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- What's Going On with GPCRs?! Find Out in This Week's Update! ⦿ Nov 4 - 10, 2024
to 10th, 2024 Industry News Lexaria Updates Fast-Moving GLP-1 'Arm's Race' Developments Five protein-design
- TM5-TM6: structural switches that modulate the coupling of serotonin receptors to Gs or Gi
is of great importance in GPCRs field as it supports the development of alternatives to improve drug design
- How Collaboration Drives GPCR Discoveries
It will hinge on the teams who can map GPCR signaling with precision and design therapies that fit real
- 📰 GPCR Weekly News, May 22 to 28, 2023
GPCR Binders, Drugs, and more Design of Drug Efficacy Guided by Free Energy Simulations of the β2 -Adrenoceptor
- 📰 GPCR Weekly News, January 23 to 29, 2023
Design, synthesis, and evaluation of substituted alkylindoles that activate G protein-coupled receptors
- 📰 GPCR Weekly News - January 9 to 15, 2023
Modelling altered signalling of G-protein coupled receptors in inflamed environment to advance drug design
- Fluorescence based HTS compatible ligand binding assays for dopamine D3 receptors in baculovirus preparations and live cells
Altogether, these aspects hint that the linker design and strategy can provide options for the tuning Structure-Based Design of High-Affinity Fluorescent Probes for the Neuropeptide Y Y1 Receptor. J. An Order of Magnitude Faster DNA-PAINT Imaging by Optimized Sequence Design and Buffer Conditions.
- Targeting GPCRs in the CNS: Advances in Drug Discovery Strategies
, Activation, and Signaling Pathways in the Brain An understanding of GPCR structure is key in drug design
- The mouse cytomegalovirus G protein-coupled receptor homolog, M33, coordinates key features of ...
The mouse CMV (MCMV) GPCR homolog, designated M33, is important for cell-associated virus spread and
- 📰 GPCR Buzz: August 5-11, 2024 | Top Highlights from DrGPCR University!
Submit your design for our Logo Contest by August 15, 2024 (Yes, it's TODAY)!
- Fentanyl and Xylazine: Why Breathing Fails in Overdose
Catherine’s work lays the foundation for designing better interventions, from preclinical models to clinical
- Exploring the Breakthroughs in GPCR Research
Logo Contest: Unleash your creativity and submit your design by August 15, 2024.
- 📰 GPCR Weekly News, June 24 to 30, 2024
Logo Contest: Unleash your creativity and submit your design by August 15th, 2024 Sponsorship Opportunities
- 📰 GPCR Weekly News, December 4 to 10, 2023
protein-coupled receptor C3aR1 reveals ligand-mediated biased agonism GPCR Binders, Drugs, and more Design
- 📰 GPCR Weekly News, July 24 to July 30, 2023
Specialist - Natural Sciences - Surgery Senior Scientist- Membrane Technologies Computational Protein Design
- From DNA day to GPCR genomics
genomics approaches, such as structural bioinformatics analysis, have facilitated drug discovery and design
- 📰 GPCR Weekly News, September 25 to October 1, 2023
You can submit your logo design by November 1st, and registration is unnecessary to participate.
- 📰 GPCR Weekly News, March 6 to 12, 2023
Novel Xanomeline-Containing Bitopic Ligands of Muscarinic Acetylcholine Receptors: Design, Synthesis
- Assay Sensitivity: The Hidden Lever Driving GPCR Drug Discovery
. ✅ Practical insights into designing assays that mimic pathophysiology , producing data with sharper
- Decoding GPCR Function: The Role of Mutagenesis in Rational Drug Discovery
G-protein coupled receptors: models, mutagenesis, and drug design.
- 📰 GPCR Weekly News, February 5 to 11, 2024
pharmacotherapeutic development updates Methods & Updates in GPCR Research GPCR-BERT: Interpreting Sequential Design
- 📰 Breaking Down the Latest GPCR Discoveries: a Weekly Update (Nov 27-Dec 3, 2023)
inhibitors of GPR52 using docking and biased sampling method for Huntington's disease therapy Rational design
- 📰 GPCR Weekly News, November 13 to 19, 2023
Screening System: A High-Throughput Engineering Platform for Genetically Encoded Fluorescent Indicators Design
- Why Biotech Fundraising Fails Due to Intellectual Property Gaps
Competitive patents are acknowledged but not contextualized 👉 There is no discussion of workarounds or design
- 📰 GPCR Weekly News, January 22 to 28, 2024
Receptor2 Pleckstrin Homology Binding Domain in Ovarian Cancer: Expression in Fallopian Tubes and Drug Design
- 📰 GPCR Weekly News, January 15 to 21, 2024
signaling GPCR Binders, Drugs, and more Computational Workflow for Refining AlphaFold Models in Drug Design
- Orthosteric Binding Experiments: How to Avoid the Most Common Data Pitfalls
Proper orthosteric binding design prevents those errors before they propagate into SAR narratives.
- 📰 GPCR Weekly News, July 1 to 7, 2024
Logo Contest: Unleash your creativity and submit your design by August 15th, 2024 Sponsorship Opportunities
- 📰 GPCR Weekly News, December 18 to 31, 2023
IpRGCs Synaptic plasticity via receptor tyrosine kinase/G-protein-coupled receptor crosstalk Optimized design
- GPCRs are not simple on-off switches: deep dive into GPCR-ligand interactions
Despite the existence of numerous drugs designed for this primary binding site, there are significant













