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The β2-adrenergic receptor (β2AR) is a prototypical and extensively studied GPCR that can provide insight

You’ll see why tight binding can backfire on tissue penetration, where k_inact/K_I beats classic Ki,

“You can try, try, try—and fail, fail, fail,” Eric says.

This can be deduced from the qRT-PCR assays; triggering CB1 receptors amplifies both NR4A1 and NR4A3

Terry Kenakin breaks down receptor pharmacology, functional selectivity, and ligand bias in a way you can

Recently, Suchismita Roy et al. have explored how growth factors can modulate canonical G protein signaling

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GPCR Activation and Signaling How can we improve the measurement of receptor signaling bias?

in an in vitro system, hints at a role as an inflammatory mediator and supports the notion that IL-6 can

Therefore, docking performance against GPCR targets can be estimated in advance based on docking target

In 2017, Gupte et al. introduced GPCR priming, which posits that non-cognate G proteins can enhance the

If you have any research you would like to showcase to our community, you can submit a poster presentation

You can now watch the live talk recordings from the previous symposiums, check them out here.

You can always adjust your email preferences in your account settings Below is your Classified GPCR News

You can always adjust your email preferences in your account settings Below is your Classified GPCR News

You can always adjust your email preferences in your account settings.

Premium members can always go back and watch the recorded talks at any time.

You can find more information about them on the Live Talks page and mark your calendar HERE.

Topics include the complex pleiotropic behaviors of GPCRs and how these can be harnessed for innovative

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You can always adjust your email preferences in your account settings. For Dr.

You can find more details about the speakers on the Live Talks page, and make sure to mark your calendar

Evidence that RXFP4 is located in enterochromaffin cells and can regulate production and release of serotonin

Allow registrants to appreciate the incredible versatility of GPCRs and how small molecules can affect

Registrations are closed but you can send an email to gpcrretreat@uottawa.ca to be added to the waitlist

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If you missed it, don't worry – you can catch the sessions on-demand with a premium membership.

You can submit your poster abstracts using this form and short talks will be selected from abstracts.

Now you can submit your job opening and offer a position in an exclusive GPCR community around the globe

GPCR Ecosystem group, where you can find Dr.