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Results found for "GPCR Drug Design"
- Session VI | Adhesion GPCR Workshop 2024 | Dr. GPCR Ecosystem
Full Agenda Adhesion GPCR workshop 2024 CINVESTAV, Mexico City, Mexico October 23-25 Download PDF Program formation, maintenance and degeneration Yimin Zou Antibody-drug conjugates targeting CD97 in glioblastoma Yimin Zou on the web UC San Diego Antibody-drug conjugates targeting CD97 in glioblastoma Dimitris Placantonakis To exploit this expression profile, we have developed antibody-drug conjugates (ADCs) targeting CD97, GPCR < Previous Session Next Session >
- Dr. David E. Gloriam | Dr. GPCR Ecosystem
Computational Receptor Biology at the University of Copenhagen where he leads a research cluster for GPCR function and drug discovery and a Pharmaceutical Data Science unit. each month retrieve reference data and access online tools for analysis, visualization, and experiment design one of the coordinators of recommendations to describe ligand bias towards signaling probes and safer drugs GPCR Ecosystem Enjoying the Dr. GPCR Podcast? Leave a Review.
- Dr. JoAnn Trejo | Dr. GPCR Ecosystem
the guidance of Professor Shaun Coughlin where she worked on the newly discovered protease-activated GPCRs PARs are GPCRs that are activated through an atypical irreversible proteolytic mechanism. biology and for the identification of drug targets and future drug development. which has important functions in hemostasis, thrombosis, inflammation, and cancer and is an important drug GPCR Ecosystem Enjoying the Dr. GPCR Podcast? Leave a Review.
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Dr GPCR is a 501(c)(3) non-profit. global GPCR community better — by upgrading the Dr GPCR University, creating more learning opportunities to make cutting-edge GPCR knowledge accessible to everyone Dr GPCR Retreat: offering free or affordable Together, we can accelerate GPCR discoveries and develop more effective drugs for everyone. 👉 Donate Now to Support the Dr GPCR Ecosystem
- Some biotech stories start in the lab. Celtarys started with a thesis project, a new chemical strategy, and a vision to make fluorescence available for drug discovery. Now, they’re growing fast and partnering with Dr. GPCR to connect with the researchers who need them most. ✳️ Learn more about the partnership: https://www.ecosystem.drgpcr.com/celtarys-research-dr-gpcr-ecosystem #GPCRcommunity #ScienceCollaboration #FluorescentLigands #BiotechStartup | Dr. GPCR Ecosystem
started with a thesis project, a new chemical strategy, and a vision to make fluorescence available for drug GPCR to connect with the researchers who need them most. ✳️ Learn more about the partnership: https:/ /www.ecosystem.drgpcr.com/celtarys-research-dr-gpcr-ecosystem #GPCRcommunity #ScienceCollaboration #FluorescentLigands to with a thesis project, a new chemical strategy, and a vision to make fluorescence available for drug GPCR to connect with the researchers who need them most. ✳️ Learn more about the partnership: https:/
- We’re excited to announce our strategic partnership with Celtarys Research, a biotech company specializing in fluorescent ligand technologies and real-time, non-radioactive GPCR assays. This collaboration combines Dr. GPCR’s global platform with Celtarys’ innovative chemical biology tools, making it easier than ever for scientists to study ligand-receptor interactions, visualize binding, and accelerate drug discovery. We’re proud to welcome Celtarys to the Dr. GPCR ecosystem to support researchers worldwide and expand access to high-performance tools for GPCR-targeted therapeutics. ✳️Read the complete press release: https://www.ecosystem.drgpcr.com/post/dr-gpcr-and-celtarys-research-join-forces-to-expand-access-to-innovative-gpcr-tools #GPCR #DrGPCR #CeltarysResearch #DrugDiscoveryTools #FluorescentLigands #GPCRresearch #ScientificPartnership | Dr. GPCR Ecosystem
scientists to study ligand-receptor interactions, visualize binding, and accelerate drug discovery. GPCR ecosystem to support researchers worldwide and expand access to high-performance tools for GPCR-targeted for scientists to study ligand-receptor interactions, visualize binding, and accelerate drug discovery GPCR ecosystem to support researchers worldwide and expand access to high-performance tools for GPCR-targeted uncomfortable truth: 👉 Your biotech is already running on an operating cadence you didn’t consciously design
- Join the Dr. GPCR Affiliate Program - Empower the GPCR Community with Dr. GPCR Ecosystem Services
GPCR Affiliate Program and earn commissions by helping connect the global GPCR community. Share our ecosystem, courses, and events to advance drug discovery together. Dr. GPCR community. The Ecosystem is designed for all GPCR professionals to have an affordable and highly effective way to GPCR Ecosystem?
- Dr. Aurélien Rizk | Dr. GPCR Ecosystem
Aurélien Rizk is a scientist and entrepreneur in drug discovery. Before focusing on the development of innovative mathematical modeling and simulation methods for drug Interdisciplinary Teamwork and Drug Development Yamina Berchiche and Aurelien Rizk emphasized the significance of interdisciplinary teamwork in drug and technology development, noting the challenges of communication Aurelien Rizk confirmed his attendance at the upcoming GPCR-Targeted Drug Discovery Summit in Boston.
- GPCR location matters with Dr. Gabriele Kockelkoren | Dr. GPCR Ecosystem
<< Back to podcast list Strategic Partner(s) GPCR location matters with Dr. In my PhD, I studied the nanoscale spatial organization of G protein-coupled receptors (GPCRs) at the revealed heterogeneous spatial patterns of receptor density and activation, that are modulated in a drug-dependent These findings identify nanoscale GPCR spatial organization as an integral element of their activity GPCR Podcast? Leave a Review.
- A Brief History of allosteric modulation with Dr. Arthur Christopoulos | Dr. GPCR Ecosystem
His research focuses on novel paradigms of drug action at GPCRs, particularly allosteric modulation and Next steps - Arthur will continue to collaborate with other researchers and drug companies to advance the understanding and application of allosteric modulation. - Arthur will work on designing ligands design principles. GPCR Podcast? Leave a Review.
- ep 175 with jens carlsson clip 1 | Dr. GPCR Ecosystem
Jens Carlsson’s lab at Uppsala University is redefining GPCR drug discovery with predictive molecular Jens Carlsson and his team are redefining what computational modeling means in drug discovery. By integrating molecular docking, molecular dynamics, and machine learning, they design ligands with drug discovery. 🎧 Explore how predictive modeling is reshaping GPCR science in this Dr. uncomfortable truth: 👉 Your biotech is already running on an operating cadence you didn’t consciously design
- Dr. Yamina Berchiche | Dr. GPCR Ecosystem
GPCR podcast , your host and founder, Dr. Yamina Berchiche introduces the very first podcast dedicated to GPCRs researcher and their work. GPCR Ecosystem, with the goal is to bring together GPCR scientists, biotech, and pharma leaders as well , grow, and thrive together to accelerate GPCR drug discovery and improve human health. GPCR Ecosystem Enjoying the Dr. GPCR Podcast? Leave a Review.
- Generic tools won’t solve tomorrow’s drug discovery challenges. That’s why Celtarys designs custom fluorescent probes for every target, built for real pharmacology, not just convenience. With Dr. GPCR and Celtarys joining forces, expect more visibility, more precision, and more scientific impact. 🚀 Get to know our media partner: https://www.ecosystem.drgpcr.com/celtarys-research-dr-gpcr-ecosystem #GPCRdrugDiscovery #GPCRecosystem #CustomLigands | Dr. GPCR Ecosystem
Home → Flash News → Generic tools won’t solve tomorrow’s drug discovery challenges. That’s why Celtarys designs custom fluorescent probes for every target, built for real pharmacology, CustomLigands Published on June 27, 2025 Category Celtarys - Media Partner Generic tools won’t solve tomorrow’s drug That’s why Celtarys designs custom fluorescent probes for every target, built for real pharmacology, uncomfortable truth: 👉 Your biotech is already running on an operating cadence you didn’t consciously design
- Eleonora Comeo | Dr. GPCR Ecosystem
Eleonora Comeo About this episode Eleonora Comeo is a doctoral candidate in Medicinal Chemistry and Drug We sat down to chat about GPCRs, synthesizing labeled ligands, and her unique position that allows her to work with GPCR scientists on 2 continents. GPCR Ecosystem Enjoying the Dr. GPCR Podcast? Leave a Review. Imaging in Native Tissue How Collaboration Sparked a GPCR Imaging Breakthrough in Chemical Biology Thanks
- Dr. Josephine (Pina) Cardarelli | Dr. GPCR Ecosystem
of GPCR Therapeutics, USA, a newly incorporated Biotechnology company in the Bay Area. Additionally, they have a library of target GPCR heteromers for Oncology. Dr. Cardarelli is a drug development leader with extensive experience driving drug discovery teams in bringing She has extensive experience working with Biologics, and Antibody Drug Conjugates as well as experience GPCR Ecosystem Enjoying the Dr. GPCR Podcast? Leave a Review.
- Dr. Paul Insel | Dr. GPCR Ecosystem
Medicine for their discovery of G-proteins and their role in signal transduction in cells, Paul was designated , Paul and his team focus on previously unrecognized receptors with the hopes to use these as novel drug GPCR Ecosystem Enjoying the Dr. GPCR Podcast? Leave a Review. Better Questions in Science: A Practical Guide for Emerging Researchers When the Islet Lit Up: Advancing GPCR Imaging in Native Tissue How Collaboration Sparked a GPCR Imaging Breakthrough in Chemical Biology Thanks
- Terry's Corner is Officially LIVE! 🎉 This is your new go-to for mastering drug discovery pharmacology. No fluff, just clear, on-demand insights from Terry Kenakin. Building core expertise? Master dose-response, binding, kinetics, and foundational models. Driving drug discovery? Apply pharmacology to selectivity, ADME, and strategic decision-making. An experienced drug hunter? Sharpen your edge with allosteric bias, residence time, and translational PK/PD. Learn on-demand, apply immediately: https://terrykenakin.com #DrGPCR #GPCR #pharmacology #TerrysCorner #DrugDiscovery | Dr. GPCR Ecosystem
🎉 This is your new go-to for mastering drug discovery pharmacology. An experienced drug hunter? Learn on-demand, apply immediately: https://terrykenakin.com #DrGPCR #GPCR #pharmacology #TerrysCorner An experienced drug hunter? Learn on-demand, apply immediately: https://terrykenakin.com #DrGPCR #GPCR #pharmacology #TerrysCorner
- Every receptor tells a story | Dr. GPCR Ecosystem
Every receptor tells a story but GPCRs speak a language of organization. Dr. Michelle Halls unpacks how GPCR signaling isn’t just about ligand–receptor interaction. Michelle Halls unpacks how GPCR signaling isn’t just about ligand–receptor interaction. level of organization defines specificity in signaling, and understanding it changes how we think about drug signaling: 👉 https://www.ecosystem.drgpcr.com/dr-gpcr-podcast/leadership-luck-and-gpcr-signaling #GPCR
- Plenary Lecture | Adhesion GPCR Workshop 2024 | Dr. GPCR Ecosystem
Full Agenda Adhesion GPCR workshop 2024 CINVESTAV, Mexico City, Mexico October 23-25 Download PDF Program Our first main research aspect is the identification of endogenous ligand of GPCRs. Our third main research aspect is working mechanism of GPCR. Our fourth main research aspect is ligand coding mechanisms and structural aided drug discovery of GPCR (Cell 2021, 2023, Nature 2023b), bile acids or its derivatives by GPCRs (Nature 2020)."
- How GPCR Collaboration Built an Innovation Engine | Dr. GPCR Ecosystem
GPCR collaboration at Monash shows how shared lab ecosystems can reshape innovation and accelerate drug Home → Flash News → How GPCR Collaboration Built an Innovation Engine How GPCR Collaboration Built an GPCR Podcast Collaboration isn’t a soft skill — it’s an innovation strategy. GPCR Premium #GPCR #DrGPCR #DrugDiscovery #Innovation #ScienceLeadership #Collaboration Previous Next uncomfortable truth: 👉 Your biotech is already running on an operating cadence you didn’t consciously design
- Dr. Prasenjit Saha | Dr. GPCR Ecosystem
Specifically, I am interested in understanding dysregulated G-protein coupled receptor (GPCR) signaling Traditional drug discovery efforts have focused on agonists and antagonists that bind to the orthosteric My long-term plan is to conduct research in the field of receptor biology, with a focus on GPCRs. ubiquitous class of plasma membrane receptors and serve as targets for more than one-third of all prescribed drugs GPCR Enjoying the Dr. GPCR Podcast? Leave a Review.
- Dr. GPCR Community Presentation | Adhesion GPCR Workshop 2024 | Dr. GPCR Ecosystem
Full Agenda Adhesion GPCR workshop 2024 CINVESTAV, Mexico City, Mexico October 23-25 Download PDF Program GPCR Community Presentation Breaking Barriers: My Journey from Mexico to the Heart of the Dr. GPCR Ecosystem and beyond About Monserrat Avila Zozaya "My doctoral research was focused on investigating My research focuses on understanding the molecular mechanisms of adhesion GPCRs (aGPCRs) in lymphatic GPCR < Previous Session Next Session >
- You never know where your GPCR takes you with Dr. Brian Hudson | Dr. GPCR Ecosystem
<< Back to podcast list Strategic Partner(s) You never know where your GPCR takes you with Dr. He has more than 20 years of experience in GPCR, primarily focused on drug discovery and developing new leads a research group that is focused on understanding the pharmacology and function of a group a GPCRs GPCR Podcast? Leave a Review. Imaging in Native Tissue How Collaboration Sparked a GPCR Imaging Breakthrough in Chemical Biology Thanks
- Chemical Probes for GPCR Imaging and Internalization with Dr. Johannes Broichhagen | Dr. GPCR Ecosystem
GPCR Podcast, chemical biologist Dr. drug discovery . He explains what chemical design can solve that antibodies can’t, how to validate functional assay systems Why this matters How a chemist with zero biology training became a leader in GPCR probe design. GPCR Podcast? Leave a Review.
- Dr. Pierre Eftekhari | Dr. GPCR Ecosystem
Pierre Eftekhari "Clinical physiologist and biologist , with more than 25 years of experience in drug development. have been engaged in GPCR cellular and clinical pharmacology as scientist or PI in neonatal I have participated and initiated methodologies for development of pharmacologically active anti-GPCR or contributed in 38 published scientific work mainly in the field of immunology and pharmacology of GPCR GPCR Enjoying the Dr. GPCR Podcast? Leave a Review.
- Session I | Adhesion GPCR Workshop 2024 | Dr. GPCR Ecosystem
Full Agenda Adhesion GPCR workshop 2024 CINVESTAV, Mexico City, Mexico October 23-25 Download PDF Program Activation: Direct Communication of Extracellular Region with Transmembrane Domain in a Holo-Adhesion GPCR point mutant knock-in mouse, H381S Frank Kwarcinski Tethered Peptide Activation Mechanism of Adhesion GPCRs ECR-mediated mechanism opens new possibilities for drugging aGPCRs. Frank Kwarcinski on the web LinkedIn Tethered Peptide Activation Mechanism of Adhesion GPCRs Peng Xiao
- Media Partner Packages | Dr. GPCR Ecosystem
GPCR Ecosystem. Elevate Your GPCR Focused Company Visibility Reach 1400+ GPCR researchers. partner, you'll gain trusted access to an engaged audience of academic researchers, biotech teams, and drug GPCR? These touch points are designed to reinforce brand presence and credibility through repeated, trusted
- Dr. Christel Menet | Dr. GPCR Ecosystem
was the 6th employee and today we are more than 60 :) I have fun every day, and I love working with GPCRs Christel Menet on the web Hyphen Projects GPCRS Drug Discovery Confo Therapeutics LinkedIn Dr. GPCR Ecosystem Enjoying the Dr. GPCR Podcast? Leave a Review. Better Questions in Science: A Practical Guide for Emerging Researchers When the Islet Lit Up: Advancing GPCR Imaging in Native Tissue How Collaboration Sparked a GPCR Imaging Breakthrough in Chemical Biology Thanks
- Robert Laprairie | Dr. GPCR Ecosystem
Robert Laprairie is an Associate Professor and the Saskatchewan Research Chair in Drug Discovery and GPCR Ecosystem Enjoying the Dr. GPCR Podcast? Leave a Review. Better Questions in Science: A Practical Guide for Emerging Researchers When the Islet Lit Up: Advancing GPCR Imaging in Native Tissue How Collaboration Sparked a GPCR Imaging Breakthrough in Chemical Biology Thanks
- Dr. Steven Foord | Dr. GPCR Ecosystem
He introduced molecular pharmacology to a wide range of the company's GPCR projects and was able to initiate He also discovered and championed a novel prostaglandin EP4 drug candidate for development. GPCR Ecosystem Enjoying the Dr. GPCR Podcast? Leave a Review. Better Questions in Science: A Practical Guide for Emerging Researchers When the Islet Lit Up: Advancing GPCR Imaging in Native Tissue How Collaboration Sparked a GPCR Imaging Breakthrough in Chemical Biology Thanks

















