📰 GPCR Weekly News, January 30 to February 5, 2023
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Below is your Classified GPCR News at a glance for January 30th to February 5th, 2023.
GPCR Activation and Signaling
Cannabinoid 1 (CB1 ) receptor arrestin subtype-selectivity and phosphorylation dependence.
Platelet P2Y1 receptor exhibits constitutive G protein signaling and β-arrestin 2 recruitment.
GPCR Binders, Drugs, and more
GPCRs in Cardiology, Endocrinology, and Taste
GPCRs in Oncology and Immunology
Methods & Updates in GPCR Research
Computational investigation of functional water molecules in GPCRs bound to G protein or arrestin.
Functional expression of oxytocin receptors in pulp-dentin complex.
Reviews, GPCRs, and more
Understanding Neuropeptide Transmission in the Brain by Optical Uncaging and Release.
Non-canonical Golgi-compartmentalized Gβγ signaling: mechanisms, functions, and therapeutic targets.
β-arrestins and G protein-coupled receptor kinases in viral entry: A graphical review.
Development and challenges in the discovery of 5-HT1A and 5-HT7 receptor ligands.
Structural and Molecular Insights into GPCR Function
Structural view of G protein-coupled receptor signaling in the retinal rod outer segment.
Cryo-EM structure of orphan G protein-coupled receptor GPR21.
Industry News
GPCR Therapeutics Announces Launch of US Phase 2 Trial of GPC-100 in Multiple Myeloma
TGA’s approval of MDMA and Psilocybin for medical use is a result of ‘renewed interest’
Addex Strategic Partner Completes Enrollment In Adx71149 Epilepsy Phase 2 Study Part 1
Domain Therapeutics to Participate in Upcoming Investor and Industry Conferences
Endocrine Society Awards Baxter Prize to Innovator in Endocrine Drug Discovery
Upstream Bio Announces the Appointment of Marcella Ruddy, M.D., to the Board of Directors
Call for GPCR Papers
GPCRs: Signal Transduction. Deadline extended to March 31st, 2023
GPCR Events, Meetings, and Webinars
2nd GPCR-Targeted Drug Discovery Summit, (February 21 - 23, 2023), Boston.
SLAS2023 International Conference and Exhibition (February 25 - March 1, 2023).
SLAS Europe 2023 Conference and Exhibition. (May 22 - 26, 2023)
2nd LEAPS Meets Life Sciences Conference. (May 14 - 19, 2023)
The Illuminating the Understudied Druggable Proteome Conference. (June 4 - 8, 2023).
2023 Molecular Pharmacology (GRS) Seminar GRC. (June 10 - 11, 2023).
19th World Congress of Basic & Clinical Pharmacology 2023. (July 2 - 7, 2023).
GPCR Jobs
Computational drug design PhD student at the Department of Drug Design and Pharmacology
Computational drug design postdoc at the Department of Drug Design and Pharmacology
Software / database development PhD student at Department of Drug Design and Pharmacology
Software / database development postdoc at the Department of Drug Design and Pharmacology
Postdoc in Bioinformatics/Data Science at Department of Drug Design and Pharmacology