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- Unlock the Hidden Complexity Behind GPCRs—From Terry Kenakin’s Vault
In the foundational lesson of Terry’s Corner , Dr. Terry Kenakin invites us to challenge outdated assumptions and step into a new era of drug discovery. Now, Terry is opening the vault. This isn’t theory. Join Terry’s Corner and stay updated on the latest in GPCR research—delivered in a format that’s as approachable Unlock "Why Terry's Corner" now
- New Tools, Smart Signals, and The Kenakin Brief
Terry Kenakin is launching a new learning space with video courses, AMAs, and practical insights . Get a sneak peek and sign up for The Kenakin Brief—his free weekly newslette r. Terry’s Corner is coming soon. Dr. Terry Kenakin. You can already explore the platform and subscribe to The Kenakin Brief—our new newsletter packed with
- GPCR Allostery: Unlock Hidden Mechanisms and Make Smarter Drug Decisions
That’s exactly what Terry’s Corner delivers this week: high-impact insight into GPCR allostery, crafted Terry's Corner : Stop Chasing Affinity and Start Reading the System In this week’s cornerstone Terry’ Terry Kenakin reframes GPCRs as dynamic, allosteric sensors—far from static binding sites. To stay in the know on upcoming courses and AMA session, get the complementary Kenakin Brief , the weekly Terry Kenakin on “The Kinetics of Allostery: The Added Benefits of Allosteric Function.”
- GPCR Drug Discovery at Discovery on Target: Why This Track Is About More Than Receptors
I’m honored to be chairing a session in this track — with none other than Terry Kenakin on the speaker Kenakin from UNC and Terry's Corner We'll continue to update this section as new videos are released Kenakin at Discovery on Target Terry Kenakin’s work on functional selectivity has transformed GPCR Kenakin Himself If you’re part of the Dr. where Terry Kenakin breaks down receptor pharmacology, functional selectivity, and ligand bias in a
- Terry’s Corner, Celtarys' Leap, and the $7B GPCR Horizon
Kenakin. Get curated content at your own pace. Subscribe to The Kenakin Brief below to stay in the know. Terry Kenakin Terry’s Corner is your space focused on GPCR pharmacology designed just for you. Terry Kenakin brings translational clarity to complex receptor concepts. Advance with nuanced lessons on allostery, residence time, and translational PK/PD Subscribe to The Kenakin
- Signals in Motion: Pain, Metabolism & Terry’s Corner
Hello GPCR Innovators , We’re preparing to launch Terry’s Corner, a new knowledge hub shaped by Dr. Terry Kenakin’s decades of GPCR insight. Kenakin Four decades of receptor theory now fit in one expert-guided hub. Terry’s Corner gives you timeless and timely tools to improve selectivity, model efficacy, and design Sign Up for The Kenakin Brief Fluorescent Ligands vs.
- Pharmacology at Your Fingertips: Terry’s Corner Launches
Welcome Back, Discovery Drivers Terry’s Corner is live, on-demand pharmacology built for drug discovery Dr.GPCR Updates Terry’s Corner is Live - Pharmacology at your fingertips Terry’s Corner is now open! Terry Kenakin with short videos, clear summaries, and curated references. Want the full breakdown and your discount code for Terry's Corner? Better pharmacology leads to better decisions—unlock it now with Terry’s Corner.
- What If Your Data is Lying to You? The Calcium Assay Dilemma
In this foundational lesson, Terry Kenakin dives deep into a widely used, often misunderstood tool in Through real-world examples (like 5-HT2A and CCR5 agonists), Terry shows how slow-onset agonists can missteps, and use calcium assays with strategic clarity. 📍 Foundational Level | Calcium Assays 📚 Part of Terry Kenakin’s Pharmacology Vault 👉 Curious what else you've been missing?
- Pharmacologic Models
Terry Kenakin’s newest foundational lesson in Terry's Corner cuts straight to it: Why models are vital Probability Models This is practical drug development expertise from Terry’s 40+ years of experience Beyond the lessons, Terry's Corner is your exclusive gateway.
- Unlock the Hidden Lives of Receptors – Are You Ready?
In this exclusive Expert Drug Hunter lesson, Terry Kenakin dismantles 100 years of receptor theory and Step into Terry’s Vault and explore “Molecular Dynamics”—where expert drug hunters forge the future.
- Mapping Motion: Intermediate States, Deorphanization & Discovery
Terry Kenakin, and catch up on cutting-edge insights through our full library of symposia recordings, Terry Kenakin.
- Is Your Agonist Really “Working”—Or Are You Just Seeing What Your System Allows?
In this eye-opening module, Terry Kenakin explores a concept that could change how you interpret pharmacological Through powerful analogies (think batteries and balance scales), Terry reveals why different tissues—and emerging drug hunter, this lesson is your bridge from data confusion to predictive clarity. 👉 Dive into Terry
- Pharmacology Isn't What You Think—It's So Much More
Welcome to Terry’s Corner , where foundational pharmacology is demystified by someone who’s spent over In his newest lesson, “The Uniqueness of Pharmacology in Drug Discovery,” Terry Kenakin explains why Whether you're heading into your first assay or trying to make sense of inconsistent data, Terry gives Don’t just look at the data—learn how to read the story it’s telling. 👉 Start your journey with Terry
- What If the Most Important Part of Your Drug Isn’t What It Binds—But What It Does?
In Terry Kenakin’s latest lesson, you’ll uncover why efficacy is the unsung hero of drug discovery and Terry walks you through real-world experiments, decades of receptor pharmacology wisdom, and the cutting-edge 🔓 Find the lesson in Terry’s Pharmacology Vault: “Efficacy and System Sensitivity Unlock "Agonism &
- Why Dose-Response Curves Are Pharmacology’s Secret Weapon
In the newest foundational lesson from Terry Kenakin’s Pharmacology Vault , we unlock the visual language In classic Terry style, the lecture walks you through: What dose-response curves are and why they’re
- Ever Wondered How Drugs Are Discovered?
Terry Kenakin , a veteran pharmacologist with over 40 years of industry experience. In this foundational-level lesson, Terry unpacks the real-life process behind discovering new drugs, trees The critical importance of translation —turning lab data into meaningful therapeutic outcomes Terry
- From Ox Liver to AI: How the History of Pharmacology Shapes Its Future
Terry Kenakin takes you on a captivating tour through the history of pharmacology : a journey that spans Kenakin also celebrates the giants on whose shoulders we stand—A.J. 👉 Join Terry’s Corner, your essential launchpad into the world of therapeutic science Unlock "The History
- Exclusive Access: Terry's Corner is LIVE + Your Premium Member Discount!
Today, we're thrilled to announce that Terry's Corner is officially live ! What's inside Terry's Corner? Kenakin himself for deeper dives A new lesson will drop every Tuesday, ensuring fresh insights are Explore Terry's Corner Better decisions start with better pharmacology. GPCR Team & Terry’s Desk
- Misread the Curve, Misjudge the Drug: Rethinking Antagonism in GPCR Pharmacology
This week in Terry’s Corner, Dr. Terry Kenakin reframes one of pharmacology’s most foundational ideas: the difference between competitive Unlock “Competitive Antagonism” Now Only in Terry’s Corner Why Terry’s Corner For discovery-phase teams Terry Kenakin Monthly Ask‑Me‑Anything sessions with live Q&A An expanding on‑demand library for novices Subscribe to The Kenakin Brief today ➤ #GPCRantagonism #CompetitiveAntagonists #NonCompetitiveAntagonists
- Allosteric Binding Demystified: Smarter GPCR Drug Discovery
Terry's Corner - The Truth About Allosteric Displacement Allosteric binding isn’t just a twist in the Terry Kenakin exposes why traditional displacement logic breaks down in allosteric systems, and how overlooking Terry Kenakin on The Kinetics of Allostery . Exclusive Discount: Use code DRGPCR25 for $200 off. Kenakin is a leading expert in the field. Kenakin is a masterful teacher and communicator." — DrGPCR University Attendee The difference between
- Inside Out: Mapping GPCRs from Membrane Codes to Market Moves
Terry Kenakin, these five modules reveal how location bias, intracellular signaling, and ligand kinetics
- Why Kinetics Matter More Than Kd in GPCR Drug Discovery
That’s exactly what Terry’s Corner delivers this week: real-world kinetic frameworks to help you move Terry Kenakin’s latest lecture in Terry’s Corner delivers exactly what your discovery teams need now Premium Members get 50%+ discount when they join Terry’s Corner. 🔒 Available only in Terry’s Corner Kenakin is a masterful teacher and communicator—and a leading expert in our field.” — Dr. Terry Kenakin’s featured talk on “The Kinetics of Allostery” offers a rare live glimpse into advanced
- The Hidden Driver of GPCR Drug Success: Why Target Residence Time Matters More Than You Think
Terry Kenakin's insights on target residence time can reshape how you evaluate and advance lead compounds Terry's Corner - Unlock the Power of Target Residence Time in Your GPCR Drug Discovery Pipeline Gain Terry Kenakin’s latest insights delve into target residence time, revealing why kinetic persistence often ➡️ Premium Members get 50%+ discount when they join Terry’s Corner.
- From Venice to Virtual Molecules: Alessandro Nicoli’s Unexpected Journey into Computational Chemistry
Explore the GPCR University or enroll in Terry's Corner for GPCR Courses led by Dr. Terry Kenakin. ________ Keyword Cloud: #GPCRresearch #DrugDiscovery #ComputationalChemistry #MolecularModeling
- How Understanding Intracellular Drug Access Can Transform Your GPCR Drug Discovery Program
That’s exactly what Terry’s Corner delivers every week: practical tools from Dr. Terry Kenakin to elevate your science and sharpen your decisions. Terry Kenakin delivers a game-changing framework for teams grappling with the gap between in vitro potency To stay in the know on upcoming courses and AMA session, get the complementary Kenakin Brief , the weekly Kenakin) teaming up with the best GPCR community platform to help train and inspire the next generation
- Enhancing GPCR Research Outreach | Dr GPCR University early-bird registration ends soon!
Terry Kenakin with our premium membership and enjoy a 1-month FREE trial! Terry Kenakin Reading Materials Access to the private group Certificate of participation Learn the essentials
- Breaking the Myth of High and Low Affinity Sites
Kenakin’s Emerging Drug Hunter lecture delivers exclusive, cutting-edge insights that help you move But as Terry Kenakin reveals, this interpretation can be misleading, and sticking with it could slow Kenakin challenges this assumption and shows that what you’re seeing may reflect something entirely different Unlock “Rethinking Affinity” Now Only in Terry's Corner _____ #GPCR #BindingAffinity #Pharmacology
- Understanding Orthosteric Binding: The Key to Drug Action
Join Terry Kenakin as he pulls back the curtain on the deceptively simple process of orthosteric binding—the Key Concepts in Binding Terry unpacks several key concepts related to orthosteric binding: Langmuir Adsorption
- Transformative GPCR Insights: Unleash New Horizons in Science | Sep 9 - 15, 2024
Terry Kenakin and Sam Hoare ! Terry Kenakin to gain insights and prepare for upcoming courses. Kenakin's upcoming courses. Our goal is to ensure that education is within reach for everyone!
- Target Residence Time: The Hidden Driver of In Vivo Efficacy
Kenakin’s latest lecture delivers a paradigm shift for pharmacologists working on drugs where in vitro From restricted tissue diffusion to PK–PD dissociation, Kenakin equips you with the kinetic models and Kenakin walks through cases where two equipotent ligands produce radically different clinical outcomes Kenakin offers not just theory, but tools to model, predict, and validate this behavior early. Terry Kenakin Monthly Ask‑Me‑Anything sessions with live Q&A An expanding on‑demand library for novices