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Results found for "Fan Liu"
- What's Going On with GPCRs?! Find Out in This Week's Update! ⊿ Nov 4 - 10, 2024
Lu GPCR-BSD: a database of binding sites of human G-protein coupled receptors under diverse states Fan Liu , Han Zhou , Xiaonong Li , Liangliang Zhou , Chungong Yu , Haicang Zhang , Dongbo Bu đ€© Seriously
- Illuminating C5aR Biology: The Role of Fluorescent Ligands in GPCR Research
.; Liu, H.; Koehler, M.; Zhang, C.; Fan, H.; Alsteens, D. Lett. 2022 , 13 (2), 243â249. https://doi.org/10.1021/acsmedchemlett.1c00598 . (7) Liu, H.; Kim, H. Y.; Fan, H.; Wei, Z.; Zhang, C. Orthosteric and Allosteric Action of the C5a Receptor Antagonists.
- đ° GPCR Weekly News, June 3 to June 9, 2024
JĂŒrgen Wess and Liu Liu for their study on A novel function of the M2 muscarinic receptor Drs.
- Conjugation Strategies for Probe Development
 (3) Fan, J.; Toth, I.; Stephenson, R. J.
- Molecular creativity in drug discovery
Welcome GPCR Fans, Most pharmacologists are trained to chase targets.
- How Schild Analysis Protects Your Conclusions in GPCR Research
Welcome back GPCR Fans, Clean data can still mislead if the underlying assumptions arenât tested.
- GPCR Allostery: Unlock Hidden Mechanisms and Make Smarter Drug Decisions
Welcome back GPCR fans, If your drug discovery strategy still relies on static GPCR models, youâre already
- đ€ŻMind-blowing GPCR Scoops! Discover the Latest Breakthroughs! ⊿ Nov 18 - 24, 2024
High-affinity agonists reveal recognition motifs for the MRGPRD GPCR Chunyu Wang , Â Yongfeng Liu , Â Marion
- Therapeutic validation of an orphan G proteinâcoupled receptor
Among these ligands are orthosteric agonists such as alkylpyrimidineâ4,6âdiol derivatives (Liu et al.
- Your GPCR Program Decisions Depend on Good Data Interpretation
Welcome GPCR Fans, Â In GPCR-targeted drug discovery, precision isnât optionalâitâs a requirement.
- đ° GPCR Weekly News, June 17 to 23, 2024
Conformation- and activation-based BRET sensors differentially report on GPCR-G protein coupling Samuel Liu
- Transmembrane domains of GPCR dimers â a novel hot spot for drug discovery
Junke Liu et al. recently provided key insights into GPCR oligomerization and biased signalling, using
- The Hidden Driver of GPCR Drug Success: Why Target Residence Time Matters More Than You Think
Hey GPCR Fans, This week's breakthroughs are crucial for staying ahead in the rapidly evolving landscape
- Why Kinetics Matter More Than Kd in GPCR Drug Discovery
Welcome GPCR Fans, Â Every discovery-phase decision you make shapes your entire pipeline trajectoryâand
- Regulators of G-protein signaling: essential players in GPCR signaling
Liu-Chen, and J.R.
- A robust and Efficient FRET-Based Assay for Cannabinoid Receptor Ligands Discovery.
.; Liu, Z.-J. Crystal Structure of the Human Cannabinoid Receptor CB1. C.; Liu, Z.-J. Crystal Structure of the Human Cannabinoid Receptor CB2.
- How Understanding Intracellular Drug Access Can Transform Your GPCR Drug Discovery Program
Welcome back GPCR fans, The pace of GPCR innovation is accelerating at a rate that can be difficult to
- â”Sailing the GPCR Seas: Your Weekly Research Voyage! ⊿ Nov 11 - 17, 2024
GPCR community members Build connections with other GPCR fans :) So much more to come!
- An overview of the compartmentalized GPCR Signaling: Relevance and Implications
Z., Wilderman, A., Katakia, T., McCann, T., Yokouchi, H., Zhang, L., Corriden, R., Liu, D., Feigin, M
- Overview of adhesion GPCRs self-activation
Qian, Y., Ma, Z., Liu, C., Li, X., Zhu, X., Wang, N., Xu, Z., Xia, R., Liang, J., Duan, Y., Yin, H.,
- Hop in the Time Machine with GPCR: Unraveling the Future of Research! ⊿ Nov 24 - Dec 1, 2024
GPCR community members Join the GPCR fan club and geek out with fellows! So much more to come!
- The Perils and Guardrails of Modifying Signalling Proteins in Bioassays
Liu S, Anderson PJ, Rajagopal S, Lefkowitz RJ, Rockman HA.
