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His research focuses on novel paradigms of drug action at GPCRs, particularly allosteric modulation and discovery. They also explored the significance of translating fundamental discoveries into clinical applications Translating Discovery Into Clinical Application Arthur and Yamina discussed the importance of translating They also emphasized the significance of fundamental discoveries, the role of biotech, and the need for

Discover how enzyme inhibition can enhance drug discovery strategies. Home → Flash News → Weekly News October 16 Published on October 16, 2025 Category GPCR Weekly News Enzymes This week’s Weekly News is your practical guide to building enzyme inhibition into discovery—not as a #DrGPCR #GPCR Previous Next Recent Articles

GPCR Podcast Strategic Partners Dr. Jean Martin Beaulieu About Dr. Jean Martin Beaulieu Dr. These receptors belong to the super-family of G-protein coupled receptors (GPCR), the major molecular target for drug development. and drug development technology. GPCR Ecosystem Enjoying the Dr. GPCR Podcast? Leave a Review.

GPCR Ecosystem. Get guidance, strategies, and insights to optimize your GPCR research and drug discovery projects. Any CRO focused on GPCRs, pharmacology, discovery biology, or antibody discovery—regardless of size or Power My Discovery Send me a message First name* Last name Company name* Email* How Can I Help? Let’s talk about how I support GPCR discovery, pharmacology strategy, and cross-functional execution

GPCR Affiliate Program and earn commissions by helping connect the global GPCR community. Share our ecosystem, courses, and events to advance drug discovery together. Dr. GPCR community. GPCR brand ambassador affiliate program Who can be a Dr. GPCR ambassador? GPCR Ecosystem?

pharmacology into creating this essential resource, designed to meet you exactly where you are in your drug discovery journey. Bridge theory to practical drug development decisions? #pharmacology #GPCRscience #drugdiscovery #TerrysCorner #biotechtraining #ScienceEducation #Pharma #GPCR

Next Recent Articles Decoding Schild Analysis: The Pharmacologist’s Lens on Competitive Antagonism Drug discovery often assumes receptor inhibition follows simple rules—agonist binds, antagonist blocks, and GPCR Podcast 2 days ago How GPCR Spatial Signaling Sparked a Scientific Journey Michelle hadn’t mapped GPCR Podcast 4 days ago Molecular creativity in drug discovery Most pharmacologists are trained to chase GPCR News 5 days ago

Kenakin shows how experimental snapshots can reveal much more—and how predictive frameworks guide modern drug discovery. 🟢 Built for pharmacologists building stronger pipelines and those rethinking legacy models . ✳️ https://www.terrykenakin.com #GPCR #DrGPCR #pharmacology #drugmodeling #terrykenakin Previous Next

Join industry leaders as they share insights, stories, and groundbreaking discoveries, enriching our Exploring discoveries, careers, and ideas shaping human health. In each episode, we sit down with leading experts to explore their career journeys, groundbreaking discoveries GPCR Podcast was created with three goals: Share discoveries – Highlight the latest advances in the GPCR Fill out this form Be our Guest In each episode, we chat with an expert about their career trajectory, discoveries

Karine Pichavant , I contributed to the development of a drug to treat hypovolemic shock after severe Cone was the first to clone the melanocortin receptors (the GPCRs that led to the discovery of MRAP2) In-vivo techniques, I adapted my arrestin recruitment assay to a high throughput screening format for drug discovery, I have started molecular work on the melanocortin receptors. GPCR Enjoying the Dr. GPCR Podcast? Leave a Review.

GPCR Newsletter 📰 and get the latest GPCR News delivered to your inbox. the GPCR G protein subtype selectivity? GPCR Newsletter 📰 and get the latest GPCR News delivered to your inbox. ➡ https:// www.ecosystem.drgpcr.com /gpcr-binders-drugs-and-more/design-of-allosteric-modulators-that-change-gpcr-g-protein-subtype-selectivity #gpcr #drgpcr Previous Next Recent Articles

GPCR Podcast Strategic Partners Dr. Alexander S. Hauser About Dr. Alexander S. During his Ph.D. with David Gloriam at the Department of Drug Design and Pharmacology in Copenhagen, of Molecular Biology in Cambridge, UK, where he was working on the impact of genetic variations on drug Award” for his work on GPCRs. Dr. Alexander S. GPCR Ecosystem Enjoying the Dr. GPCR Podcast? Leave a Review.

GPCR Podcast Strategic Partners Dr. Marta Filizola About Dr. Marta Filizola Dr. into the structure, dynamics, and function of important classes of membrane proteins and prominent drug targets, including G protein-coupled receptors (GPCRs), transporters, channels, and 3 integrins. To this end, her lab uses several computational structural biology tools and rational drug design approaches GPCR Ecosystem Enjoying the Dr. GPCR Podcast? Leave a Review.

Full Agenda Adhesion GPCR workshop 2024 CINVESTAV, Mexico City, Mexico October 23-25 Download PDF Program formation, maintenance and degeneration Yimin Zou Antibody-drug conjugates targeting CD97 in glioblastoma Yimin Zou on the web UC San Diego Antibody-drug conjugates targeting CD97 in glioblastoma Dimitris Placantonakis To exploit this expression profile, we have developed antibody-drug conjugates (ADCs) targeting CD97, GPCR < Previous Session Next Session >

Weekly News, featuring expert insights on target engagement, a practical framework for irreversible drugs GPCR Weekly News - Oct 23 - The Power and Peril of Irreversible Drugs Published on October 23, 2025 Category GPCR Weekly News This week’s Weekly News breaks down how to control target engagement—so duration, penetration Premium sneak peek inside. 🔹 Terry’s Corner: A practical framework for irreversible drugs—defining “ #DrGPCR #GPCR Previous Next Recent Articles

GPCR Podcast Strategic Partners Dr. Andrew Tobin About Dr. the University of Glasgow, his primary research interests are focused on the rational design of novel drugs staff supported by basic research grants investigating aspects of disease biology and the action of drugs GPCR Ecosystem Enjoying the Dr. GPCR Podcast? Leave a Review. Collaboration Built an Innovation Engine From Pipettes to Platforms: The Evolution of GPCR Research

Full Agenda Adhesion GPCR workshop 2024 CINVESTAV, Mexico City, Mexico October 23-25 Download PDF Program GPCR Community Presentation Breaking Barriers: My Journey from Mexico to the Heart of the Dr. GPCR Ecosystem and beyond About Monserrat Avila Zozaya "My doctoral research was focused on investigating My research focuses on understanding the molecular mechanisms of adhesion GPCRs (aGPCRs) in lymphatic GPCR < Previous Session Next Session >

GPCR Podcast Strategic Partners Dr. Steven Foord About Dr. He also discovered and championed a novel prostaglandin EP4 drug candidate for development. GPCR Ecosystem Enjoying the Dr. GPCR Podcast? Leave a Review. Collaboration Built an Innovation Engine From Pipettes to Platforms: The Evolution of GPCR Research How GPCR Spatial Signaling Sparked a Scientific Journey Thanks for listening to this podcast episode

GPCR Podcast Strategic Partners The Role of Quantitative Sciences in GPCRs with Dr. molecular dynamics simulation methods with emphasis on application to G-protein coupled receptors and drug GPCR Enjoying the Dr. GPCR Podcast? Leave a Review. Collaboration Built an Innovation Engine From Pipettes to Platforms: The Evolution of GPCR Research How GPCR Spatial Signaling Sparked a Scientific Journey Thanks for listening to this podcast episode

GPCR Podcast Strategic Partners Dr. Pierre Eftekhari About Dr. Pierre Eftekhari "Clinical physiologist and biologist , with more than 25 years of experience in drug development. have been engaged in GPCR cellular and clinical pharmacology as scientist or PI in neonatal I have participated and initiated methodologies for development of pharmacologically active anti-GPCR GPCR Enjoying the Dr. GPCR Podcast? Leave a Review.

GPCR Podcast Strategic Partners Steve McCloskey About Steve McCloskey Steve McCloskey is an Alumni from Scientists and Engineers working at the nanoscale, specifically protein engineering and small molecule drug GPCR Ecosystem Enjoying the Dr. GPCR Podcast? Leave a Review. Collaboration Built an Innovation Engine From Pipettes to Platforms: The Evolution of GPCR Research How GPCR Spatial Signaling Sparked a Scientific Journey Thanks for listening to this podcast episode

GPCR Podcast Strategic Partners Dr. Lauren M. Slosky About Dr. Lauren M. Lauren Slosky is an Assistant Professor in the Department of Pharmacology and a member of the Medical Discovery within the University of Minnesota’s Medical School to advance research and treatment in the field of drug Slosky’s research is focused on understanding how neuropeptide G protein-coupled receptors (GPCRs) regulate GPCR Ecosystem Enjoying the Dr. GPCR Podcast? Leave a Review.

Michelle describes how reading those early papers on lipid-rich domains and GPCR–G protein compartmentalization This moment cuts straight to the heart of how many of us fell in love with GPCR biology — that realization The way signals are organized defines specificity, drug response, and potential for targeted therapies /leadership-luck-and-gpcr-signaling ✨ Join Premium: https://www.ecosystem.drgpcr.com/gpcr-university-pricing #GPCR #DrGPCR Previous Next Recent Articles

Full Agenda Adhesion GPCR workshop 2024 CINVESTAV, Mexico City, Mexico October 23-25 Download PDF Program Activation: Direct Communication of Extracellular Region with Transmembrane Domain in a Holo-Adhesion GPCR point mutant knock-in mouse, H381S Frank Kwarcinski Tethered Peptide Activation Mechanism of Adhesion GPCRs ECR-mediated mechanism opens new possibilities for drugging aGPCRs. Frank Kwarcinski on the web LinkedIn Tethered Peptide Activation Mechanism of Adhesion GPCRs Peng Xiao

Subscribe to the Adhesion GPCR Workshop 2024 newsletter. Adhesion GPCR workshop 2024 CINVESTAV, Mexico City, Mexico October 23-25 Register AGPCR Newsletter Adhesion GPCR Consortium Newsletter - May 2024 Welcome to the 4th official Adhesion GPCR Consortium newsletter GPCR News Register for the Adhesion GPCR 2024 Learn more about the Adhesion GPCR workshop 2024 Up About the event Learn more about the Adhesion GPCR workshop 2024 and its preliminary program.

GPCR Podcast Strategic Partners Dr. Claudia Stäubert About Dr. Umeå, Sweden), I broadened my methodical and scientific horizon and focused on cellular metabolism and drug Metabolite Activation of GPCRs: A Fascinating Discovery Claudia and Yamina discussed the role of metabolites in activating GPCRs, a process that they found fascinating. GPCR Podcast? Leave a Review.

They also discussed the ongoing developments in the GPCR field, the upcoming adhesion GPCR consortium Demet explained that since the year 2000, the field has seen significant growth, with important discoveries adhesion GPCRs. also discussed the importance of the extracellular region of these receptors and its potential as a drug GPCR Podcast? Leave a Review.

GPCR Podcast! Explore the fascinating career journeys, groundbreaking discoveries, and impactful contributions of experts We discuss breakthrough discoveries, career paths in pharmacology and molecular biology, and how each If you’re working on exciting GPCR-related research — from structural biology to drug discovery — we’ GPCR Podcast with three major goals in mind: Share the latest scientific discoveries in the GPCR field

GPCR Podcast Strategic Partners Dr. Mark Connor About Dr. Focus on study of drugs and toxins on GPCR (opioid, cannabinoid receptor) and ion channel (K, Ca, TRP GPCR Ecosystem Enjoying the Dr. GPCR Podcast? Leave a Review. Collaboration Built an Innovation Engine From Pipettes to Platforms: The Evolution of GPCR Research How GPCR Spatial Signaling Sparked a Scientific Journey Thanks for listening to this podcast episode

GPCR Podcast Strategic Partners Dr. Graeme Milligan About Dr. main research group centers on the function, structure, and regulation of G protein-coupled receptors (GPCRs and identification of small molecule regulators of these proteins, and progressing such ligands in drug GPCR Ecosystem Enjoying the Dr. GPCR Podcast? Leave a Review. Collaboration Built an Innovation Engine From Pipettes to Platforms: The Evolution of GPCR Research