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GPCR Podcast Strategic Partners Eleonora Comeo About this episode Eleonora Comeo is a doctoral candidate in Medicinal Chemistry and Drug Discovery in the joint program of the University of Nottingham in the We sat down to chat about GPCRs, synthesizing labeled ligands, and her unique position that allows her to work with GPCR scientists on 2 continents. GPCR Ecosystem Enjoying the Dr. GPCR Podcast? Leave a Review.

Home → Flash News → master gpcr pharmacologic models before its too late Published on July 11, 2025 Category GPCR Weekly News Most GPCR teams aren’t failing because of bad science. This week’s GPCR Weekly News helps you fix that. Yamina’s Corner exposes the silent drift killing GPCR programs (and how to reverse it). ✳️ Read the Weekly News → https://www.ecosystem.drgpcr.com/post/crush-data-confusion-conquer-gpcr-drug-discovery

“I think I don’t have a linear trajectory… the beauty of seeing molecule design and reactions—thinking Alessandro Nicoli He studied pharmaceutical chemistry in Padua, where his fascination with molecular design close to experimental structures, provided a powerful starting point for docking, dynamics, and ligand design—especially drug discovery pipelines. GPCR ecosystem , GPCR online course , GPCR scientist network , GPCR drug discovery , GPCR training program

GPCR Podcast Strategic Partners Dr. Paul Insel About this episode In 1975, Dr. Medicine for their discovery of G-proteins and their role in signal transduction in cells, Paul was designated , Paul and his team focus on previously unrecognized receptors with the hopes to use these as novel drug GPCR Ecosystem Enjoying the Dr. GPCR Podcast? Leave a Review. Collaboration Built an Innovation Engine From Pipettes to Platforms: The Evolution of GPCR Research

GPCR Podcast Strategic Partners A Brief History of allosteric modulation with Dr. His research focuses on novel paradigms of drug action at GPCRs, particularly allosteric modulation and the understanding and application of allosteric modulation. - Arthur will work on designing ligands design principles. GPCR Podcast? Leave a Review.

Full Agenda Adhesion GPCR workshop 2024 CINVESTAV, Mexico City, Mexico October 23-25 Download PDF Program signaling pathway of the ADGRA homolog Remoulade in Drosophila Beatriz Blanco Redondo The Adhesion GPCR The mammalian Remo homolog ADGRA2/Gpr124 cooperates with other GPCRs of the Frizzled family, and the Langenhan where I am studying and characterizing newly generated adhesion GPCR receptors in Drosophila Anaesthesiology and Intensive Care, Medical Faculty, Leipzig University, Leipzig, Germany 5 Institute for Drug

Dr GPCR is a 501(c)(3) non-profit. global GPCR community better — by upgrading the Dr GPCR University, creating more learning opportunities to make cutting-edge GPCR knowledge accessible to everyone Dr GPCR Retreat: offering free or affordable Together, we can accelerate GPCR discoveries and develop more effective drugs for everyone. 👉 Donate Now to Support the Dr GPCR Ecosystem

started with a thesis project, a new chemical strategy, and a vision to make fluorescence available for drug GPCR to connect with the researchers who need them most. ✳️ Learn more about the partnership: https:/ /www.ecosystem.drgpcr.com/celtarys-research-dr-gpcr-ecosystem #GPCRcommunity #ScienceCollaboration #FluorescentLigands to with a thesis project, a new chemical strategy, and a vision to make fluorescence available for drug GPCR to connect with the researchers who need them most. ✳️ Learn more about the partnership: https:/

Aurélien Rizk is a scientist and entrepreneur in drug discovery. Before focusing on the development of innovative mathematical modeling and simulation methods for drug Interdisciplinary Teamwork and Drug Development Yamina Berchiche and Aurelien Rizk emphasized the significance of interdisciplinary teamwork in drug and technology development, noting the challenges of communication Aurelien Rizk confirmed his attendance at the upcoming GPCR-Targeted Drug Discovery Summit in Boston.

GPCR Podcast Strategic Partners Dr. Josephine (Pina) Cardarelli About Dr. Additionally, they have a library of target GPCR heteromers for Oncology. Dr. Cardarelli is a drug development leader with extensive experience driving drug discovery teams in bringing She has extensive experience working with Biologics, and Antibody Drug Conjugates as well as experience GPCR Ecosystem Enjoying the Dr. GPCR Podcast? Leave a Review.

Full Agenda Adhesion GPCR workshop 2024 CINVESTAV, Mexico City, Mexico October 23-25 Download PDF Program formation, maintenance and degeneration Yimin Zou Antibody-drug conjugates targeting CD97 in glioblastoma Yimin Zou on the web UC San Diego Antibody-drug conjugates targeting CD97 in glioblastoma Dimitris Placantonakis To exploit this expression profile, we have developed antibody-drug conjugates (ADCs) targeting CD97, GPCR < Previous Session Next Session >

GPCR Podcast Strategic Partners Dr. GPCR podcast , your host and founder, Dr. GPCR Ecosystem, with the goal is to bring together GPCR scientists, biotech, and pharma leaders as well , grow, and thrive together to accelerate GPCR drug discovery and improve human health. GPCR Ecosystem Enjoying the Dr. GPCR Podcast? Leave a Review.

#gpcr#drgpcr Published on May 26, 2025 Category GPCR Weekly News How do GPCRs sense pH changes? Antagonism Drug discovery often assumes receptor inhibition follows simple rules—agonist binds, antagonist GPCR Podcast 4 days ago Molecular creativity in drug discovery Most pharmacologists are trained to chase That’s exactly what Terry’s Corner delivers this week: a deep dive into molecular creativity, rational design GPCR News 5 days ago

GPCR Podcast Strategic Partners You never know where your GPCR takes you with Dr. He has more than 20 years of experience in GPCR, primarily focused on drug discovery and developing new GPCR Podcast? Leave a Review. Collaboration Built an Innovation Engine From Pipettes to Platforms: The Evolution of GPCR Research How GPCR Spatial Signaling Sparked a Scientific Journey Thanks for listening to this podcast episode

GPCR Podcast Strategic Partners Dr. Prasenjit Saha About Dr. Specifically, I am interested in understanding dysregulated G-protein coupled receptor (GPCR) signaling Traditional drug discovery efforts have focused on agonists and antagonists that bind to the orthosteric ubiquitous class of plasma membrane receptors and serve as targets for more than one-third of all prescribed drugs GPCR Enjoying the Dr. GPCR Podcast? Leave a Review.

GPCR Affiliate Program and earn commissions by helping connect the global GPCR community. Share our ecosystem, courses, and events to advance drug discovery together. Dr. GPCR community. The Ecosystem is designed for all GPCR professionals to have an affordable and highly effective way to GPCR Ecosystem?

unveiled the cryo-EM structure of TAS2R14, the most promiscuous bitter taste receptor, bound to the drug This discovery reveals an unusual dual binding mode of FFA and offers tools for site-targeted compound design Published on December 5, 2024 Category GPCR Weekly News Ever wondered how we perceive bitterness? This discovery reveals an unusual dual binding mode of FFA and offers tools for site-targeted compound design signaling. ➡️ https://www.ecosystem.drgpcr.com/receptor-activation-and-signaling/a-bitter-anti-inflammatory-drug-binds-at-two-distinct-sites-of-a-human-bitter-taste-gpcr

GPCR Podcast Strategic Partners Murat Tunaboylu & Ben Holland About Murat Tunaboylu "Murat Tunaboylu, His current focus is to realise Antiverse’s mission: engineering the future of drug discovery." Murat Tunaboylu on the web Antiverse DSV Future of Drug Discovery Podcast Twist Bioscience LinkedIn Twitter GPCR Enjoying the Dr. GPCR Podcast? Leave a Review. Collaboration Built an Innovation Engine From Pipettes to Platforms: The Evolution of GPCR Research

GPCR Podcast Strategic Partners Chris Langmead Chris Langmead is Professor, Deputy Director, and Better He is an acknowledged expert in drug discovery, particularly in the field of psychiatry, where he has He has published over 70 research articles, reviews and book chapters on drug discovery, which have been GPCR Ecosystem Enjoying the Dr. GPCR Podcast? Leave a Review. Collaboration Built an Innovation Engine From Pipettes to Platforms: The Evolution of GPCR Research

GPCR Podcast Strategic Partners Robert Laprairie About Dr. Robert Laprairie Dr. Robert Laprairie is an Associate Professor and the Saskatchewan Research Chair in Drug Discovery and GPCR Ecosystem Enjoying the Dr. GPCR Podcast? Leave a Review. Collaboration Built an Innovation Engine From Pipettes to Platforms: The Evolution of GPCR Research How GPCR Spatial Signaling Sparked a Scientific Journey Thanks for listening to this podcast episode

Full Agenda Adhesion GPCR workshop 2024 CINVESTAV, Mexico City, Mexico October 23-25 Download PDF Program Our first main research aspect is the identification of endogenous ligand of GPCRs. Our third main research aspect is working mechanism of GPCR. Our fourth main research aspect is ligand coding mechanisms and structural aided drug discovery of GPCR (Cell 2021, 2023, Nature 2023b), bile acids or its derivatives by GPCRs (Nature 2020)."

Full Agenda Adhesion GPCR workshop 2024 CINVESTAV, Mexico City, Mexico October 23-25 Download PDF Program GPCR Community Presentation Breaking Barriers: My Journey from Mexico to the Heart of the Dr. GPCR Ecosystem and beyond About Monserrat Avila Zozaya "My doctoral research was focused on investigating My research focuses on understanding the molecular mechanisms of adhesion GPCRs (aGPCRs) in lymphatic GPCR < Previous Session Next Session >

GPCR Podcast Strategic Partners Dr. Oliver Hartley About Dr. Oliver Hartley Oliver Hartley is VP for Drug Discovery at Orion Biotechnology . GPCR Ecosystem Enjoying the Dr. GPCR Podcast? Leave a Review. Collaboration Built an Innovation Engine From Pipettes to Platforms: The Evolution of GPCR Research How GPCR Spatial Signaling Sparked a Scientific Journey Thanks for listening to this podcast episode

GPCR Podcast Strategic Partners Dr. Steven Foord About Dr. He also discovered and championed a novel prostaglandin EP4 drug candidate for development. GPCR Ecosystem Enjoying the Dr. GPCR Podcast? Leave a Review. Collaboration Built an Innovation Engine From Pipettes to Platforms: The Evolution of GPCR Research How GPCR Spatial Signaling Sparked a Scientific Journey Thanks for listening to this podcast episode

GPCR Podcast Strategic Partners Dr. Pierre Eftekhari About Dr. Pierre Eftekhari "Clinical physiologist and biologist , with more than 25 years of experience in drug development. have been engaged in GPCR cellular and clinical pharmacology as scientist or PI in neonatal I have participated and initiated methodologies for development of pharmacologically active anti-GPCR GPCR Enjoying the Dr. GPCR Podcast? Leave a Review.

GPCR Podcast Strategic Partners Steve McCloskey About Steve McCloskey Steve McCloskey is an Alumni from Scientists and Engineers working at the nanoscale, specifically protein engineering and small molecule drug GPCR Ecosystem Enjoying the Dr. GPCR Podcast? Leave a Review. Collaboration Built an Innovation Engine From Pipettes to Platforms: The Evolution of GPCR Research How GPCR Spatial Signaling Sparked a Scientific Journey Thanks for listening to this podcast episode

Principles of Pharmacology in Drug Discovery I Techniques for Effective Lead Optimization of Candidate still are the most prolific and fertile therapeutic drug targets; this course describes the essential of new Drugs. receive a comprehensive understanding of the unique science of pharmacology and how it can describe drug Modules: October 3rd: GPCR Project Initiation and Design for Discovery of New Molecules.

GPCR Podcast Strategic Partners Dr. Kari Johnson About this episode Dr. University before continuing her training as a postdoctoral fellow at the Vanderbilt Center for Neuroscience Drug Join me and learn more about how Kari studies GPCRs in basal ganglia circuits following chronic alcohol GPCR Ecosystem Enjoying the Dr. GPCR Podcast? Leave a Review. Collaboration Built an Innovation Engine From Pipettes to Platforms: The Evolution of GPCR Research

GPCR Podcast Strategic Partners Dr. Michel Bouvier About Dr. He is a world-renowned expert in the field of cell signaling and GPCRs and made seminal contributions to our understanding of this major class of drug targets. energy transfer (BRET) resulted in the development of screening assays that are now widely used for drug GPCR Ecosystem Enjoying the Dr. GPCR Podcast? Leave a Review.

Full Agenda Adhesion GPCR workshop 2024 CINVESTAV, Mexico City, Mexico October 23-25 Download PDF Program Activation: Direct Communication of Extracellular Region with Transmembrane Domain in a Holo-Adhesion GPCR point mutant knock-in mouse, H381S Frank Kwarcinski Tethered Peptide Activation Mechanism of Adhesion GPCRs ECR-mediated mechanism opens new possibilities for drugging aGPCRs. Frank Kwarcinski on the web LinkedIn Tethered Peptide Activation Mechanism of Adhesion GPCRs Peng Xiao