Drugs | Dr. GPCR Ecosystem #GPCR #DrGPCR #Pharma #Biotech #Research Previous Next Recent Articles

signaling and function NovoiSMART - A new platform for GPCR antibody drug discovery Gavin Zhang Read Signaling and Pharmacology-Enabling Drug Discovery Fabian Pohl Structural Determinants Of GAIN Domain Stephanie Häfner The NTF Release Sensor Approach for Drug Discovery for Human Adhesion GPCRs Anne Bormann Placantonakis Antibody-drug conjugates targeting CD97 in glioblastoma Gabriela Aust Critical role for map of thermogenic fat Gavin Zhang NovoiSMART - A new platform for GPCR antibody drug discovery

Drug Discovery with Tom Sakmar & Ilana Kotliar In this episode, host Dr. Ilana Kotliar , his former graduate student, to explore the development of powerful multiplex tools designed , GPCR drug discovery , GPCR online course Summary created by AI ________ About Tom Sakmar Tom Sakmar is a physician-scientist and Rockefeller University professor dedicated to drug discovery and chemical He and his artist/designer wife, Karina Åberg, have three teenage children.

GPCR Ecosystem – the ultimate hub for GPCR professionals to connect, collaborate, and advance drug discovery Home: About Accelerating GPCR Drug Discovery, Together Dr. GPCR is the global hub where academia and industry meet to advance GPCR research, accelerate drug discovery Mastery Flexible, career-ready courses designed by scientists for scientists. field 🧠 Designed for researchers at every career stage 🚀 Don’t just keep up — lead the way. 🔒 Grandfather

Home → Flash News → 🚀 Ready to dive into the world of GPCR drug development? Join Dr. Terry Kenakin for the 4-week course “Development of GPCR Ligands as Therapeutic Drugs”! 👉 https://www.ecosystem.drgpcr.com/event-details-registration/development-of-gpcr-ligands-as-therapeutic-drugs GPCR Courses 🚀 Ready to dive into the world of GPCR drug development? Join Dr. Terry Kenakin for the 4-week course “Development of GPCR Ligands as Therapeutic Drugs”!

GPCR, an ecosystem designed to bring together stakeholders interested in using G-Protein Coupled Receptors (GPCRs) that control virtually everything in the body as drug targets. GPCR is to accelerate GPCR drug discovery by sharing the latest research and technology advances in the on GPCRs. biology and for the identification of drug targets and future drug development.

Principles of Pharmacology in Drug Discovery I Dr. Terry Kenakin Get Started Premium Members benefits: - Subscribe and save 25% on every GPCR Course - Early-bird access - Recordings will be available < Back to GPCR courses Watch recording Your Instructor Dr.

Principles of Pharmacology in Drug Discovery II Dr. Terry Kenakin Get Started Premium Members benefits: - Subscribe and save 25% on every GPCR Course - Early-bird access - Recordings will be available < Back to GPCR courses Watch recording Your Instructor Dr.

<< Back to podcast list Strategic Partner(s) Empowering Drug Discovery for the GPCR Community with Dr GPCR Enjoying the Dr. GPCR Podcast? Leave a Review. Better Questions in Science: A Practical Guide for Emerging Researchers When the Islet Lit Up: Advancing GPCR Imaging in Native Tissue How Collaboration Sparked a GPCR Imaging Breakthrough in Chemical Biology Thanks

GPCR Foundry: Accelerate GPCR Drug Discovery Move from idea to insight—faster, smarter, and with confidence GPCR Foundry is a nonprofit platform designed to help biotech leaders accelerate GPCR drug discovery De-risk decisions: gain expert strategic guidance on study design, timelines, and partner selection before Stay ahead of the curve with expert-led programs designed for real-world biotech challenges. → Explore innovators and showcase your expertise Training & Upskilling Specialized, insight-packed courses designed

Explore the kinetic principles behind persistent binding and smarter drug design. Home → Flash News → irreversible drugs post 2 Persistent binding ≠ just covalent. Published on October 24, 2025 Category Terry's Corner Why do some inhibitors act long after the drug Binding kinetics are a design variable, as critical as potency or clearance. #GPCR #DrGPCR #Pharmacology #DrugDiscovery #BindingKinetics #ReceptorPharmacology #MedicinalChemistry

Your One-Stop-Shop for GPCR Drug Discovery and Development Researchers developing GPCR-targeted therapeutics These industry-standard assays, designed for regulatory submissions, are backed by partnerships with research and drug discovery and development. GPCR services, the benefits from integration provide the most comprehensive GPCR research and drug discovery Learn how pH Sense changes the game for drug discovery. Dr.

GPCR University: "Development of GPCR Ligands as Therapeutic Drugs." 🗓 Dates: March 20 - April 10, 2025 Gain deep insights into GPCR drug candidates and learn the critical assays and techniques required to GPCR Courses 🚨 Exciting Opportunity for Professionals in Drug Development! GPCR University: "Development of GPCR Ligands as Therapeutic Drugs." 🗓 Dates: March 20 - April 10, 2025 Gain deep insights into GPCR drug candidates and learn the critical assays and techniques required to

Full Agenda Adhesion GPCR workshop 2024 CINVESTAV, Mexico City, Mexico October 23-25 Download PDF Program - A new platform for GPCR antibody drug discovery Abstract Developing monoclonal antibody drugs against GPCRs and other multi-pass transmembrane targets, such as ion channels, remains a significant challenge Several case studies of GPCR and other multi-pass transmembrane targets are presented, including GPRC5D developing highly specific antibodies for complex targets, with implications for overcoming challenges like drug

GPCR location within the cell can change everything: function, pharmacology, and even drug response. from the lab to the broader biotech world This episode is packed with knowledge for scientists, drug GPCR Podcast 🎧 Why Does GPCR Location Make All the Difference? GPCR location within the cell can change everything: function, pharmacology, and even drug response. from the lab to the broader biotech world This episode is packed with knowledge for scientists, drug

Your go-to hub for everything GPCR! Read Full Issue November 14 - 20, 2025 Crafting Chemical Keys for GPCR Drug Discovery Read Full Issue GPCR initiative. research and drug discovery. field 🧠 Designed for researchers at every career stage 🚀 Don’t just keep up — lead the way. 🔒 Grandfather

Home → Flash News → terrys corner predict drug behavior Published on July 12, 2025 Category Terry's Corner Dive into the logic of drug modeling with Terry Kenakin. Learn to “extend your eyes” and predict complex drug behaviors. 🟢 Browse the full catalog (and expect ✳️ https://www.terrykenakin.com #pharmacology #drugmechanism #kenakin #GPCR #DrGPCR Previous Next Recent

Coordinated Universal Time) Details Neomorphic mutations in GNAO1 encephalopathy: from mechanisms to drug drug discovery enabled by the Confo Therapeutics technology Dr. & G protein biosensors for drug discovery & assessment of constitutive activity Dr. Structure-based Drug Design: The Orexin System and Suvorexant Daniel Gruffat, M.Sc Thu Oct 13 2022 14 drug discovery: Focus on psychedelics Dr.

Measuring and understanding bias helps design drugs that maximize therapeutic benefits while minimizing recording Strategic Project Management for scientists Gain practical project management skills explicitly designed Yamina Berchiche 🔒 Premium Content Watch recording Applying Pharmacology to Drug Discovery Class 1 - Kinetics to Candidate Design Lecture 4: Unconventional GPCR Ligands as Drugs Lecture 5: Unique Exploitable Lecture 1: GPCR Project Initiation and Design for Discovery of New Molecules Lecture 2: Drug Affinity

Home → Flash News → terrys corner model drug response Published on July 10, 2025 Category Terry's Corner What if a single experimental snapshot could predict an entire in vivo drug profile in a range of organs discussed. 🟢 Read the full breakdown: ✳️ https://www.ecosystem.drgpcr.com/post/what-if-you-could-predict-drug-behavior-with-just-a-snapshot #GPCR #DrGPCR #pharmacology #DrugDiscovery #TerryKenakin #FoundationalScience Previous Next Recent Articles

GPCR: Advancing GPCR Drug Discovery Through Collaboration Discovery On Target 2024 GPCR targeted drug discovery Summit 2024 GPCR targeted drug discovery Summit 2023 The Dr. GPCR Podcast GPCR targeted drug discovery Summit 2022 Dr. GPCR: Where all GPCRs are created equal Dr. GPCR: Beyond the lab Dr. GPCR: From idea to Ecosystem Dr. GPCR: Beyond the lab