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colleagues and Alfred Gillman , co-recipient of the 1994 Nobel Prize in Physiology or Medicine for their discovery , Paul and his team focus on previously unrecognized receptors with the hopes to use these as novel drug GPCR Ecosystem Enjoying the Dr. GPCR Podcast? Leave a Review. Better Questions in Science: A Practical Guide for Emerging Researchers When the Islet Lit Up: Advancing GPCR Imaging in Native Tissue How Collaboration Sparked a GPCR Imaging Breakthrough in Chemical Biology Thanks

He has been also studying what aspects of GPCR signaling are regulated in a sex-selective manner and how this can influence drug discovery in the area of neurodegenerative diseases. GPCR Ecosystem Enjoying the Dr. GPCR Podcast? Leave a Review. Better Questions in Science: A Practical Guide for Emerging Researchers When the Islet Lit Up: Advancing GPCR Imaging in Native Tissue How Collaboration Sparked a GPCR Imaging Breakthrough in Chemical Biology Thanks

GPCR Affiliate Program and earn commissions by helping connect the global GPCR community. Share our ecosystem, courses, and events to advance drug discovery together. Dr. GPCR community. GPCR brand ambassador affiliate program Who can be a Dr. GPCR ambassador? GPCR Ecosystem?

His interests are in receptor pharmacology, allosteric protein function, and drug discovery. Dr. GPCR Ecosystem Enjoying the Dr. GPCR Podcast? Leave a Review. Better Questions in Science: A Practical Guide for Emerging Researchers When the Islet Lit Up: Advancing GPCR Imaging in Native Tissue How Collaboration Sparked a GPCR Imaging Breakthrough in Chemical Biology Thanks

GPCR Ecosystem. Get guidance, strategies, and insights to optimize your GPCR research and drug discovery projects. Any CRO focused on GPCRs, pharmacology, discovery biology, or antibody discovery—regardless of size or Power My Discovery Send me a message First name* Last name Company name* Email* How Can I Help? Let’s talk about how I support GPCR discovery, pharmacology strategy, and cross-functional execution

He is a world-renowned expert in the field of cell signaling and GPCRs and made seminal contributions to our understanding of this major class of drug targets. energy transfer (BRET) resulted in the development of screening assays that are now widely used for drug discovery. GPCR Ecosystem Enjoying the Dr. GPCR Podcast? Leave a Review.

His research focuses on novel paradigms of drug action at GPCRs, particularly allosteric modulation and discovery. They also explored the significance of translating fundamental discoveries into clinical applications Translating Discovery Into Clinical Application Arthur and Yamina discussed the importance of translating They also emphasized the significance of fundamental discoveries, the role of biotech, and the need for

His research focuses on novel paradigms of drug action at GPCRs, particularly allosteric modulation and discovery. They also explored the significance of translating fundamental discoveries into clinical applications Translating Discovery Into Clinical Application Arthur and Yamina discussed the importance of translating They also emphasized the significance of fundamental discoveries, the role of biotech, and the need for

pharmacology into creating this essential resource, designed to meet you exactly where you are in your drug discovery journey. Bridge theory to practical drug development decisions? #pharmacology #GPCRscience #drugdiscovery #TerrysCorner #biotechtraining #ScienceEducation #Pharma #GPCR

🌟 This discovery reveals an unusual dual binding mode of FFA and offers tools for site-targeted compound 🌟 This discovery reveals an unusual dual binding mode of FFA and offers tools for site-targeted compound signaling. ➡️ https://www.ecosystem.drgpcr.com/receptor-activation-and-signaling/a-bitter-anti-inflammatory-drug-binds-at-two-distinct-sites-of-a-human-bitter-taste-gpcr And that’s exactly what carries strong discovery programs into 2026. Dr. Yet discovery teams routinely lose time and misallocate resources because the underlying biology behaves

These receptors belong to the super-family of G-protein coupled receptors (GPCR), the major molecular target for drug development. and drug development technology. GPCR Ecosystem Enjoying the Dr. GPCR Podcast? Leave a Review. Imaging in Native Tissue How Collaboration Sparked a GPCR Imaging Breakthrough in Chemical Biology Thanks

Join industry leaders as they share insights, stories, and groundbreaking discoveries, enriching our Exploring discoveries, careers, and ideas shaping human health. In each episode, we sit down with leading experts to explore their career journeys, groundbreaking discoveries GPCR Podcast was created with three goals: Share discoveries – Highlight the latest advances in the GPCR Fill out this form Be our Guest In each episode, we chat with an expert about their career trajectory, discoveries

Full Agenda Adhesion GPCR workshop 2024 CINVESTAV, Mexico City, Mexico October 23-25 Download PDF Program formation, maintenance and degeneration Yimin Zou Antibody-drug conjugates targeting CD97 in glioblastoma Yimin Zou on the web UC San Diego Antibody-drug conjugates targeting CD97 in glioblastoma Dimitris Placantonakis To exploit this expression profile, we have developed antibody-drug conjugates (ADCs) targeting CD97, GPCR < Previous Session Next Session >

GPCR Newsletter 📰 and get the latest GPCR News delivered to your inbox. the GPCR G protein subtype selectivity? GPCR Newsletter 📰 and get the latest GPCR News delivered to your inbox. ➡ https:// www.ecosystem.drgpcr.com /gpcr-binders-drugs-and-more/design-of-allosteric-modulators-that-change-gpcr-g-protein-subtype-selectivity #gpcr #drgpcr Previous Next Recent Articles

<< Back to podcast list Strategic Partner(s) GPCR location matters with Dr. In my PhD, I studied the nanoscale spatial organization of G protein-coupled receptors (GPCRs) at the revealed heterogeneous spatial patterns of receptor density and activation, that are modulated in a drug-dependent These findings identify nanoscale GPCR spatial organization as an integral element of their activity GPCR Podcast? Leave a Review.

Weekly News, featuring expert insights on target engagement, a practical framework for irreversible drugs GPCR Weekly News - Oct 23 - The Power and Peril of Irreversible Drugs Published on October 23, 2025 Category GPCR Weekly News This week’s Weekly News breaks down how to control target engagement—so duration, penetration Premium sneak peek inside. 🔹 Terry’s Corner: A practical framework for irreversible drugs—defining “ #DrGPCR #GPCR Previous Next Recent Articles

Karine Pichavant , I contributed to the development of a drug to treat hypovolemic shock after severe Cone was the first to clone the melanocortin receptors (the GPCRs that led to the discovery of MRAP2) In-vivo techniques, I adapted my arrestin recruitment assay to a high throughput screening format for drug discovery, I have started molecular work on the melanocortin receptors. GPCR Enjoying the Dr. GPCR Podcast? Leave a Review.

Discover how enzyme inhibition can enhance drug discovery strategies. Home → Flash News → Weekly News October 16 Published on October 16, 2025 Category GPCR Weekly News Enzymes This week’s Weekly News is your practical guide to building enzyme inhibition into discovery—not as a And that’s exactly what carries strong discovery programs into 2026. Dr. Yet discovery teams routinely lose time and misallocate resources because the underlying biology behaves

Every receptor tells a story but GPCRs speak a language of organization. Dr. Michelle Halls unpacks how GPCR signaling isn’t just about ligand–receptor interaction. Michelle Halls unpacks how GPCR signaling isn’t just about ligand–receptor interaction. level of organization defines specificity in signaling, and understanding it changes how we think about drug signaling: 👉 https://www.ecosystem.drgpcr.com/dr-gpcr-podcast/leadership-luck-and-gpcr-signaling #GPCR

During his Ph.D. with David Gloriam at the Department of Drug Design and Pharmacology in Copenhagen, of Molecular Biology in Cambridge, UK, where he was working on the impact of genetic variations on drug Award” for his work on GPCRs. Dr. Alexander S. GPCR Ecosystem Enjoying the Dr. GPCR Podcast? Leave a Review. Imaging in Native Tissue How Collaboration Sparked a GPCR Imaging Breakthrough in Chemical Biology Thanks

into the structure, dynamics, and function of important classes of membrane proteins and prominent drug targets, including G protein-coupled receptors (GPCRs), transporters, channels, and 3 integrins. To this end, her lab uses several computational structural biology tools and rational drug design approaches GPCR Ecosystem Enjoying the Dr. GPCR Podcast? Leave a Review. Imaging in Native Tissue How Collaboration Sparked a GPCR Imaging Breakthrough in Chemical Biology Thanks

Full Agenda Adhesion GPCR workshop 2024 CINVESTAV, Mexico City, Mexico October 23-25 Download PDF Program GPCR Community Presentation Breaking Barriers: My Journey from Mexico to the Heart of the Dr. GPCR Ecosystem and beyond About Monserrat Avila Zozaya "My doctoral research was focused on investigating My research focuses on understanding the molecular mechanisms of adhesion GPCRs (aGPCRs) in lymphatic GPCR < Previous Session Next Session >

Kenakin shows how experimental snapshots can reveal much more—and how predictive frameworks guide modern drug discovery. 🟢 Built for pharmacologists building stronger pipelines and those rethinking legacy models . ✳️ https://www.terrykenakin.com #GPCR #DrGPCR #pharmacology #drugmodeling #terrykenakin Previous Next And that’s exactly what carries strong discovery programs into 2026. Dr. Yet discovery teams routinely lose time and misallocate resources because the underlying biology behaves

Join Terry’s Corner AMA to master GPCR signaling, allosteric modulation, and kinetic strategy in drug discovery. In the discovery phase, one overlooked kinetic parameter or a misjudged model can set your team back Don’t fall behind on what will shape the next decade of discovery. And that’s exactly what carries strong discovery programs into 2026. Dr.

Pierre Eftekhari "Clinical physiologist and biologist , with more than 25 years of experience in drug development. have been engaged in GPCR cellular and clinical pharmacology as scientist or PI in neonatal I have participated and initiated methodologies for development of pharmacologically active anti-GPCR or contributed in 38 published scientific work mainly in the field of immunology and pharmacology of GPCR GPCR Enjoying the Dr. GPCR Podcast? Leave a Review.

Full Agenda Adhesion GPCR workshop 2024 CINVESTAV, Mexico City, Mexico October 23-25 Download PDF Program Activation: Direct Communication of Extracellular Region with Transmembrane Domain in a Holo-Adhesion GPCR point mutant knock-in mouse, H381S Frank Kwarcinski Tethered Peptide Activation Mechanism of Adhesion GPCRs ECR-mediated mechanism opens new possibilities for drugging aGPCRs. Frank Kwarcinski on the web LinkedIn Tethered Peptide Activation Mechanism of Adhesion GPCRs Peng Xiao

Michelle describes how reading those early papers on lipid-rich domains and GPCR–G protein compartmentalization This moment cuts straight to the heart of how many of us fell in love with GPCR biology — that realization The way signals are organized defines specificity, drug response, and potential for targeted therapies /leadership-luck-and-gpcr-signaling ✨ Join Premium: https://www.ecosystem.drgpcr.com/gpcr-university-pricing #GPCR #DrGPCR Previous Next Recent Articles

the University of Glasgow, his primary research interests are focused on the rational design of novel drugs staff supported by basic research grants investigating aspects of disease biology and the action of drugs GPCR Ecosystem Enjoying the Dr. GPCR Podcast? Leave a Review. Better Questions in Science: A Practical Guide for Emerging Researchers When the Islet Lit Up: Advancing GPCR Imaging in Native Tissue How Collaboration Sparked a GPCR Imaging Breakthrough in Chemical Biology Thanks

He introduced molecular pharmacology to a wide range of the company's GPCR projects and was able to initiate He also discovered and championed a novel prostaglandin EP4 drug candidate for development. GPCR Ecosystem Enjoying the Dr. GPCR Podcast? Leave a Review. Better Questions in Science: A Practical Guide for Emerging Researchers When the Islet Lit Up: Advancing GPCR Imaging in Native Tissue How Collaboration Sparked a GPCR Imaging Breakthrough in Chemical Biology Thanks

<< Back to podcast list Strategic Partner(s) The Role of Quantitative Sciences in GPCRs with Dr. molecular dynamics simulation methods with emphasis on application to G-protein coupled receptors and drug GPCR Enjoying the Dr. GPCR Podcast? Leave a Review. Better Questions in Science: A Practical Guide for Emerging Researchers When the Islet Lit Up: Advancing GPCR Imaging in Native Tissue How Collaboration Sparked a GPCR Imaging Breakthrough in Chemical Biology Thanks