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Results found for "GPCR Drug Design"
- Custom Molecules, Fluorescent Probes: When Chemists Think Like Biologists with Dr. Maria Majellaro from Celtarys | Dr. GPCR Ecosystem
at the bench and in translational drug discovery. Galicia’s robust biotech network, and the company quickly defined its value: building better tools for drug , probe design, and the realities of scaling innovation from lab bench to product launch. Whether you're designing assays, developing probes, or seeking better tools for GPCR drug discovery, GPCR ecosystem , GPCR drug discovery , fluorescent ligands , GPCR scientist network , custom ligand development
- ep 175 with jens carlsson clip 3 | Dr. GPCR Ecosystem
AI is transforming GPCR modeling. scientists to go beyond explaining data — and start predicting the future of receptor function and drug GPCR Podcast AI is changing how we think about structure, function, and discovery — but Jens Carlsson That’s where the future of GPCR research lies — not in describing the past, but in anticipating it. Whether you’re running simulations, screening compounds, or designing next-gen molecules, this insight
- Think βCGRP is just αCGRP’s understudy? Think again. New research shows that βCGRP triggers distinct receptor signaling profiles across the CGRP receptor family, challenging the long-held assumption of redundancy. 🔬 A closer look reveals differences in G protein coupling, second messenger production, and receptor trafficking. 📊 This could reshape how we understand CGRP-related physiology—and how we target it in drug design. 🧠 Pain, inflammation, metabolism: the implications go far beyond signaling bias. 🔗 Read the full paper in Biochemistry: Unique Biased Agonism Profile of βCGRP on CGRP Family Receptors #GPCR #CGRP #DrugDiscovery #Pharmacology #SignalTransduction #Neuropeptides | Dr. GPCR Ecosystem
. 📊 This could reshape how we understand CGRP-related physiology—and how we target it in drug design #DrugDiscovery #Pharmacology #SignalTransduction #Neuropeptides Published on June 16, 2025 Category GPCR trafficking. 📊 This could reshape how we understand CGRP-related physiology—and how we target it in drug design. 🧠 Pain, inflammation, metabolism: the implications go far beyond signaling bias. 🔗 Read the full paper in Biochemistry : Unique Biased Agonism Profile of βCGRP on CGRP Family Receptors #GPCR #
- Chris Langmead | Dr. GPCR Ecosystem
He is an acknowledged expert in drug discovery, particularly in the field of psychiatry, where he has He has published over 70 research articles, reviews and book chapters on drug discovery, which have been GPCR Ecosystem Enjoying the Dr. GPCR Podcast? Leave a Review. Better Questions in Science: A Practical Guide for Emerging Researchers When the Islet Lit Up: Advancing GPCR Imaging in Native Tissue How Collaboration Sparked a GPCR Imaging Breakthrough in Chemical Biology Thanks
- Dr. Kari Johnson | Dr. GPCR Ecosystem
University before continuing her training as a postdoctoral fellow at the Vanderbilt Center for Neuroscience Drug All through her career, the recurring theme in Kari’s work has been GPCRs and more specifically Metabotropic Join me and learn more about how Kari studies GPCRs in basal ganglia circuits following chronic alcohol GPCR Ecosystem Enjoying the Dr. GPCR Podcast? Leave a Review. Imaging in Native Tissue How Collaboration Sparked a GPCR Imaging Breakthrough in Chemical Biology Thanks
- Newsletter for Adhesion GPCR Workshop 2024 | Dr. GPCR Ecosystem
Subscribe to the Adhesion GPCR Workshop 2024 newsletter. Adhesion GPCR workshop 2024 CINVESTAV, Mexico City, Mexico October 23-25 Register AGPCR Newsletter Adhesion GPCR Consortium Newsletter - May 2024 Welcome to the 4th official Adhesion GPCR Consortium newsletter GPCR News Register for the Adhesion GPCR 2024 Learn more about the Adhesion GPCR workshop 2024 Up About the event Learn more about the Adhesion GPCR workshop 2024 and its preliminary program.
- Steve McCloskey | Dr. GPCR Ecosystem
Scientists and Engineers working at the nanoscale, specifically protein engineering and small molecule drug GPCR Ecosystem Enjoying the Dr. GPCR Podcast? Leave a Review. Better Questions in Science: A Practical Guide for Emerging Researchers When the Islet Lit Up: Advancing GPCR Imaging in Native Tissue How Collaboration Sparked a GPCR Imaging Breakthrough in Chemical Biology Thanks
- Dr. Oliver Hartley | Dr. GPCR Ecosystem
Oliver Hartley Oliver Hartley is VP for Drug Discovery at Orion Biotechnology . Since then Oliver has worked at the University of Geneva, where his research on peptide engineering and GPCR GPCR Ecosystem Enjoying the Dr. GPCR Podcast? Leave a Review. Better Questions in Science: A Practical Guide for Emerging Researchers When the Islet Lit Up: Advancing GPCR Imaging in Native Tissue How Collaboration Sparked a GPCR Imaging Breakthrough in Chemical Biology Thanks
- terrys corner no fluff pure insight | Dr. GPCR Ecosystem
✨ We've poured our passion for pharmacology into creating this essential resource, designed to meet you exactly where you are in your drug discovery journey. Bridge theory to practical drug development decisions? #pharmacology #GPCRscience #drugdiscovery #TerrysCorner #biotechtraining #ScienceEducation #Pharma #GPCR
- Dr. Nicholas Holliday | Dr. GPCR Ecosystem
and the immune system, and the molecular mechanisms underlying the signaling and regulation of their GPCRs Excellerate is involved in several pre-clinical drug discovery projects for both GPCR and non-GPCR targets GPCR Ecosystem Enjoying the Dr. GPCR Podcast? Leave a Review. Better Questions in Science: A Practical Guide for Emerging Researchers When the Islet Lit Up: Advancing GPCR Imaging in Native Tissue How Collaboration Sparked a GPCR Imaging Breakthrough in Chemical Biology Thanks
- 🚀 New Workshop: Practical Quantification of Allosteric Modulation Join Dr. Terry Kenakin on May 1st, 2025, for an advanced live workshop on allosteric modulators in GPCR drug discovery. Learn how to: ✔️ Identify, measure, and quantify allosteric properties ✔️ Apply functional allosteric models to determine mechanisms of action ✔️ Confirm allostery through kinetic analysis 📅 Date: May 1st, 2025 ⏳ Registration deadline: April 18th 📍 Live on Google Meet 🔗 Register now: https://www.ecosystem.drgpcr.com/event-details-registration/practical-quantification-of-allosteric-modulation #GPCR #Allostery #DrugDiscovery #Pharmacology | Dr. GPCR Ecosystem
Terry Kenakin on May 1st, 2025, for an advanced live workshop on allosteric modulators in GPCR drug discovery www.ecosystem.drgpcr.com/event-details-registration/practical-quantification-of-allosteric-modulation #GPCR #Allostery #DrugDiscovery #Pharmacology Published on March 3, 2025 Category GPCR University 🚀 New Workshop Terry Kenakin on May 1st, 2025 , for an advanced live workshop on allosteric modulators in GPCR drug www.ecosystem.drgpcr.com/event-details-registration/practical-quantification-of-allosteric-modulation #GPCR
- “Research is all about knowing when to walk and when to run.” –Ben Clements In Ep. 166 of the Dr.GPCR Podcast, hear how a postdoc is reshaping the conversation on opioid use, imposter syndrome, and the power of collaborative science. Why early-career voices are critical in GPCR drug discovery —and how lab culture makes all the difference. 🎧 Watch here: https://buff.ly/Kr3qKud #GPCRresearch #DrGPCR #GPCRpodcast #OpioidPharmacology #DrugDiscovery | Dr. GPCR Ecosystem
Why early-career voices are critical in GPCR drug discovery —and how lab culture makes all the difference GPCR Podcast “Research is all about knowing when to walk and when to run.” Why early-career voices are critical in GPCR drug discovery —and how lab culture makes all the difference
- Dr. Michel Bouvier | Dr. GPCR Ecosystem
He is a world-renowned expert in the field of cell signaling and GPCRs and made seminal contributions to our understanding of this major class of drug targets. energy transfer (BRET) resulted in the development of screening assays that are now widely used for drug been able to work with him and his team and use the tools developed in his lab to better understand GPCR GPCR Ecosystem Enjoying the Dr. GPCR Podcast? Leave a Review.
- pharmacology at your fingertips terrys corner launches | Dr. GPCR Ecosystem
Flash News → pharmacology at your fingertips terrys corner launches Published on July 4, 2025 Category GPCR Weekly News Stronger pharmacology drives smarter decisions in GPCR discovery. Elevate your drug discovery program with 45+ lessons yearly. GPCR Weekly: ♦️ Yamina’s Corner—GPCR consulting to de-risk and accelerate your pipeline ♦️ Celtarys’ validated TR-FRET assay for CB1/CB2 ♦️ Chemokine-GPCR selectivity decoded ♦️ PTH1R structures reveal
- Dr. Rosie Dawaliby | Dr. GPCR Ecosystem
Rosie Dawaliby "I’m an expert in early-stage drug discovery, targeting membrane proteins, especially GPCR. I have developed my expertise in the field of pharmacology and biochemistry of GPCR and the crucial role In 2016, I joined a company that specialized in therapeutic candidate discovery targeting GPCR ( Confo GPCR Ecosystem G.CLIPS Biotech on the web Website LinkedIn Enjoying the Dr. GPCR Podcast?
- Dr. Sai Prasad Pydi | Dr. GPCR Ecosystem
. from the University of Manitoba – Canada, where he was introduced to G protein-coupled receptors (GPCRs (NIDDK) - NIH, USA as a postdoctoral fellow and trained on understanding the physiological role of GPCR Pydi's laboratory is to develop GPCR-based drugs for the treatment of obesity and Type 2 Diabetes (T2D GPCR Ecosystem Enjoying the Dr. GPCR Podcast? Leave a Review. Imaging in Native Tissue How Collaboration Sparked a GPCR Imaging Breakthrough in Chemical Biology Thanks
- Ever wondered how we perceive bitterness? 👅🔬 Researchers have unveiled the cryo-EM structure of TAS2R14, the most promiscuous bitter taste receptor, bound to the drug flufenamic acid (FFA) and its signaling partner gustducin! 🌟 This discovery reveals an unusual dual binding mode of FFA and offers tools for site-targeted compound design. 🧪✨ Learn more about this exciting breakthrough in bitter taste signaling. | Dr. GPCR Ecosystem
unveiled the cryo-EM structure of TAS2R14, the most promiscuous bitter taste receptor, bound to the drug This discovery reveals an unusual dual binding mode of FFA and offers tools for site-targeted compound design This discovery reveals an unusual dual binding mode of FFA and offers tools for site-targeted compound design signaling. ➡️ https://www.ecosystem.drgpcr.com/receptor-activation-and-signaling/a-bitter-anti-inflammatory-drug-binds-at-two-distinct-sites-of-a-human-bitter-taste-gpcr uncomfortable truth: 👉 Your biotech is already running on an operating cadence you didn’t consciously design
- Dr. Khaled Abdelrahman | Dr. GPCR Ecosystem
He has been also studying what aspects of GPCR signaling are regulated in a sex-selective manner and how this can influence drug discovery in the area of neurodegenerative diseases. GPCR Ecosystem Enjoying the Dr. GPCR Podcast? Leave a Review. Better Questions in Science: A Practical Guide for Emerging Researchers When the Islet Lit Up: Advancing GPCR Imaging in Native Tissue How Collaboration Sparked a GPCR Imaging Breakthrough in Chemical Biology Thanks
- Exploring Career Paths in GPCR Research with Dr. Jacek Mokrosiński | Dr. GPCR Ecosystem
<< Back to podcast list Strategic Partner(s) Exploring Career Paths in GPCR Research with Dr. name mispronunciations, cultural differences, and the importance of a multidisciplinary approach in drug discussed their professional backgrounds, highlighting the benefits of a multidisciplinary approach in drug their research interests and achievements, particularly in the field of GPCR. GPCR Podcast? Leave a Review.
- Media Partner Packages | Dr. GPCR Ecosystem
GPCR Ecosystem. Elevate Your GPCR Focused Company Visibility Reach 1300+ GPCR researchers. GPCR is the world's largest nonprofit community focused on GPCRs. partner, you'll gain trusted access to an engaged audience of academic researchers, biotech teams, and drug GPCR?
- Dr. Patrick Sexton | Dr. GPCR Ecosystem
He is a leader in the study of GPCRs, biased agonism, and also on allosteric interactions between GPCRs has been at the forefront of the application of cryo-EM to elucidate of the structure and dynamics of GPCRs of the International Union of Basic and Clinical Pharmacology Committee on Receptor Nomenclature and Drug GPCR Ecosystem Enjoying the Dr. GPCR Podcast? Leave a Review. Imaging in Native Tissue How Collaboration Sparked a GPCR Imaging Breakthrough in Chemical Biology Thanks
- Dr. Graeme Milligan | Dr. GPCR Ecosystem
main research group centers on the function, structure, and regulation of G protein-coupled receptors (GPCRs and identification of small molecule regulators of these proteins, and progressing such ligands in drug GPCR Ecosystem Enjoying the Dr. GPCR Podcast? Leave a Review. Better Questions in Science: A Practical Guide for Emerging Researchers When the Islet Lit Up: Advancing GPCR Imaging in Native Tissue How Collaboration Sparked a GPCR Imaging Breakthrough in Chemical Biology Thanks
- Courses by Terry | Dr. GPCR Ecosystem
Home Courses Articles About Log In / Sign Up Terry's Pharmacology Corner Lost in GPCR Complexity? Valid until canceled 7 day free trial Select Watch 4 New Courses Each Month Connect in a Private Drug Skip The Fluff, Learn What Matters Join Monthly AMAs with Terry Unlock 40+ Years of Expertise Master GPCRs GPCR . Stay connected on LinkedIn and YouTube . Explore : Foundational Lessons — Build Your Pharmacology Core Emerging Drug Hunter — Expand Your Edge
- Sponsorship Prospectus for Adhesion GPCR Workshop 2024 | Dr. GPCR Ecosystem
Explore sponsorship opportunities for the Adhesion GPCR Workshop 2024. We are delighted to present the sponsorship opportunities available for Adhesion GPCR Workshop 2024, About the Adhesion GPCR Workshop 2024: Adhesion GPCR Workshop 2024 is a high-profile expert conference Opportunity to be designated in print on the 1 st ever “aGPCR Excellence and Mentoring Award” Customized GPCR workshop 2024 and its preliminary program.
- Scott Struthers | Dr. GPCR Ecosystem
he led contract research efforts at Biosym Technologies to develop and apply computational tools for drug GPCR Ecosystem Enjoying the Dr. GPCR Podcast? Leave a Review. Better Questions in Science: A Practical Guide for Emerging Researchers When the Islet Lit Up: Advancing GPCR Imaging in Native Tissue How Collaboration Sparked a GPCR Imaging Breakthrough in Chemical Biology Thanks
- The Scientist's Compass: From Academia to Entrepreneurship with Dr. Dmitry Veprintsev | Dr. GPCR Ecosystem
Why GPCRs? Building Z7 Biotech – The unexpected journey into biotech entrepreneurship, providing GPCR profiling Interdisciplinary Research & Future Directions – Exploring combinatorial drug actions, receptor interactions In 2021 he co-founded Z7 Biotech, developing and providing innovative GPCR drug screening and precision GPCR Podcast? Leave a Review.
- Dr. Mark Connor | Dr. GPCR Ecosystem
Focus on study of drugs and toxins on GPCR (opioid, cannabinoid receptor) and ion channel (K, Ca, TRP GPCR Ecosystem Enjoying the Dr. GPCR Podcast? Leave a Review. Better Questions in Science: A Practical Guide for Emerging Researchers When the Islet Lit Up: Advancing GPCR Imaging in Native Tissue How Collaboration Sparked a GPCR Imaging Breakthrough in Chemical Biology Thanks
- Dr. Terry Kenakin | Dr. GPCR Ecosystem
His interests are in receptor pharmacology, allosteric protein function, and drug discovery. Dr. GPCR Ecosystem Enjoying the Dr. GPCR Podcast? Leave a Review. Better Questions in Science: A Practical Guide for Emerging Researchers When the Islet Lit Up: Advancing GPCR Imaging in Native Tissue How Collaboration Sparked a GPCR Imaging Breakthrough in Chemical Biology Thanks
- GPCR Retreat Logo Contest | Dr. GPCR Ecosystem
Unleash your creativity with this logo contest for the GPCR Retreat 23. Design our brand's identity today! Retreat Logo Contest In anticipation of the next GPCR Retreat, we are delighted to announce the GPCR The winning logo designer will receive well-deserved recognition and a cash prize of $250. Transmembranaires du Québec 22nd GPCR Retreat Sponsored by
- Dr. Gunnar Schulte | Dr. GPCR Ecosystem
Molecular Neurobiology; 2003-2005) and later with Roger J Summers (Monash University, Melbourne Australia, GPCR ultimate aim is to use the new knowledge to find, create and optimize Frizzled-targeting small molecule drugs GPCR Ecosystem Enjoying the Dr. GPCR Podcast? Leave a Review. Better Questions in Science: A Practical Guide for Emerging Researchers When the Islet Lit Up: Advancing GPCR Imaging in Native Tissue How Collaboration Sparked a GPCR Imaging Breakthrough in Chemical Biology Thanks



















