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Systems That Drive Progress:  From assay tracking to data workflows, I design simple, scalable tools

who has just released an incredible article on our site and a GPCR Paper with his team: Targeted Drug Design November 14th : The Application of GPCR Ligand Kinetics to Candidate Design.

Group Corporation (“the Company”; TSE: 4565), the world leader in GPCR-focused structure-based drug design

Our updated course schedule is designed to fit seamlessly into your routine, offering an enriched learning  Boston, MA 📅 October 2 -3, 2024 Join top researchers to explore the latest in GPCR-targeted drug design

We designed an integrative approach to improve comparative modeling of TAS2Rs.

co-internalization Kilian Roßmann , Ramona Birke , Joshua Levitz , Ben Jones , Johannes Broichhagen Design extracellular loops on a soluble scaffold enabled the discovery of antibodies, which recognized native receptor Design

Here’s what I bring: Biology-First Strategy I’ve designed GPCR assays, led collaborations across research

brain vs. peripheral contributions to metabolic therapy Guide how next-generation incretin drugs are designed

restoration of tension in epithelial cells GPCR Binders, Drugs, and more Advances in structure-based drug design copolymers and SMALPs as a platform for investigating GPCRs Reviews, GPCRs, and more Fragment-Based Design

understandings of CB2 signaling, tools that preserve cellular context will be increasingly important for designing Three-dimensional quantitative structure–selectivity relationships analysis guided rational design of

We designed and synthetized peptides that interfered with integrin αIIb binding (pCIB and pCIBm) or mimicked

Nasdaq debutante Septerna swells its IPO to $331m Nxera Pharma and Antiverse Enter Collaboration To Design Using Generative AI Zombie Fungi Hijack Hosts’ Brains GPCR Therapeutics, Inc. has received Orphan Drug Designation

Our refreshed schedule is designed to fit seamlessly into your calendar and enhance your learning experience (October 2-3, 2024, in Boston and online) gathers top researchers to explore the latest advances in designing

The pharmacological profiles and mechanistic insights of our study provide clues for the future design

The process of designing and evaluating biased ligands for GPCRs is complex but essential for understanding Advances in understanding the structural and mechanistic aspects of biased GPCR signaling are crucial for designing

MQ1-K39A represents the first step in the improvement of the MQ1 design from a medicinal perspective.

to PK–PD dissociation, Kenakin equips you with the kinetic models and biological context needed to design

Kenakin’s latest   lecture delivers exclusive, real-world insight designed to equip you to move beyond

Logo Contest : Let your creativity shine by submitting your design for the Logo Contest before August

At Celtarys, our GPCR fluorescent ligands are designed with a variety of photophysical properties to

radioligand binding but suppresses functional response, it’s not broken pharmacology—it’s biology working as designed

receptor, which could participate in the recognition of MT1-selective ligands and may be exploited in the design

GPCR Binders, Drugs, and more Rational design of highly stabilized and selective adrenomedullin analogs

Methods: To address this question, we studied mice that express a Gs-coupled designer G protein-coupled

GPCR University content, and an integrated view of publications, events, insights, and opportunities designed

At Celtarys, we support this transition by offering optimized fluorescent ligands specifically designed

lectures, classified industry news, priority event alerts, job opportunities, and insider commentary—designed

beyond natural agonist analogs Awareness of how GPCR allostery and biased signaling are redefining drug design

translational research models, further refining his interest in bridging molecular insights with therapeutic design

Methods & Updates in GPCR Research A coiled-coil-based design strategy for the thermostabilization of