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Results found for "GPCR Therapeutics"
- Dr. Yamina Berchiche | Dr. GPCR Ecosystem
GPCR, an ecosystem designed to bring together stakeholders interested in using G-Protein Coupled Receptors (GPCRs) that control virtually everything in the body as drug targets. GPCR is to accelerate GPCR drug discovery by sharing the latest research and technology advances in the GPCR podcast. Dr. GPCR Ecosystem Enjoying the Dr. GPCR Podcast? Leave a Review.
- Game-changer for GPCR research! 🔬🧪 Molecular glues offer a new way to fine-tune receptor signaling, opening doors for next-gen drug discovery Subscribe to the Dr. GPCR Newsletter 📰 and get the latest GPCR News delivered to your inbox ➡️https://www.ecosystem.drgpcr.com/reviews/molecular-glues%3A-a-new-approach-to-modulating-gpcr-signaling-bias #gpcr #drgpcr | Dr. GPCR Ecosystem
GPCR Newsletter 📰 and get the latest GPCR News delivered to your inbox ➡️https://www.ecosystem.drgpcr.com /reviews/molecular-glues%3A-a-new-approach-to-modulating-gpcr-signaling-bias #gpcr #drgpcr Published on February 17, 2025 Category GPCR Weekly News Game-changer for GPCR research! GPCR Newsletter 📰 and get the latest GPCR News delivered to your inbox ➡️ https:// www.ecosystem.drgpcr.com /reviews/molecular-glues%3A-a-new-approach-to-modulating-gpcr-signaling-bias #gpcr #drgpcr Previous Next
- Eleonora Comeo | Dr. GPCR Ecosystem
We sat down to chat about GPCRs, synthesizing labeled ligands, and her unique position that allows her to work with GPCR scientists on 2 continents. GPCR Ecosystem Enjoying the Dr. GPCR Podcast? Leave a Review. Better Questions in Science: A Practical Guide for Emerging Researchers When the Islet Lit Up: Advancing GPCR Imaging in Native Tissue How Collaboration Sparked a GPCR Imaging Breakthrough in Chemical Biology Thanks
- Dr. Demet Araç | Dr. GPCR Ecosystem
They also discussed the ongoing developments in the GPCR field, the upcoming adhesion GPCR consortium GPCR field and the upcoming adhesion GPCR consortium meeting, which Anthony will be organizing in Mexico adhesion GPCRs. research in the GPCR (G protein-coupled receptor) field, specifically focusing on adhesion GPCRs. GPCR Podcast? Leave a Review.
- Did you know? 🌟 Researchers have developed reversibly photoswitchable allosteric modulators for Class A GPCRs! 🧬💡 These innovative compounds, “Photo-BQCisA” and “Photo-BQCtrAns,” offer subtype-selective precision by combining allosteric modulation with light control, paving the way for new therapeutic strategies targeting muscarinic receptors (M1-M5). 🔬✨ Learn more about this breakthrough in the Ecosystem! | Dr. GPCR Ecosystem
🌟 Researchers have developed reversibly photoswitchable allosteric modulators for Class A GPCRs! subtype-selective precision by combining allosteric modulation with light control, paving the way for new therapeutic Published on December 3, 2024 Category GPCR Weekly News Did you know? 🌟 Researchers have developed reversibly photoswitchable allosteric modulators for Class A GPCRs! subtype-selective precision by combining allosteric modulation with light control, paving the way for new therapeutic
- Brendan Wilkins | Dr. GPCR Ecosystem
Victor Chang Cardiac Research Institute where he investigated the orphan G protein-coupled receptor (GPCR Brendan’s PhD project focuses on the orphan GPCR GPR146. validate the proposed ligands of GPR146 in line with IUPHAR-NC guidelines on deorphanisation of orphan GPCRs GPCR Enjoying the Dr. GPCR Podcast? Leave a Review. Imaging in Native Tissue How Collaboration Sparked a GPCR Imaging Breakthrough in Chemical Biology Thanks
- Smells Like GPCR Spirit: Cracking Olfactory Codes with Alessandro Nicoli | Dr. GPCR Ecosystem
GPCRs, Receptors of Infinite Variety When asked about his favorite GPCR, Nicoli refused to pick. Keyword Cloud GPCR research community , Dr. GPCR ecosystem , GPCR online course , GPCR scientist network , GPCR drug discovery , GPCR training program , G protein-coupled receptors , GPCR podcast , GPCR webinar series , GPCR data platform Summary created GPCR Podcast? Leave a Review.
- New cryo-EM insights reveal how extracellular domains communicate with transmembrane regions in holo-adhesion GPCRs, uncovering mechanisms behind receptor activation. Subscribe to the Dr. GPCR Newsletter 📰 and get the latest GPCR News delivered to your inbox ➡️https://www.ecosystem.drgpcr.com/adhesion-gpcrs/conformational-coupling-between-extracellular-and-transmembrane-domains-modulates-holo-adhesion-gpcr-function #gpcr #drgpcr | Dr. GPCR Ecosystem
GPCR Newsletter 📰 and get the latest GPCR News delivered to your inbox ➡️https://www.ecosystem.drgpcr.com /adhesion-gpcrs/conformational-coupling-between-extracellular-and-transmembrane-domains-modulates-holo-adhesion-gpcr-function #gpcr #drgpcr Published on January 7, 2025 Category GPCR Weekly News New cryo-EM insights reveal how GPCR Newsletter 📰 and get the latest GPCR News delivered to your inbox ➡️ https://www.ecosystem.drgpcr.com /adhesion-gpcrs/conformational-coupling-between-extracellular-and-transmembrane-domains-modulates-holo-adhesion-gpcr-function
- Session V | Adhesion GPCR Workshop 2024 | Dr. GPCR Ecosystem
Full Agenda Adhesion GPCR workshop 2024 CINVESTAV, Mexico City, Mexico October 23-25 Download PDF Program Autoproteolysis And Cleavage Resistance Of Adhesion G Protein-Coupled Receptors Fabian Pohl Abstract "The GPCR Many ADGRs are autoproteo-lytically cleaved at the GPCR proteolysis site (GPS), an HXS/T motif within ) are a family of 32 mammalian proteins with a defining conserved GPCR autoproteolysis inducing (GAIN ) domain that catalyzes receptor self-cleavage at a GPCR proteolysis site (GPS).
- irreversible drugs post 3 | Dr. GPCR Ecosystem
lesson: Target depletion vs. replenishment dynamics — how offset rates control exposure windows, shape therapeutic GPCR Ecosystem #GPCR #DrGPCR #Pharmacology #DrugDiscovery #Kinetics #ReceptorPharmacology #MedicinalChemistry Operating cadence Attila Foris Dec 24, 2025 GPCR Binding Affinity Experiments: Interpreting Data With GPCR News Dec 18, 2025 Scientific Isolation: The Real Reason Early Biotechs Lose Traction The Quiet Drift GPCRs couple, decouple, isomerize, deplete tracers, and shift apparent affinity depending on stoichiometry
- Dylan Eiger | Dr. GPCR Ecosystem
Dylan's graduate research focuses on the mechanisms underlying biased signaling at GPCRs, specifically , the role of differential receptor phosphorylation (phosphorylation barcodes) and subcellular GPCR signaling He hopes to continue his research on biased agonism at GPCRs with a particular focus on the treatment GPCR Ecosystem Enjoying the Dr. GPCR Podcast? Leave a Review. Imaging in Native Tissue How Collaboration Sparked a GPCR Imaging Breakthrough in Chemical Biology Thanks
- Vaithish Velazhahan | Dr. GPCR Ecosystem
His Ph.D. work has been focused on understanding the structure and activation of Class D fungal GPCRs He has developed novel tools and methodologies to study fungal GPCRs which allowed the determination of the first structures of the prototypical fungal GPCR Ste2. GPCR Ecosystem Enjoying the Dr. GPCR Podcast? Leave a Review. Imaging in Native Tissue How Collaboration Sparked a GPCR Imaging Breakthrough in Chemical Biology Thanks
- Departure | Adhesion GPCR Workshop 2024 | Dr. GPCR Ecosystem
Full Agenda Adhesion GPCR workshop 2024 CINVESTAV, Mexico City, Mexico October 23-25 Download PDF Program
- Did you know allosteric modulators can change the GPCR G protein subtype selectivity? Have a look at this study to dive deep into its molecular mechanism. Subscribe to the Dr. GPCR Newsletter 📰 and get the latest GPCR News delivered to your inbox. | Dr. GPCR Ecosystem
GPCR Newsletter 📰 and get the latest GPCR News delivered to your inbox. the GPCR G protein subtype selectivity? GPCR Newsletter 📰 and get the latest GPCR News delivered to your inbox. ➡ https:// www.ecosystem.drgpcr.com /gpcr-binders-drugs-and-more/design-of-allosteric-modulators-that-change-gpcr-g-protein-subtype-selectivity #gpcr #drgpcr Previous Next Recent Articles
- Check out our #SpotifyWrapped 🚀! In 2024, Dr. GPCR reached listeners worldwide, sparking conversations about GPCRs with top experts. Thank you for tuning in! 📊🎙️ ✳️Check out our top episode: https://www.ecosystem.drgpcr.com/dr-gpcr-podcast/ep-148-with-dr-arthur-christopoulos #gpcr #drgpcr | Dr. GPCR Ecosystem
GPCR reached listeners worldwide, sparking conversations about GPCRs with top experts. 📊🎙️ ✳️Check out our top episode: https://www.ecosystem.drgpcr.com/dr-gpcr-podcast/ep-148-with-dr-arthur-christopoulos #gpcr #drgpcr Published on January 29, 2025 Category Check out our #SpotifyWrapped 🚀! GPCR reached listeners worldwide, sparking conversations about GPCRs with top experts. #gpcr #drgpcr Previous Next Recent Articles
- Did you know that GPR180 helps regulate lipid metabolism and may play a role in preventing obesity? recent study shows that overexpression of GPR180 in adipose tissue improves lipid metabolism and protects against HFD-induced obesity, while its knockout worsens lipid accumulation. This finding highlights GPR180 as a potential therapeutic target for metabolic disorders! Catch up on this exciting research in the Ecosystem today! 🏆📖 You’ll need to register, but don’t worry—it’s free! ➡️https://www.ecosystem.drgpcr.com/gpcrs-in-cardiology-endocrinology-and-taste/gpr180-reduces-adiposity-by-inhibiting-lipogenesis-and-fatty-acid-uptake-in-adipocytes #gpcr #drgpcr #metabolism #obesity | Dr. GPCR Ecosystem
This finding highlights GPR180 as a potential therapeutic target for metabolic disorders! #gpcr #drgpcr #metabolism #obesity Published on March 3, 2025 Category GPCR Weekly News Did you know This finding highlights GPR180 as a potential therapeutic target for metabolic disorders! #gpcr #drgpcr #metabolism #obesity Previous Next Recent Articles Why Biotech Fundraising Fails Due to Operating cadence Attila Foris Dec 24, 2025 GPCR Binding Affinity Experiments: Interpreting Data With
- A large-scale analysis of GPCR molecular dynamics reveals hidden allosteric sites and lateral gateways, unlocking new possibilities for drug discovery. Subscribe to the Dr. GPCR Newsletter 📰 and get the latest GPCR News delivered to your inbox ➡️https://www.ecosystem.drgpcr.com/structural-and-molecular-insights-into-gpcr-function/large-scale-investigation-of-gpcr-molecular-dynamics-data-uncovers-allosteric-sites-and-lateral-gateways #gpcr#drgpcr | Dr. GPCR Ecosystem
GPCR Newsletter 📰 and get the latest GPCR News delivered to your inbox ➡️https://www.ecosystem.drgpcr.com /structural-and-molecular-insights-into-gpcr-function/large-scale-investigation-of-gpcr-molecular-dynamics-data-uncovers-allosteric-sites-and-lateral-gateways #gpcr#drgpcr Published on March 17, 2025 Category GPCR Weekly News A large-scale analysis of GPCR molecular GPCR Newsletter 📰 and get the latest GPCR News delivered to your inbox ➡️ https:// www.ecosystem.drgpcr.com /structural-and-molecular-insights-into-gpcr-function/large-scale-investigation-of-gpcr-molecular-dynamics-data-uncovers-allosteric-sites-and-lateral-gateways
- A GPCR imaging breakthrough that didn’t start in a grant proposal | Dr. GPCR Ecosystem
A collaboration between chemistry and biology sparked a GPCR imaging breakthrough, leading to new chemical Home → Flash News → A GPCR imaging breakthrough that didn’t start in a grant proposal A GPCR imaging experiments, the pivot to chemical probes, and the trust-driven partnership that sparked a new era in GPCR Operating cadence Attila Foris Dec 24, 2025 GPCR Binding Affinity Experiments: Interpreting Data With GPCR News Dec 18, 2025 Scientific Isolation: The Real Reason Early Biotechs Lose Traction The Quiet Drift
- Dr. Benjamin Myers | Dr. GPCR Ecosystem
Ben’s research focuses on Smoothened and other class F GPCRs which play essential roles in embryonic These studies have revealed new and unexpected ways for membrane lipids to regulate GPCR activity and for GPCRs to control intracellular kinases. More recently, Ben’s lab has begun studying GPCR signaling pathways that operate within the primary cilium GPCR Ecosystem Enjoying the Dr. GPCR Podcast? Leave a Review.
- Dr. Elva Zhao | Dr. GPCR Ecosystem
After her Ph.D., she moved to Australia and continues working on GPCRs. Her current research focuses on class B GPCRs and understanding how GPCR signaling and function is mediated Join me to learn more about Elva, class B GPCRs, and Tilly. Dr. GPCR Ecosystem Enjoying the Dr. GPCR Podcast? Leave a Review. Imaging in Native Tissue How Collaboration Sparked a GPCR Imaging Breakthrough in Chemical Biology Thanks
- Dr. Pierre Eftekhari | Dr. GPCR Ecosystem
physiologist and biologist , with more than 25 years of experience in drug development. have been engaged in GPCR I have participated and initiated methodologies for development of pharmacologically active anti-GPCR or contributed in 38 published scientific work mainly in the field of immunology and pharmacology of GPCR Since the creation of Inoviem scientific in Nov. 2011 by myself we have been regularly working with GPCRs GPCR Enjoying the Dr. GPCR Podcast? Leave a Review.
- Every receptor tells a story | Dr. GPCR Ecosystem
Every receptor tells a story but GPCRs speak a language of organization. Dr. Michelle Halls unpacks how GPCR signaling isn’t just about ligand–receptor interaction. a story Published on November 11, 2025 Category Dr.GPCR Podcast Every receptor tells a story — but GPCRs Michelle Halls unpacks how GPCR signaling isn’t just about ligand–receptor interaction. signaling: 👉 https://www.ecosystem.drgpcr.com/dr-gpcr-podcast/leadership-luck-and-gpcr-signaling #GPCR
- How does nanoscale GPCR organization shape signaling? 🤔 We explore this & more with Dr. Gabriele Kockelkoren, a physicist-turned-biologist with expertise in GPCR spatial dynamics. And if you wonder what his favorite GPCR could be, here’s the answer 😉 ✅Listen now Ep 162 with Dr. Gabriele Kockelkoren #gpcr #drgpcr | Dr. GPCR Ecosystem
Home → Flash News → How does nanoscale GPCR organization shape signaling? Gabriele Kockelkoren, a physicist-turned-biologist with expertise in GPCR spatial dynamics. Gabriele Kockelkoren #gpcr #drgpcr Published on March 20, 2025 Category Dr. GPCR Podcast How does nanoscale GPCR organization shape signaling? Gabriele Kockelkoren #gpcr #drgpcr Previous Next Recent Articles
- Empowering Drug Discovery for the GPCR Community with Dr. Justin English | Dr. GPCR Ecosystem
<< Back to podcast list Strategic Partner(s) Empowering Drug Discovery for the GPCR Community with Dr GPCR Enjoying the Dr. GPCR Podcast? Leave a Review. Better Questions in Science: A Practical Guide for Emerging Researchers When the Islet Lit Up: Advancing GPCR Imaging in Native Tissue How Collaboration Sparked a GPCR Imaging Breakthrough in Chemical Biology Thanks
- Developing new tools to uncover GPCR signaling patterns with Remi Janicot | Dr. GPCR Ecosystem
<< Back to podcast list Strategic Partner(s) Developing new tools to uncover GPCR signaling patterns Mikel Garcia-Marcos seemed like a good fit as GPCRs are integral to the functioning of the nervous system My particular projects revolve around developing new tools to study GPCR activity in ways that were not GPCR Podcast? Leave a Review. Imaging in Native Tissue How Collaboration Sparked a GPCR Imaging Breakthrough in Chemical Biology Thanks
- Let’s connect the dots! Update your Dr. GPCR profile to make meaningful connections in the global GPCR network 🌐 ✳️Visit https://www.ecosystem.drgpcr.com/account/my-account and fill out the boxes with your most updated information. #gpcr #drgpcr | Dr. GPCR Ecosystem
GPCR profile to make meaningful connections in the global GPCR network 🌐 ✳️Visit https://www.ecosystem.drgpcr.com #gpcr #drgpcr Published on January 8, 2025 Category Dr. GPCR Profiles Let’s connect the dots! GPCR profile to make meaningful connections in the global GPCR network 🌐 ✳️Visit https://www.ecosystem.drgpcr.com #gpcr #drgpcr Previous Next Recent Articles
- Stay ahead in the GPCR field 💼 Updating your profile ensures you’re ready for the next opportunity. ✳️Go to https://www.ecosystem.drgpcr.com/account/my-account and let our GPCR-exclusive community know what you’re up to #gpcr #drgpcr | Dr. GPCR Ecosystem
Home → Flash News → Stay ahead in the GPCR field 💼 Updating your profile ensures you’re ready for the ✳️Go to https://www.ecosystem.drgpcr.com/account/my-account and let our GPCR-exclusive community know what you’re up to #gpcr #drgpcr Published on January 29, 2025 Category Dr. GPCR Profiles Stay ahead in the GPCR field 💼 Updating your profile ensures you’re ready for the next community know what you’re up to #gpcr #drgpcr Previous Next Recent Articles
- Lauren Celano | Dr. GPCR Ecosystem
GPCR podcast episode, we sat down to chat with Lauren Celano to talk about career options for Ph.D.’s GPCR Ecosystem Enjoying the Dr. GPCR Podcast? Leave a Review. Better Questions in Science: A Practical Guide for Emerging Researchers When the Islet Lit Up: Advancing GPCR Imaging in Native Tissue How Collaboration Sparked a GPCR Imaging Breakthrough in Chemical Biology Thanks
- Dr. Maria Waldhoer | Dr. GPCR Ecosystem
GPCRs led Maria to Thue W. Even though Maria stumbled upon the GPCR field, her 20 years in both academia and in the industry working on GPCRs make her a strong and dedicated scientific leader. GPCR Ecosystem Enjoying the Dr. GPCR Podcast? Leave a Review. Imaging in Native Tissue How Collaboration Sparked a GPCR Imaging Breakthrough in Chemical Biology Thanks
- Dr. Tobi Langenhan | Dr. GPCR Ecosystem
studies, I joined the lab of Dr Andreas Russ at the Department of Biochemistry and first came across GPCRs , particularly the receptor family I have been investigating ever since: adhesion GPCRs. pick apart the physiological and pharmacological principles that underlie the workings of adhesion GPCRs This entails the deciphering of cellular and organ functions, which require individual adhesion GPCRs GPCR Enjoying the Dr. GPCR Podcast? Leave a Review.















