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- Mexico City Nocturnal Tour, Food and drinks | Adhesion GPCR Workshop 2024 | Dr. GPCR Ecosystem
Full Agenda Adhesion GPCR workshop 2024 CINVESTAV, Mexico City, Mexico October 23-25 Download PDF Program
- Targeting adenosine signaling for immuno-oncology
Retreat 2023 About Program Registration Logo Contest Committee Sponsors GPCR Retreat Program < Back to clinical stage company developing next generation immunotherapies, and member of the SAB of Domain Therapeutics , a biopharmaceutical company focused on GPCR in immuno-oncology." GPCR Previous Event Next Event Great Lakes GPCR Retreat and Club des Récepteurs à Sept Domaines Transmembranaires 22nd GPCR Retreat Sponsored by
- Exploring the combination of molecular simulation, pharmacological assays, and NMR to reveal the molecular mechanism of biased activation at the vasopressin V2 receptor. Did you know that we work hard to bring you the most recent GPCR News, weekly? Catch up today in the Ecosystem using your free site membership! | Dr. GPCR Ecosystem
Did you know that we work hard to bring you the most recent GPCR News, weekly? Published on December 10, 2024 Category GPCR Weekly News Exploring the combination of molecular simulation Did you know that we work hard to bring you the most recent GPCR News, weekly? Breakthroughs this week: Potentiation of GPCR signaling by ATP and sugar monophosphates; Pharmacology Oct 14 Assay Volume Control: Your GPCR Drug Discovery Power Lever If you want cleaner decisions, start
- Partners Submition Form | Dr. GPCR Ecosystem
GPCR Ecosystem and collaborate with us to make a positive impact.
- Generic tools won’t solve tomorrow’s drug discovery challenges. That’s why Celtarys designs custom fluorescent probes for every target, built for real pharmacology, not just convenience. With Dr. GPCR and Celtarys joining forces, expect more visibility, more precision, and more scientific impact. 🚀 Get to know our media partner: https://www.ecosystem.drgpcr.com/celtarys-research-dr-gpcr-ecosystem #GPCRdrugDiscovery #GPCRecosystem #CustomLigands | Dr. GPCR Ecosystem
GPCR and Celtarys joining forces, expect more visibility, more precision, and more scientific impact. 🚀 Get to know our media partner: https://www.ecosystem.drgpcr.com/celtarys-research-dr-gpcr-ecosystem GPCR and Celtarys joining forces, expect more visibility, more precision, and more scientific impact. 🚀 Get to know our media partner: https://www.ecosystem.drgpcr.com/celtarys-research-dr-gpcr-ecosystem
- Terms and Conditions | Dr. GPCR Ecosystem
GPCR Ecosystem. Explore our Terms and Conditions page now! Terms and Conditions Dr. GPCR, Corp (“Dr. GPCR”) provides its Service to you through our websites referred to as Dr. GPCR, Ecosystem.DrGPCR.com, DrGPCR.com. 1. GPCR, Corp (“Dr. GPCR, Corp (“Dr. GPCR”) may change this ATS from time to time without prior notice.
- Ep 167 with Drs. Tom Sakmar & Ilana Kotliar
GPCR signaling in disease. GPCR Podcast << Back to podcast list Hacking GPCRs: Tools, Tech & Drug Discovery with Tom Sakmar & Ilana This could accelerate discovery of therapeutic targets by combining multiplex data with focused downstream Keyword Cloud GPCR-RAMP interactions , multiplex assays , GPCR research community , Dr. GPCR ecosystem , GPCR data platform , GPCR autoantibodies , Addgene GPCR library , GPCR training program
- Seeking to gain more knowledge on signaling bias? We’ve got the perfect opportunity for you 🚀 Registrations open until February 14th ⚠️ Last spots available for “The Practical Assessment of Signaling Bias” with Dr. Terry Kenakin ✳️Register today at https://www.ecosystem.drgpcr.com/event-details-registration/the-practical-assessment-of-signaling-bias #gpcr #drgpcr | Dr. GPCR Ecosystem
https://www.ecosystem.drgpcr.com/event-details-registration/the-practical-assessment-of-signaling-bias #gpcr GPCR Courses Seeking to gain more knowledge on signaling bias? a strategic edge. 11 hours ago How Breakthroughs Happen: Eric Trinquet on Innovation, Serendipity & GPCRs Breakthroughs this week: Potentiation of GPCR signaling by ATP and sugar monophosphates; Pharmacology Oct 14 Assay Volume Control: Your GPCR Drug Discovery Power Lever If you want cleaner decisions, start
- Ep 152 with Dr Arthur Christopoulos
Award and the Goodman and Gilman Award from the American Society for Pharmacology and Experimental Therapeutics They explored the evolution of the field, allosteric modulation concepts, and potential therapeutic approaches Arthur will work on designing ligands for specific receptors, aiming to create biased agonists for therapeutic Yamina discussed the potential of autoantibodies and allosteric modulation in the context of disease and therapeutic endogenous allosteric ligands and the possibility of using a neutral allosteric ligand as a preferred therapeutic
- Ep 146 with Dr Michael Feigin
Michael Feigin is an Associate Professor in the Department of Pharmacology and Therapeutics, and Director of Graduate Studies of Experimental Therapeutics at Roswell Park Comprehensive Cancer Center in Buffalo GPCR Targeted Drugs and Gene Regulation in Cancer Cells Mike presented research on the effect of GPCR-targeted disrupting histone processing on rapidly proliferating cells, such as cancer cells, and suggested a therapeutic GPCR Podcast? Leave a Review.
- Ep 153 with Dr Jacek Mokrosiński
GPCR Podcast << Back to podcast list Exploring Career Paths in GPCR Research with Dr. Yamina will schedule a future talk with Jacek about GPCRs as therapeutic modalities. their research interests and achievements, particularly in the field of GPCR. The discussion revealed their interest in GPCRs as therapeutic modalities and possible future collaborations GPCR Podcast? Leave a Review.
- Distinct sub-cellular signal propagation as a component of functional selectivity
Retreat 2023 About Program Registration Logo Contest Committee Sponsors GPCR Retreat Program < Back to He is a world-renowned expert in the field of cell signaling and GPCRs and made seminal contributions of Canada (2014), the Julie Axelrod award from the American Society of Pharmacology and Exerimental Therapeutics GPCR Previous Event Next Event Great Lakes GPCR Retreat and Club des Récepteurs à Sept Domaines Transmembranaires 22nd GPCR Retreat Sponsored by
- Ep 80 with Dr. Andrew Tobin
GPCR Podcast << Back to podcast list Dr. Andrew Tobin About Dr. vehicle by which Andrew is translating fundamental findings to commercial products is Keltic Pharma Therapeutics GPCR Ecosystem Enjoying the Dr. GPCR Podcast? Leave a Review. Apple Podcasts ★ Rate on Spotify ✉️ Send feedback to the team Recent Podcast Articles The Truth About GPCR Making Innovative Data-Driven Solutions: The pHSense Revolution How a Failed Med School Dream Sparked a GPCR
- 🚀 New Workshop: Practical Quantification of Allosteric Modulation Join Dr. Terry Kenakin on May 1st, 2025, for an advanced live workshop on allosteric modulators in GPCR drug discovery. Learn how to: ✔️ Identify, measure, and quantify allosteric properties ✔️ Apply functional allosteric models to determine mechanisms of action ✔️ Confirm allostery through kinetic analysis 📅 Date: May 1st, 2025 ⏳ Registration deadline: April 18th 📍 Live on Google Meet 🔗 Register now: https://www.ecosystem.drgpcr.com/event-details-registration/practical-quantification-of-allosteric-modulation #GPCR #Allostery #DrugDiscovery #Pharmacology | Dr. GPCR Ecosystem
Terry Kenakin on May 1st, 2025, for an advanced live workshop on allosteric modulators in GPCR drug discovery www.ecosystem.drgpcr.com/event-details-registration/practical-quantification-of-allosteric-modulation #GPCR Terry Kenakin on May 1st, 2025 , for an advanced live workshop on allosteric modulators in GPCR drug Breakthroughs this week: Potentiation of GPCR signaling by ATP and sugar monophosphates; Pharmacology Oct 14 Assay Volume Control: Your GPCR Drug Discovery Power Lever If you want cleaner decisions, start
- Content Guidelines | Dr. GPCR Ecosystem
GPCR Ecosystem website. Get the information you need to create engaging and impactful content. GPCR, Corp, LLC (“Dr. GPCR”) provides its Service to you through our websites referred to as Dr. GPCR, Ecosystem.DrGPCR.com, DrGPCR.com. Please note that Ecosystem.DrGPCR.com is specializes in GPCR and related subjects. GPCR conducts business Affiliate Policy Content and Conduct Policy Content Guidance Privacy Policy Terms
- Removing the GPCR-mediated brake on exocytosis enhances insulin action, promotes adipocyte browning, and protects against diet-induced obesity
Retreat 2023 About Program Registration Logo Contest Committee Sponsors GPCR Retreat Program < Back to schedule Removing the GPCR-mediated brake on exocytosis enhances insulin action, promotes adipocyte The Department’s strengths lie in GPCR signal transduction and neuroscience, and she has expanded it GPCR Previous Event Next Event Great Lakes GPCR Retreat and Club des Récepteurs à Sept Domaines Transmembranaires 22nd GPCR Retreat Sponsored by
- In case you haven’t heard, our next Dr.GPCR University course is open for registrations 🙂 Learn about "The Practical Assessment of Signaling Bias" with Dr. Terry Kenakin. 🙌 Hands-on exercises included! ✳️Only 25 spots available ➡️Enjoy a 25% discount with your Premium Membership https://www.ecosystem.drgpcr.com/event-details-registration/the-practical-assessment-of-signaling-bias #gpcr #drgpcr | Dr. GPCR Ecosystem
https://www.ecosystem.drgpcr.com/event-details-registration/the-practical-assessment-of-signaling-bias #gpcr #drgpcr Published on January 24, 2025 Category GPCR University In case you haven’t heard, our next Dr.GPCR a strategic edge. 11 hours ago How Breakthroughs Happen: Eric Trinquet on Innovation, Serendipity & GPCRs Breakthroughs this week: Potentiation of GPCR signaling by ATP and sugar monophosphates; Pharmacology Oct 14 Assay Volume Control: Your GPCR Drug Discovery Power Lever If you want cleaner decisions, start
- How do GRK-specific phosphorylation barcodes influence β-arrestin binding to GPCRs? New cryo-EM structures from Chen et al. (Nature, 2025) reveal that β-arrestin1 and β-arrestin2 form distinct complexes with ACKR3 depending on whether it's phosphorylated by GRK2 or GRK5, shaping arrestin conformation, complex stability, and engagement mode. Surprisingly, arrestin’s finger loop didn’t dive into the receptor core. Instead, it latched onto the micelle surface, breaking canonical expectations. Also, β-arrestin2 lacks a membrane anchor, making it more dynamic — a potential clue to its functional specialization. These findings underscore how barcode location + arrestin isoform = unique signaling outcomes. open book Read the full study: Inside Out: Mapping GPCRs from Membrane Codes to Market Moves #GPCRs #Arrestin #ACKR3 #GRKs #CryoEM #StructuralBiology #SignalingBias #Phosphorylation #DrGPCR | Dr. GPCR Ecosystem
Home → Flash News → How do GRK-specific phosphorylation barcodes influence β-arrestin binding to GPCRs + arrestin isoform = unique signaling outcomes. open book Read the full study: Inside Out: Mapping GPCRs from Membrane Codes to Market Moves #GPCRs #Arrestin #ACKR3 #GRKs #CryoEM #StructuralBiology #SignalingBias barcodes influence β-arrestin binding to GPCRs? Read the full study: Inside Out: Mapping GPCRs from Membrane Codes to Market Moves #GPCRs #Arrestin #
- Ep 70 with Dr. Stephen Ferguson
GPCR Podcast << Back to podcast list Dr. Stephen Ferguson About Dr. Stephen Ferguson Dr. Brian Collier in the Department of Pharmacology and Therapeutics at McGill University (1994). GPCR Ecosystem Enjoying the Dr. GPCR Podcast? Leave a Review. Apple Podcasts ★ Rate on Spotify ✉️ Send feedback to the team Recent Podcast Articles The Truth About GPCR Making Innovative Data-Driven Solutions: The pHSense Revolution How a Failed Med School Dream Sparked a GPCR
- New strategic partnership alert! 🚀 Dr.GPCR x Celtarys are teaming up to revolutionize fluorescent ligand development for GPCR research. Get custom, fast, and functional ligands backed by real scientists solving real assay problems. 🧪 “We don’t just deliver compounds. We solve assay problems.” – Dr. Maria Majellaro, CSO, Celtarys Listen to Ep. 168 now and meet your new assay partner 😉 ✳️ https://www.ecosystem.drgpcr.com/dr-gpcr-podcast/ep-168-with-dr.-maria-majellaro-from-celtarys #GPCRdrugDiscovery #FluorescentLigands #DrGPCR #BiotechTools #AssayDevelopment | Dr. GPCR Ecosystem
🚀 Dr.GPCR x Celtarys are teaming up to revolutionize fluorescent ligand development for GPCR research Celtarys Listen to Ep. 168 now and meet your new assay partner 😉 ✳️ https://www.ecosystem.drgpcr.com/dr-gpcr-podcast GPCR Podcast New strategic partnership alert! 🚀 Dr.GPCR x Celtarys are teaming up to revolutionize fluorescent ligand development for GPCR research Celtarys Listen to Ep. 168 now and meet your new assay partner 😉 ✳️ https://www.ecosystem.drgpcr.com/dr-gpcr-podcast
- Ep 166 with Dr. Ben Clements
GPCR Podcast << Back to podcast list When to Walk, When to Run: Lessons from the GPCR Trenches with Dr GPCR ecosystem , GPCR online course , GPCR scientist network , GPCR drug discovery , GPCR training program , G protein-coupled receptors , GPCR podcast , GPCR webinar series , GPCR data platform Summary created Clements' work is primarily focused on translational developments of small molecule therapeutics, and GPCR Podcast? Leave a Review.
- ⚠️Registration Deadline today! This is your last chance to register for “The Practical Assessment of Signaling Bias” with Dr. Terry Kenakin. Learn theoretical background for the techniques and apply with hands-on exercises 💪 ✳️Last chance!!! https://www.ecosystem.drgpcr.com/event-details-registration/the-practical-assessment-of-signaling-bias #gpcr #drgpcr | Dr. GPCR Ecosystem
https://www.ecosystem.drgpcr.com/event-details-registration/the-practical-assessment-of-signaling-bias #gpcr GPCR Courses ⚠️ Registration Deadline today! https://www.ecosystem.drgpcr.com/event-details-registration/the-practical-assessment-of-signaling-bias #gpcr
- Ep 36 with Dr. Michel Bouvier
GPCR Podcast << Back to podcast list Dr. Michel Bouvier About Dr. He is a world-renowned expert in the field of cell signaling and GPCRs and made seminal contributions of Canada (2014), the Julie Axelrod award from the American Society of Pharmacology and Exerimental Therapeutics been able to work with him and his team and use the tools developed in his lab to better understand GPCR GPCR Ecosystem Enjoying the Dr. GPCR Podcast? Leave a Review.
- Ben Clements reveals a 10x improvement in efficacy using GPCR-targeted PAMs, in Ep.166 of the Dr.GPCR Podcast,. The catch? It’s all about understanding the system, not replacing it. From neuromas to novel modulators, this episode is full of breakthroughs that matter for patients. 📲 Watch now: Ep 166 with Dr. Ben Clements #GPCRresearch #DrGPCR #GPCRpodcast #OpioidPharmacology #DrugDiscovery | Dr. GPCR Ecosystem
Home → Flash News → Ben Clements reveals a 10x improvement in efficacy using GPCR-targeted PAMs, in Ep GPCR Podcast Ben Clements reveals a 10x improvement in efficacy using GPCR-targeted PAMs, in Ep.166 of
- Interested in learning more about signaling bias? You’re in the right place! 🙌 Join an interactive workshop with the pharmacology master Dr. Terry Kenakin and deepen your knowledge. Reading materials are already available for registered participants 👀 ✳️ Go to https://www.ecosystem.drgpcr.com/event-details-registration/the-practical-assessment-of-signaling-bias #gpcr #drgpcr | Dr. GPCR Ecosystem
https://www.ecosystem.drgpcr.com/event-details-registration/the-practical-assessment-of-signaling-bias #gpcr GPCR Courses Interested in learning more about signaling bias? You’re in the right place! https://www.ecosystem.drgpcr.com/event-details-registration/the-practical-assessment-of-signaling-bias #gpcr
- Forget one receptor at a time. Go big.Ep.167 of the Dr.GPCR Podcast with Tom Sakmar & Ilana Kotliar is about scaling GPCR research with multiplexing, miniaturization, and collaboration. The tools are built. The data is free. What will you ask next? 📲 Dive in: Ep 167 with Drs. Tom Sakmar & Ilana Kotliar #GPCRtraining #GPCRresearchcommunity #DrGPCR #GPCRdata | Dr. GPCR Ecosystem
Go big.Ep.167 of the Dr.GPCR Podcast with Tom Sakmar & Ilana Kotliar is about scaling GPCR research with GPCR Podcast Forget one receptor at a time. Go big.Ep.167 of the Dr.GPCR Podcast with Tom Sakmar & Ilana Kotliar is about scaling GPCR research with
- Ep 170 with Dr. Alex Serafini
GPCR Podcast << Back to podcast list GPCRs and the Science Behind Pain and Recovery with Dr. analysis, revealed nuanced roles of RGS4, RGS9, and RGSZ — not just as modulators but as potential therapeutic Keyword Cloud GPCR research community, Dr. GPCR ecosystem, GPCR drug discovery, GPCR podcast, GPCR data platform, GPCR training program, RGS4, chronic GPCR Podcast? Leave a Review.
- What do mission-driven teams and world-class science have in common? ✅ Integrity ✅ Systems that last ✅ The right people In this episode, Joe & Chuck from Company Launch Partners share what it means to build something that endures. 🎧 Catch the full episode: Ep 165 with Chuck DeWeese & Joe St. Germain #gpcr #DrGPCR #ScienceStartup | Dr. GPCR Ecosystem
Germain #gpcr #DrGPCR #ScienceStartup Published on May 6, 2025 Category Dr. GPCR Podcast What do mission-driven teams and world-class science have in common? Germain #gpcr #DrGPCR #ScienceStartup Recent Articles Previous Next
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GPCR Ecosystem and promote a positive online community. Content and Conduct Policy Dr. GPCR, Corp, LLC (“Dr. GPCR”) provides its Service to you through our websites referred to as Dr. GPCR, Ecosystem.DrGPCR.com, DrGPCR.com. Please note that Ecosystem.DrGPCR.com is specializes in GPCR and related subjects. GPCR conducts business Affiliate Policy Content and Conduct Policy Content Guidance Privacy Policy Terms
- terrys corner predict drug behavior | Dr. GPCR Ecosystem
✳️ https://www.terrykenakin.com #pharmacology #drugmechanism #kenakin #GPCR #DrGPCR Recent Articles Previous
