Search Results

translational pharmacologists, biotech discovery teams, and decision-makers who need concise, credible, high-value

. -            High-throughput applications Bright and stable fluorescent ligands can be used in HTS,

Forge high-value connections in an intimate setting.

That’s exactly what Terry’s Corner delivers this week: high-impact insight into GPCR allostery, crafted

A small step toward leveling the playing field.

The chemokines CXCL8 and CXCL12: molecular and functional properties, role in disease and efforts towards

The development of antibodies directed towards an OR could either drive receptor inactivation or activation

Where high-throughput screening saw chaos, Ajay saw patterns waiting to be decoded.

For high-throughput screens where sensitivity isn’t critical, you’ll save time by running fewer replicates

Structural and Molecular Insights into GPCR Function Structure-Activity Relationship Study of the High-Affinity

Prior to this report we did not know how different serotonin receptor subtypes which share high sequence

S-transferase; HCC: hepatocellular carcinoma; HBV: hepatitis B virus; HBx: hepatitis B virus X protein; HMGB1: high

Cone Pigment Activation Molecular dynamics-based identification of binding pathways and two distinct high-affinity

dependent signalling correlated with reduced mobilisation of lytically-infected DC to draining lymph node high

GPCR Premium: Sneak Peek Here’s a curated, high-signal preview of what Premium Members get this week—no

A high-affinity ligand often has higher efficacy, but the relationship is not linear.

GPCR Premium: Sneak Peek Here’s a fast, high-level preview of what Premium Members are unpacking this

here ➤ Discovery on Target 2025 – GPCR Speaker Spotlight DOT 2025 (Sept 22–25, Boston) is set to be a high-signal

Herbal Compounds as Potential Drugs for Chronic Myeloid Leukemia Methods & Updates in GPCR Research High-throughput

site-selective activation of mTOR GPCR Binders, Drugs, and more Molecular glues as potential GPCR therapeutics A high-affinity

translational success:  How post-COVID insights and unconventional decision-making shaped Serafini’s high-impact

lipid second messenger signaling Methods & Updates in GPCR Research An image-based abplex method for high-throughput

Insomnia Patient in its Phase 3 Clinical Trial of Daridorexant in South Korea Septerna Touches New High

Recently, several high-throughput screening (HTS) assays for ERK activation have been developed, each

A huge thank you to our amazing speakers and everyone who showed up.

sets the activity pattern in the C. elegans egg-laying circuit Methods & Updates in GPCR Research High-throughput

receptor sensor GPCRs in Oncology and Immunology Phase 1/2 study of sorafenib added to cladribine, high-dose

Should Enroll Now: Cost-effective & Distinctive Educational Experience Affordable courses that maintain high-quality

The Tissue Penetration Trap Here’s a paradox: high-affinity, slow-offset compounds can undermine their

Prostaglandin E2 EP3 Receptor Has Disparate Effects on Islet Insulin Secretion and Content in β-cells in a High