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Emmanouil Kyrloglou on the web Adhesion GPCR Consortium LinkedIn A single cell GPCR map of thermogenic , located within the GPCR autoproteolysis inducing (GAIN) domain. This research focuses on the design of a new endogenous ADGRB1 activation reporter assay to test analogs University" About Jesse Stillwell "Jesse Stillwell is a 3rd year graduate student with a research focus in drug His project is drug discovery focused, with particular interest in use of a novel epigenetic therapy

GPCR Podcast Strategic Partners Dr. Alexander S. Hauser About Dr. Alexander S. During his Ph.D. with David Gloriam at the Department of Drug Design and Pharmacology in Copenhagen, of Molecular Biology in Cambridge, UK, where he was working on the impact of genetic variations on drug Award” for his work on GPCRs. Dr. Alexander S. GPCR Ecosystem Enjoying the Dr. GPCR Podcast? Leave a Review.

GPCR Podcast Strategic Partners Dr. Michael Feigin About Dr. Michael Feigin "Dr. as a potential drug target due to its high expression in triple negative breast cancer. GPCR Targeted Drugs and Gene Regulation in Cancer Cells Mike presented research on the effect of GPCR-targeted GPCRs and Cancer Immune Modulation Yamina and Mike had a discussion about their research on GPCRs, specifically GPCR Podcast? Leave a Review.

Now at the University of Glasgow, his primary research interests are focused on the rational design of novel drugs to treat the three global health challenges of dementia, asthma, and malaria. staff supported by basic research grants investigating aspects of disease biology and the action of drugs at the University of Glasgow underpinned by a £118M new build that will house over 550 researchers designed GPCR Ecosystem Enjoying the Dr. GPCR Podcast? Leave a Review.

GPCR Podcast Strategic Partners Dr. Marta Filizola About Dr. Marta Filizola Dr. into the structure, dynamics, and function of important classes of membrane proteins and prominent drug targets, including G protein-coupled receptors (GPCRs), transporters, channels, and 3 integrins. To this end, her lab uses several computational structural biology tools and rational drug design approaches GPCR Ecosystem Enjoying the Dr. GPCR Podcast? Leave a Review.

with numerous pharma and biotechs in understanding and applying in vitro pharmacology data to advance drug He specializes in kinetic analysis of drug action and is known for applying binding kinetics to the development He guided the in vitro biology efforts of the company for numerous drug discovery campaigns. of GPCR function to better target receptors. GPCR Member ResearchGate Dr. GPCR Ecosystem Enjoying the Dr. GPCR Podcast? Leave a Review.

Weekly News, featuring expert insights on target engagement, a practical framework for irreversible drugs GPCR Weekly News - Oct 23 - The Power and Peril of Irreversible Drugs Published on October 23, 2025 Category Premium sneak peek inside. 🔹 Terry’s Corner: A practical framework for irreversible drugs—defining “ Jens Carlsson on predictive modeling—where structure-based design and MD guide experiments (and where #DrGPCR #GPCR Previous Next Recent Articles

GPCR Podcast Strategic Partners Dr. Katarina Nemec About Dr. engaged in researching molecular mechanisms that govern human (patho-)physiology and their interplay with drugs I aim to discover new therapeutic approaches, and druggable molecules or refine canonical drug targets to create drugs with fewer adverse effects. GPCR Enjoying the Dr. GPCR Podcast? Leave a Review.

Gabriele Kockelkoren shares: 🔬 How GPCR spatial organization shapes signaling and drug responses 🌍 the unknown is key to scientific breakthroughs A must-listen for biophysicists, pharmacologists, and drug GPCR Podcast 🎧 "You will always feel like you know nothing— and that’s completely fine." Gabriele Kockelkoren shares:🔬 How GPCR spatial organization shapes signaling and drug responses🌍 His the unknown is key to scientific breakthroughs A must-listen for biophysicists, pharmacologists, and drug

GPCR Podcast Strategic Partners Dr. Jean Martin Beaulieu About Dr. Jean Martin Beaulieu Dr. These receptors belong to the super-family of G-protein coupled receptors (GPCR), the major molecular target for drug development. and drug development technology. GPCR Ecosystem Enjoying the Dr. GPCR Podcast? Leave a Review.

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If you work with GPCRs, this perspective changes how you design experiments and interpret data. 🎧 Watch It shaped how we design experiments, make decisions, and lead teams. In this week’s Dr. #EarlyDiscovery #PharmaR&D #BiotechInnovation Irreversible kinetics = strategic lever in drug design Binding kinetics are a design variable, as critical as potency or clearance. Start designing them to happen.

Stay current in drug discovery with the University Vault. Quickly get up to speed on new GPCR targets and mechanisms, and gain a competitive edge with our extensive University Vault: The Ultimate On-Demand GPCR Learning Library Every talk inside the University Vault field 🧠 Designed for researchers at every career stage 🚀 Don’t just keep up — lead the way. Anonymous This looks super useful for drug discovery!

GPCR collaboration at Monash shows how shared lab ecosystems can reshape innovation and accelerate drug Home → Flash News → How GPCR Collaboration Built an Innovation Engine How GPCR Collaboration Built an GPCR Podcast Collaboration isn’t a soft skill — it’s an innovation strategy. An ecosystem where GPCR innovation accelerated — not because of a single star scientist, but because GPCR Premium #GPCR #DrGPCR #DrugDiscovery #Innovation #ScienceLeadership #Collaboration Previous Next

GPCR Podcast Strategic Partners The Role of Quantitative Sciences in GPCRs with Dr. She has advanced the use of computational methods to meet the challenges of designing therapeutics with molecular dynamics simulation methods with emphasis on application to G-protein coupled receptors and drug design." GPCR Enjoying the Dr. GPCR Podcast? Leave a Review.

Learn from leading GPCR experts — anytime, anywhere Access trusted, on-demand courses designed to help networking, AMAs & matchmaking 💡 Support open resources for the global GPCR field 🧠 Designed for researchers At Dr.GPCR University, you’ll find: Courses: Dive deep into curated educational content designed by experts GPCR University Masterclasses designed for? Some classes may require basic knowledge of GPCRs, but many are designed to accommodate beginners as

Stay at the Forefront of GPCR Drug Discovery Gain insider methods from the pioneers shaping biased signaling , assay design, and pharmacology—skills you won't find in any textbook or paper. ⧖ 20+ Hours of Expert research Access exclusive training from the scientists shaping the future of GPCR drug discovery Dr. for assay design strategies. field 🧠 Designed for researchers at every career stage 🚀 Don’t just keep up — lead the way.

His journey highlights the transition from general drug development to a deep dive into G protein-coupled Allosteric Modulation: The New Frontier of GPCR Drug Discovery Ben reflects on the emerging potential “The goal is to smash all the amazing biology together and make a drug.” design . 8. GPCR ecosystem , GPCR online course , GPCR scientist network , GPCR drug discovery , GPCR training program

Juan José Fung is a Principal Scientist at GPCR Therapeutics, Inc , a drug discovery company focused Brian Kobilka , studying the dimerization of GPCRs. Dr. spent significant time in the industry studying membrane proteins, antibodies, and HTS methods for drug Juan José Fung on the web LinkedIn GPCR Therapeutics Dr. GPCR Ecosystem Enjoying the Dr. GPCR Podcast? Leave a Review.

schedule Illuminating Functional Selectivity and Allosterism at GPCRs. receptors involved in many, if not all, physiological responses, with the ultimate goal of improving drug in-cellulo measurement of protein-protein interactions, receptor trafficking and signalling, useful for drug GPCR Previous Event Next Event Great Lakes GPCR Retreat and Club des Récepteurs à Sept Domaines Transmembranaires 22nd GPCR Retreat Sponsored by

GPCR Podcast Strategic Partners Dr. David E. function and drug discovery and a Pharmaceutical Data Science unit. each month retrieve reference data and access online tools for analysis, visualization, and experiment design one of the coordinators of recommendations to describe ligand bias towards signaling probes and safer drugs GPCR Ecosystem Enjoying the Dr. GPCR Podcast? Leave a Review.

Discover how strategic collaboration drives real GPCR drug discovery impact. GPCR Podcast If your model can’t change an experiment, what’s the point? That’s the standard Dr. The kind of impact that shows up in how experiments are designed, which compounds get prioritized, and In GPCR drug discovery, where complexity is the rule and timelines are tight, this kind of cross-functional GPCR Podcast: model predict discover #DrGPCR #GPCR #CollaborationInScience #ComputationalChemistry #Pharmacology

GPCR Podcast Strategic Partners Dr. JoAnn Trejo About Dr. JoAnn Trejo Dr. PARs are GPCRs that are activated through an atypical irreversible proteolytic mechanism. biology and for the identification of drug targets and future drug development. which has important functions in hemostasis, thrombosis, inflammation, and cancer and is an important drug GPCR Ecosystem Enjoying the Dr. GPCR Podcast? Leave a Review.

GPCR Podcast Strategic Partners Leadership, Impact, and GPCR Signaling with Dr. signaling opens new doors in drug discovery. the Guest Michelle Halls is an Associate Professor at Monash University and Deputy Theme Leader of Drug GPCR Premium . GPCR Podcast? Leave a Review.

GPCR Podcast Strategic Partners Dr. Daniel Wacker About Dr. and in vitro drug discovery. Icahn School of Medicine at Mount Sinai in NYC, where I have been working on structure-function and drug discovery of GPCRs and transporters. GPCR Ecosystem Enjoying the Dr. GPCR Podcast? Leave a Review.

From her early doubts to designing preclinical models of fentanyl and xylazine overdose, she reflects drugs. pharmacologist—led her to investigate how these drugs shut down breathing in different ways. Who Should Listen This episode is especially relevant for: GPCR drug discovery scientists Respiratory GPCR ecosystem , GPCR training program , GPCR podcast , opioid pharmacology , xylazine research , mu

drug discovery . circuits — insights that inform next-generation functional assay development and translational therapeutic design Why this matters How receptor distribution in islets and brain circuits shapes incretin hormone drug collaborative chemistry enabled in designing receptor-targeted fluorescent ligands The moment when structural assays Worked across disciplines where chemistry, pharmacology, and physiology converge Questioned how drug

Michelle describes how reading those early papers on lipid-rich domains and GPCR–G protein compartmentalization The way signals are organized defines specificity, drug response, and potential for targeted therapies If you work with GPCRs, this perspective changes how you design experiments and interpret data. 🎧 Watch /leadership-luck-and-gpcr-signaling ✨ Join Premium: https://www.ecosystem.drgpcr.com/gpcr-university-pricing #GPCR #DrGPCR Previous Next Recent Articles

Accelerated Program Progression: Design robust assay cascades and establish key go/no-go points to speed Accelerated Preclinical Progression I streamline critical operational processes, from advanced assay design drug discovery. Berchiche, and I understand the intricate challenges of GPCR drug discovery. drug discovery.

targets — a top-down rethink for drug discovery. << Back to podcast list Dr. GPCR Podcast Strategic Partners GPCRs and the Science Behind Pain and Recovery with Dr. “We’re using outdated drugs. There are more elegant GPCR targets waiting to be explored.” He’s fascinated by transgenerational epigenetics — how parental pain, diet, or drug exposure can leave GPCR ecosystem, GPCR drug discovery, GPCR podcast, GPCR data platform, GPCR training program, RGS4, chronic