Search Results
Results found for "GPCR Pharmacology"
- 📰 GPCR Weekly News, May 1 to 7, 2023
GPCR Symposium on GPCR Activation and Signaling. ASPET 2023 - American Society for Pharmacology and Experimental Therapeutics (May 18 - 21, 2023). (June 4 - 8, 2023). 2023 Molecular Pharmacology (GRS) Seminar GRC. (June 10 - 11, 2023). 1, 2023) 19th World Congress of Basic & Clinical Pharmacology 2023. GPCR Ecosystem
- 📰 GPCR Weekly News, September 25 to October 1, 2023
Hello GPCR enthusiasts! Join us for our weekly GPCR round-up. This week's highlights: Drs. GPCR Symposia? GPCR Newsletter! , and more Network pharmacology -based study on the mechanism of traditional Chinese medicine in the GPCR Ecosystem
- 📰 GPCR Weekly News, April 24 to 30, 2023
GPCR Symposium on GPCR Activation and Signaling on May 19th, 2023. Events, Meetings, and Webinars ASPET 2023 - American Society for Pharmacology and Experimental Therapeutics (June 4 - 8, 2023). 2023 Molecular Pharmacology (GRS) Seminar GRC. (June 10 - 11, 2023). 1, 2023) 19th World Congress of Basic & Clinical Pharmacology 2023. GPCR Ecosystem
- 📰 GPCR Weekly News, April 17 to 23, 2023
GPCR Symposium on GPCR Activation and Signaling, May 19th, 2023. GPCR Events, Meetings, and Webinars ASPET 2023 - American Society for Pharmacology and Experimental Therapeutics (June 4 - 8, 2023). 2023 Molecular Pharmacology (GRS) Seminar GRC. (June 10 - 11, 2023). 1, 2023) 19th World Congress of Basic & Clinical Pharmacology 2023. GPCR Ecosystem
- Cholesterol-Dependent Dynamics of the Serotonin1A Receptor Utilizing Single Particle Tracking: ...
Receptor Utilizing Single Particle Tracking: Analysis of Diffusion Modes "G protein-coupled receptors (GPCRs Serotonin1A receptors are important members of the GPCR family and are implicated in neuropsychiatric To explore the role of cholesterol in lateral dynamics of GPCRs, we utilized single particle tracking results bring out the interdependence of cholesterol and actin cytoskeleton in regulating diffusion of GPCRs Read more at the source #DrGPCR #GPCR #IndustryNews
- Dimerization of β2-adrenergic receptor is responsible for the constitutive activity subjected to inv
Read more at the source #DrGPCR #GPCR #IndustryNews Subscribe to the Dr. GPCR Newsletter HERE
- 📰 GPCR Weekly News, April 10 to 16, 2023
GPCR Symposium on GPCR Activation and Signaling on May 19th, 2023. (April 20 - 21, 2023) Swiss Biotech Day (April 24 - 25, 2023) ASPET 2023 - American Society for Pharmacology (June 4 - 8, 2023). 2023 Molecular Pharmacology (GRS) Seminar GRC. (June 10 - 11, 2023). 1, 2023) 19th World Congress of Basic & Clinical Pharmacology 2023. GPCR Ecosystem
- Lipid Modulation of a Class B GPCR: Elucidating the Modulatory Role of PI(4,5)P 2 Lipids
lipids have been shown to stabilize an active conformation of class A G-protein coupled receptors (GPCRs ) through a conserved binding site, not present in class B GPCRs. For class B GPCRs, previous molecular dynamics (MD) simulation studies have shown PI(4,5)P2 interacting conformation of GCGR through a binding site conserved across class B GPCRs but absent in class A GPCRs Read more at the source #DrGPCR #GPCR #IndustryNews
- 📰 GPCR Weekly News, April 3 to 9, 2023
subset-specific receptor expression in Caenorhabditis elegans. β- Arrestins: Structure, Function, Physiology, and Pharmacological (April 20 - 21, 2023) Swiss Biotech Day (April 24 - 25, 2023) NEW ASPET 2023 - American Society for Pharmacology (June 4 - 8, 2023). 2023 Molecular Pharmacology (GRS) Seminar GRC. (June 10 - 11, 2023). 1, 2023) 19th World Congress of Basic & Clinical Pharmacology 2023. GPCR Ecosystem
- 📰 GPCR Weekly News, August 28 to September 3, 2023
Stay informed with our GPCR roundup. GPCR Symposium on 'GPCRs as Therapeutic Modalities' Showcase your project with a 1-minute abstract video : a guard of women's health β-Arrestins: Structure, Function, Physiology, and Pharmacological Perspectives Postdoc Research Associate Director, Regulatory Affairs Research Scientist/Senior Scientist I - Molecular Pharmacology GPCR Ecosystem
- Purpose-Driven Opioid Research: Catherine Demery’s Academic Path
Rather than treating opioid pharmacology as a purely theoretical exercise, she collaborates with harm-reduction This approach makes her models not just rigorous, but translational—bridging the gap between receptor pharmacology That personal loss transforms complex receptor pharmacology into something immediate and human. And GPCR pharmacology isn’t just an academic pursuit—it’s essential to understanding and responding to
- Dr. Simone Promel
GPCR Virtual Cafe? Join us for another virtual cafe talk to hear about the amazing work that Dr. Simone Promel / Promel Lab is doing on adhesion #GPCRs. Register here (free): https://www.ecosystem.drgpcr.com/dr-gpcr-virtual-cafe/ #gpcr #drgpcr #podcast
- 📰 GPCR Weekly News, March 20 to 26, 2023
GPCR Ecosystem. GPCR Events, Meetings, and Webinars FREE 5th ERNEST GPCR ECI zoominar. (June 4 - 8, 2023). 2023 Molecular Pharmacology (GRS) Seminar GRC. (June 10 - 11, 2023). 1, 2023) 19th World Congress of Basic & Clinical Pharmacology 2023. GPCR Ecosystem
- PH-Binding Motif in PAR4 Oncogene: From Molecular Mechanism to Drug Design
October 2022 "While the role of G-protein-coupled receptors (GPCR) in cancer is acknowledged, their underlying Protease-activated receptors (PAR), a subgroup of GPCRs, form a family of four members (PAR1-4) centrally Read more at the source #DrGPCR #GPCR #IndustryNews
- 📰 GPCR Weekly News, March 13 to 19, 2023
Pharmacological characterization of novel small molecule agonists and antagonists for the orphan receptor G protein-coupled receptor pharmacology - insights from mass spectrometry. (June 4 - 8, 2023). 2023 Molecular Pharmacology (GRS) Seminar GRC. (June 10 - 11, 2023). , 2023) 19th World Congress of Basic & Clinical Pharmacology 2023. GPCR Ecosystem
- 📰 GPCR Weekly News, July 31 to August 6, 2023
Greetings, GPCR fellows! Prepare for the latest GPCR updates. This week's highlights: Dr. GPCR Symposium on 'GPCRs as Therapeutic Modalities' is set for September 22nd. Adhesion GPCRs Functional partnerships between GPI-anchored proteins and adhesion GPCRs GPCR Activation NEW Research Scientist/Senior Scientist I - Molecular Pharmacology NEW Director, Clinical Data Management GPCR Ecosystem
- Production of human A2AAR in lipid nanodiscs for 19F-NMR and single-molecule fluorescence...
describe production of the human A2A adenosine receptor (A2AAR), a class A G protein-coupled receptor (GPCR Read more at the source #DrGPCR #GPCR #IndustryNews
- 📰 GPCR Weekly News, July 24 to July 30, 2023
Welcome, GPCR fellows! Get excited about the latest GPCR news! GPCR Symposium on GPCRs as Therapeutic Modalities is on September 22nd. GPCR Activation and Signaling Endosome positioning coordinates spatially selective GPCR signaling. The Neuromedin U system: pharmacological implications for the treatment of obesity and binge eating behavior GPCR Ecosystem
- Network pharmacological investigation into the mechanism of Kaixinsan powder for the treatment of...
October 2022 Network pharmacological investigation into the mechanism of Kaixinsan powder for the treatment The network pharmacology method was used to constructe the "herb-component-target" network, and elucidated indicated that the mechanism of KXS in treating depression was involved in the biological process of GPCR Read more at the source #DrGPCR #GPCR #IndustryNews
- Focusing on the role of secretin/adhesion (Class B) G protein-coupled receptors in placental...
Read more at the source #DrGPCR #GPCR #IndustryNews
- 📰 GPCR Weekly News, July 17 to July 23, 2023
Welcome, GPCR fellows! Get ready for the latest GPCR news. This week's highlighted papers: Dr. GPCR Symposium on GPCRs as Therapeutic Modalities on September 22nd. GPCR Newsletter! Postdoctoral Fellow, Caron Lab Clinical Trial Associate Research Scientist/Senior Scientist I - Molecular Pharmacology GPCR Ecosystem
- 📰 GPCR Weekly News, March 6 to 12, 2023
GPCR Activation and Signaling Autoregulation of GPCR signalling through the third intracellular loop. (June 4 - 8, 2023). 2023 Molecular Pharmacology (GRS) Seminar GRC. (June 10 - 11, 2023). 1, 2023) 19th World Congress of Basic & Clinical Pharmacology 2023. PhD Studentship - Integrated Approaches In Pharmacology, Computer Simulations And Machine Learning To GPCR Ecosystem
- Bell-Evans model and steered molecular dynamics in uncovering the dissociation kinetics of ligands..
ZMA241385 and agonist NECA that target the A2A adenosine receptor of the G-protein-coupled receptor (GPCR Read more at the source #DrGPCR #GPCR #IndustryNews
- Opioid Ligands Addressing Unconventional Binding Sites and More Than One Opioid Receptor Subtype
"Opioid receptors (ORs) represent one of the most significant groups of G-protein coupled receptor (GPCR ) drug targets and also act as prototypical models for GPCR function. develop drugs with less side effects, and tools to explore the ORs nature and function, various (poly)pharmacological Read more at the source #DrGPCR #GPCR #IndustryNews
- Unlock the Future of GPCR Science: Breakthroughs and Courses Await | Sep 2 - Sep 8, 2024
: Pharmacologic activity measurement, mechanisms of action, and GPCR discovery strategies. Principles of Pharmacology II October 31, November 7, 14, 21, December 5 (five sessions) (we skipped The Principles of Pharmacology I & II BUNDLE is your key to mastering the field. Papers Emerging Voices in GPCR Biology in Special Issue of Molecular Pharmacology GPCR Events, Meetings Congress of Basic and Clinical Pharmacology GPCR Jobs HIGHLIGHT Research Associate - Professor Graeme
- 📰 GPCR Weekly News, February 20 to 26, 2023
(June 4 - 8, 2023). 2023 Molecular Pharmacology (GRS) Seminar GRC. (June 10 - 11, 2023). (June 11 - 16, 2023). 19th World Congress of Basic & Clinical Pharmacology 2023. GPCR Jobs PhD Studentship - Integrated Approaches In Pharmacology, Computer Simulations And Machine Learning development PhD student at Department of Drug Design and Pharmacology Software / database development postdoc at the Department of Drug Design and Pharmacology Postdoc in Bioinformatics/Data Science at
- How Fast Does a Drug Work?
How do competing ligands slow or alter binding rates, and what does this tell you about real-world pharmacology candidates faster Unlock “Drug Binding Kinetics” Now Only in Terry’s Corner ______ #DrugDiscovery #Pharmacology #DrugKinetics #PipelineEfficiency #PharmaInnovation #GPCR #BindingKinetics #MedicinalChemistry #LeadOptimization
- 8th RSC / SCI symposium on GPCRs in Medicinal Chemistry. October 5-7, 2022, Verona, Italy
August 2022 "GPCRs in Medicinal Chemistry Event 8th RSC / SCI symposium on GPCRs in Medicinal Chemistry 6th September 30th September – online registration (card payments)" Read more at the source #DrGPCR #GPCR
- Exploiting Dependence of Castration-Resistant Prostate Cancer on the Arginine Vasopressin ...
We previously demonstrated that the G protein-coupled receptor (GPCR) arginine vasopressin receptor type1A AVPR1A is part of a family of GPCR's including arginine vasopressin receptor type 2 (AVPR2). Read more at the source #DrGPCR #GPCR #IndustryNews
- Functional Characterization of the Venus Flytrap Domain of the Human TAS1R2 Sweet Taste Receptor
sweet taste receptor is a heterodimeric receptor composed of two distinct G-protein-coupled receptors (GPCRs The TAS1R2 and TAS1R3 subunits are members of a small family of class C GPCRs whose members share the Read more at the source #DrGPCR #GPCR #IndustryNews




