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- Xylazine, Fentanyl, and the Fight for Breath with Catherine Demery | Dr. GPCR Ecosystem
How GPCR pharmacology connects molecular insights to real-world interventions. how fentanyl and xylazine shut down breathing through different mechanisms—work that blends receptor pharmacology now and see how one scientist is turning molecules into a mission, bridging the gap between receptor pharmacology GPCR ecosystem , GPCR training program , GPCR podcast , opioid pharmacology , xylazine research , mu opioid receptor , pharmacogenomics , fentanyl epidemic , preclinical pharmacology Enjoying the Dr.
- Pharmacological and Genetic Preclinical Models of Ghrelin Receptor Functional Selectivity to Investigate Metabolic Disease Pathophysiology
About Program Registration Logo Contest Committee Sponsors GPCR Retreat Program < Back to schedule Pharmacological and Genetic Preclinical Models of Ghrelin Receptor Functional Selectivity to Investigate Metabolic Disease , Durham, NC 27710. 3-National Center for Advancing Translational Sciences (NCATS), NIH Division of Preclinical With my expertise in reward behavior, neurophysiology, GPCR signaling, and preclinical drug development
- Yamina's Corner | Dr. GPCR Ecosystem
accelerate your pipeline Book My Consultation Critical Bottlenecks in Your GPCR Pipeline ❌ Overwhelming pharmacology Actionable Scientific Validation: Ensure target companies execute the right GPCR pharmacology experiments With over two decades dedicated to GPCR pharmacology across biotech, academia, and the non-profit sector to complex pharmacological programs. Let’s talk about how I support GPCR discovery, pharmacology strategy, and cross-functional execution
- Chris Langmead | Dr. GPCR Ecosystem
discovery, particularly in the field of psychiatry, where he has led multiple projects into late stage preclinical He has a degree and PhD in pharmacology from Queens' College, Cambridge and University College London in 2012, and was the recipient of the British Pharmacological Society Novartis Prize in 2017. Chris serves on the editorial boards of the British Journal of Pharmacology, ACS Chemical Neuroscience , ACS Pharmacology & Translational Science and Frontiers in Pharmacology.
- Irfan Dhanidina, Dr. Kathleen Caron and Dr. Lauren Slosky | Dr. GPCR Ecosystem
Biotechnology, I work at the intersection of science and business, which includes target selection, preclinical Caron is also past Associate Editor at JCI and served as the inaugural Associate Editor at ACS-Pharmacology Lauren Slosky "Lauren Slosky is an Assistant Professor in the Department of Pharmacology and a member Integrating GPCR biology, behavioral pharmacology, and systems neuroscience approaches, the Slosky Lab She is currently a faculty trainer for the University of Minnesota's MS and Ph.D. programs in Pharmacology
- A Brief History of allosteric modulation with Dr. Arthur Christopoulos | Dr. GPCR Ecosystem
Arthur Christopoulos " Arthur Christopoulos is the Professor of Analytical Pharmacology and the Dean , medicinal chemistry, and preclinical models of behaviour and disease. and Toxicologists; the British Pharmacological Society’s Gaddum Memorial Award; the IUPHAR Sir James Black Analytical Pharmacology Lecturer; the GSK Award for Research Excellence and a Doctor of Laws ( Since 2014, Clarivate Analytics have annually named him a Highly Cited Researcher in ‘Pharmacology &
- Session III | Adhesion GPCR Workshop 2024 | Dr. GPCR Ecosystem
bioSens-All: A Multiparametric BRET-Based Platform for Comprehensive Profiling of adhesion GPCR Signaling and Pharmacology-Enabling dissociation across different species, we plan to adapt this technology for high-throughput screening of pharmacological examples will demonstrate how the bioSens-All platform was used to advance projects from discovery to preclinical Department of Pharmacology-Physiology, Université de Sherbrooke, Sherbrooke, Quebec, Canada 2. Our research aims to leverage this knowledge to identify novel pharmacological targets and contribute
- Biotech Growth | Dr. GPCR Ecosystem
I work with early-stage biotechs—typically preclinical through IND-enabling—who need strategic clarity Let’s talk about how I support GPCR discovery, pharmacology strategy, and cross-functional execution
- Dr. Arthur Christopoulos | Dr. GPCR Ecosystem
Arthur Christopoulos " Arthur Christopoulos is the Professor of Analytical Pharmacology and the Dean , medicinal chemistry, and preclinical models of behaviour and disease. and Toxicologists; the British Pharmacological Society’s Gaddum Memorial Award; the IUPHAR Sir James Black Analytical Pharmacology Lecturer; the GSK Award for Research Excellence and a Doctor of Laws ( Since 2014, Clarivate Analytics have annually named him a Highly Cited Researcher in ‘Pharmacology &
- Dr. Arthur Christopoulos | Dr. GPCR Ecosystem
Arthur Christopoulos " Arthur Christopoulos is the Professor of Analytical Pharmacology and the Dean , medicinal chemistry, and preclinical models of behaviour and disease. and Toxicologists; the British Pharmacological Society’s Gaddum Memorial Award; the IUPHAR Sir James Black Analytical Pharmacology Lecturer; the GSK Award for Research Excellence and a Doctor of Laws ( Since 2014, Clarivate Analytics have annually named him a Highly Cited Researcher in ‘Pharmacology &
- Applying Pharmacology to Drug Discovery
Applying Pharmacology to Drug Discovery by Terry Kenakin | Dr. GPCR Courses Applying Pharmacology to Drug Discovery Dr. Pharmacology is a unique discipline and is critical to drug discovery. What makes each drug type unique to therapeutic pharmacology? 3. Modules: Week 1 - Fundamentals of Pharmacology Week 2 - Characterizing Agonists Week 3 - Characterizing
- Session VI | Adhesion GPCR Workshop 2024 | Dr. GPCR Ecosystem
early in Alzheimer’s disease, and subsequent massive loss of synapses are closely correlated with the decline Collectively, these data suggest that ADCs targeting CD97 impair tumor growth in preclinical GBM models Javitch1,2 1Departments of Psychiatry and Molecular Pharmacology and Therapeutics, Columbia University initially became interested in GPCR signal transduction during my graduate training in the Department of Pharmacology
- GPCR Courses
premium to get access The Practical Assessment of Signaling Bias Signaling bias is an inherent feature of pharmacology Yamina Berchiche 🔒 Premium Content Watch recording Applying Pharmacology to Drug Discovery Class 1 - Fundamentals of Pharmacology Class 2 - Characterizing Agonists Class 3 - Characterizing Antagonists and biased agonism Class 3 - Antagonist pharmacology and binding assay analysis Class 4 - New dimensions Also super-valuable for those of us learning how to teach pharmacology Anonymous Dr.
- Complex Allosteric Cannabinoid Receptor Pharmacology
Committee Sponsors GPCR Retreat Program < Back to schedule Complex Allosteric Cannabinoid Receptor Pharmacology Robert and his lab have been interested in the molecular pharmacology of cannabinoids for nearly 10 years
- GPCR Retreat Schedule 2023
in Parkinson's Disease Ali Salahpour University of Toronto Read More Friday, November 3rd / 9:45 AM Pharmacological and Genetic Preclinical Models of Ghrelin Receptor Functional Selectivity to Investigate Metabolic Disease Monash University Read More Friday, November 3rd / 11:30 AM Complex Allosteric Cannabinoid Receptor Pharmacology 00 PM Coffee Break 4 Read More Friday, November 3rd / 3:30 PM G Proteins and GPCRs in Cancer: Novel Precision
- Terry's Corner is Officially LIVE! 🎉 This is your new go-to for mastering drug discovery pharmacology. No fluff, just clear, on-demand insights from Terry Kenakin. Building core expertise? Master dose-response, binding, kinetics, and foundational models. Driving drug discovery? Apply pharmacology to selectivity, ADME, and strategic decision-making. An experienced drug hunter? Sharpen your edge with allosteric bias, residence time, and translational PK/PD. Learn on-demand, apply immediately: https://terrykenakin.com #DrGPCR #GPCR #pharmacology #TerrysCorner #DrugDiscovery | Dr. GPCR Ecosystem
🎉 This is your new go-to for mastering drug discovery pharmacology. Apply pharmacology to selectivity, ADME, and strategic decision-making. An experienced drug hunter? Learn on-demand, apply immediately: https://terrykenakin.com #DrGPCR #GPCR #pharmacology #TerrysCorner 🎉 This is your new go-to for mastering drug discovery pharmacology. Apply pharmacology to selectivity, ADME, and strategic decision-making. An experienced drug hunter?
- Unlock your pharmacology potential with Terry’s Corner. No fluff. Just clear, on-demand insight from Dr. Terry Kenakin—built for scientists at every level. 🟢 Building core expertise? Learn dose-response, agonism, binding, bias, kinetics, and the models that build real confidence. 🟢 Driving drug discovery? Apply pharmacology to selectivity, ADME, early safety, and smarter decision-making. 🟢 Already a drug hunter? Sharpen your edge with allosteric modulation, residence time, molecular dynamics, and translational PK/PD. Learn on-demand. Apply immediately. Early access begins July 1 → https://www.terrykenakin.com #pharmacology #GPCRscience #drugdiscovery #TerrysCorner #biotechtraining | Dr. GPCR Ecosystem
Home → Flash News → Unlock your pharmacology potential with Terry’s Corner. No fluff. Apply pharmacology to selectivity, ADME, early safety, and smarter decision-making. 🟢 Already a drug Early access begins July 1 → https://www.terrykenakin.com #pharmacology #GPCRscience #drugdiscovery # Apply pharmacology to selectivity, ADME, early safety, and smarter decision-making. 🟢 Already a drug Early access begins July 1 → https://www.terrykenakin.com #pharmacology #GPCRscience #drugdiscovery #
- What’s one key piece of advice from Ian Chronis in Ep.164 of the Dr.GPCR Podcast?Listen to other scientists’ research—it’s a great way to stay motivated and inspired 🚀 Don’t miss this insightful conversation on GPCRs, pharmacology, and scientific discovery! ✅ https://buff.ly/FTB69y9 #GPCR #DrGPCR #SciencePodcast #Pharmacology #CancerResearch | Dr. GPCR Ecosystem
research—it’s a great way to stay motivated and inspired 🚀 Don’t miss this insightful conversation on GPCRs, pharmacology ✅ https://buff.ly/FTB69y9 #GPCR #DrGPCR #SciencePodcast #Pharmacology #CancerResearch Published on April research—it’s a great way to stay motivated and inspired 🚀 Don’t miss this insightful conversation on GPCRs, pharmacology ✅ https://buff.ly/FTB69y9 #GPCR #DrGPCR #SciencePodcast #Pharmacology #CancerResearch Previous Next Recent
- 🎧 "You will always feel like you know nothing— and that’s completely fine." In Ep.162 of the Dr.GPCR Podcast, Dr. Gabriele Kockelkoren shares: 🔬 How GPCR spatial organization shapes signaling and drug responses 🌍 His interdisciplinary journey from physics to pharmacology 💡 Why embracing the unknown is key to scientific breakthroughs A must-listen for biophysicists, pharmacologists, and drug hunters pushing the boundaries of discovery! 🎙️ Tune in now:Ep 162 with Dr. Gabriele Kockelkoren #DrGPCR #GPCR #Biophysics #Pharmacology #DrugDiscovery #SciencePodcast | Dr. GPCR Ecosystem
spatial organization shapes signaling and drug responses 🌍 His interdisciplinary journey from physics to pharmacology 💡 Why embracing the unknown is key to scientific breakthroughs A must-listen for biophysicists, pharmacologists Gabriele Kockelkoren #DrGPCR #GPCR #Biophysics #Pharmacology #DrugDiscovery #SciencePodcast Published spatial organization shapes signaling and drug responses🌍 His interdisciplinary journey from physics to pharmacology Gabriele Kockelkoren #DrGPCR #GPCR #Biophysics #Pharmacology #DrugDiscovery #SciencePodcast Previous
- Applying Pharmacology to Drug Discovery | Dr. GPCR Ecosystem
Applying Pharmacology to Drug Discovery Dr.
- pharmacology at your fingertips terrys corner launches | Dr. GPCR Ecosystem
Home → Flash News → pharmacology at your fingertips terrys corner launches Published on July 4, 2025 Category GPCR Weekly News Stronger pharmacology drives smarter decisions in GPCR discovery. https://www.ecosystem.drgpcr.com/post/pharmacology-at-your-fingertips-terry-s-corner-launches #DrGPCR #GPCR #DrugDiscovery #pharmacology #biotechnews #terrykenakin #GPCRconsulting Previous Next Recent Articles
- 10 GPCR pharmacology lessons. Zero fluff. Launching July 1, Terry’s Corner gives you the clarity and confidence to make better decisions—starting with: • The role of pharmacology in discovery strategy • Black & Leff’s operational model—finally made practical • Binding curves, orthosteric vs allosteric function, and real vs apparent affinity • Molecular dynamics and how they guide ligand design • Why Terry built this—and how it sharpens your next move 📅 Learn anytime. New course every week. 📬 Subscribe to The Kenakin Brief → https://www.terrykenakin.com #GPCRscience #drugdiscovery #TerrysCorner #GPCRpharmacology #ligandbinding | Dr. GPCR Ecosystem
Home → Flash News → 10 GPCR pharmacology lessons. Zero fluff. s Corner gives you the clarity and confidence to make better decisions—starting with: • The role of pharmacology TerrysCorner #GPCRpharmacology #ligandbinding Published on June 30, 2025 Category Terry's Corner 10 GPCR pharmacology Corner gives you the clarity and confidence to make better decisions—starting with: 🟢 The role of pharmacology
- master gpcr pharmacologic models before its too late | Dr. GPCR Ecosystem
Home → Flash News → master gpcr pharmacologic models before its too late Published on July 11, 2025 Category Terry’s Corner breaks down the 4 pharmacologic models that separate forecasting from guessing. Dr. utm_content=bufferd9b30&utm_medium=social&utm_source=twitter.com&utm_campaign=buffer #GPCR #Pharmacology
- GPCRs and the Science Behind Pain and Recovery with Dr. Alex Serafini | Dr. GPCR Ecosystem
Although not a self-proclaimed GPCR specialist, Serafini found himself repeatedly drawn to them, or more precisely equally focused on sex differences in pain processing and the failure of "one-size-fits-all" models in pharmacology Whether it’s challenging legacy targets, redefining preclinical models, or exploring the epigenetic inheritance
- Dr. Gunnar Schulte | Dr. GPCR Ecosystem
Gunnar Schulte Gunnar Schulte is a Professor in receptor pharmacology and research group leader for the section Receptor Biology and Signaling at the Department of Physiology and Pharmacology. has a background in biochemistry from the Free University in Berlin/Germany and a Ph.D. in molecular pharmacology , British Journal of Pharmacology, Pharmacological Reviews, and The Journal of Biological Chemistry. General Research Interest: The focus in the Schulte lab is on Frizzled signaling and pharmacology aiming
- Principles of Pharmacology in Drug Discovery I | Dr. GPCR Ecosystem
Principles of Pharmacology in Drug Discovery I Dr.
- Advanced data analysis for GPCR pharmacology | Dr. GPCR Ecosystem
Advanced data analysis for GPCR pharmacology Dr.
- Principles of Pharmacology in Drug Discovery II | Dr. GPCR Ecosystem
Principles of Pharmacology in Drug Discovery II Dr.
- terrys corner no fluff pure insight | Dr. GPCR Ecosystem
✨ We've poured our passion for pharmacology into creating this essential resource, designed to meet you Ready to: Strengthen your pharmacology fundamentals? Terry's Corner helps you make better decisions through better pharmacology. Enroll now: https://www.terrykenakin.com #pharmacology #GPCRscience #drugdiscovery #TerrysCorner #biotechtraining
- Courses (All) - Premium | Dr. GPCR Ecosystem
The Practical Assessment of Signaling Bias Signaling bias is an inherent feature of pharmacology, influencing Yamina Berchiche 🔒 Premium Content Watch recording Applying Pharmacology to Drug Discovery Class 1 - Fundamentals of Pharmacology Class 2 - Characterizing Agonists Class 3 - Characterizing Antagonists and biased agonism Class 3 - Antagonist pharmacology and binding assay analysis Class 4 - New dimensions Also super-valuable for those of us learning how to teach pharmacology Anonymous Dr.













