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Mark your calendars for these important events: September 22: Save the date for the Dr. ASCEPT Annual Scientific Meeting February 3 - 7, 2024 | SLAS2024 International Conference and Exhibition March 23 - 24, 2024 | Ligand Recognition and Molecular Gating Seminar March 24 - 29, 2024 | Ligand Recognition

Mark your calendar, it's happening September 22-25, 2025. Aaron McGrath from Takeda   🎥 Interview with Kris Borzilleri & Alison Heick Varghese from Pfizer 🎥 Let’s move GPCR drug discovery forward — together. 🚨 Mark your calendar for the GPCR Happy Hour Join

Must-read publications:  A structural modeling study revealing non-canonical mechanisms of chemokine-driven

appointed President of Heptares Therapeutics Ltd., and Head of UK R&D Tokyo, Japan and Cambridge, UK, 24 March

effectors along the Gαq/Phospholipase C (PLC) pathway, which results in an IkB kinases (IKK)-mediated canonical

blood group antigen ( Cutbush et al., 1950 ), also called Duffy-antigen/receptor for chemokines, or DARC

GPCR Events Mark your glittery calendar with dates in 2025 ! February 16 - 21, 2025 | Harnessing the Power of Advanced Multimodal Approaches to GPCR Drug Discovery March 12 - 14, 2025 | NextGen Biomed 2025 March 25 - 28, 2025 | 10th German Pharm-Tox Summit April 1 - 5,

non-cognate G proteins can enhance the coupling efficiency of cognate G proteins to GPCRs, thereby amplifying canonical

It’s time to mark your calendars and save the dates—let’s make some stellar memories together! February 16 - 21, 2025 | Harnessing the Power of Advanced Multimodal Approaches to GPCR Drug Discovery NEW March 12 - 14, 2025 | NextGen Biomed 2025 NEW March 25 - 28, 2025 | 10th German Pharm-Tox Summit NEW April

genes unveiled via RNA polymerase II degradation Growth factor-dependent phosphorylation of Gαi shapes canonical

GPCR-Targeted Drug Discovery Summit | February 21-23, Boston. 2nd ERNEST Training School – February 20th to March GEM2023 (14-17 March 2023). 8th and final ERNEST Meeting May 3-7, 2023 in Crete.

GPCR-Targeted Drug Discovery Summit | February 21-23, Boston. 2nd ERNEST Training School – February 20th to March GEM2023 (14-17 March 2023). 8th and final ERNEST Meeting May 3-7, 2023 in Crete.

of titratable residues spans from the extracellular surface to the transmembrane area, linking with canonical

We’ve also highlighted the latest research on non-canonical internalization mechanisms of mGlu receptors Gain the insights, tools, and connections you need to excel in your field and make your mark.

July 21st marks our next Dr. , 2023) Structure, Mechanism, and Drug Interactions of GPCRs, Ion Channels, and Transport Proteins (March

, 2023) Structure, Mechanism, and Drug Interactions of GPCRs, Ion Channels, and Transport Proteins (March

Before we dive into the latest news, mark your calendars for July 21st for our next Dr. Structure, Mechanism, and Drug Interactions of GPCRs, Ion Channels, and Transport Proteins (March 24

Graaf, C., et al., Glucagon-Like Peptide-1 and Its Class B G Protein-Coupled Receptors: A Long March

experimental design, wet lab work is performed to acquire high-content cell images, which then require several canonical

This week's highlight includes congrats to: Clementine E Philibert and Mikel Garcia-Marcos for their

Mikel Garcia-Marcos for their work on Get ready to sharpen your tools:A short guide to heterotrimeric Early-bird registration for premium Ecosystem members opens on July 31st, so mark your calendars and

into this week’s news, we’d like to draw your attention to some of our events and resources: Please mark 2023) NEW Structure, Mechanism, and Drug Interactions of GPCRs, Ion Channels, and Transport Proteins (March

Registrations close on September 6 at 12pm EST Mark your calendars for September 22nd! , 2023) Structure, Mechanism, and Drug Interactions of GPCRs, Ion Channels, and Transport Proteins (March

, 2023) Structure, Mechanism, and Drug Interactions of GPCRs, Ion Channels, and Transport Proteins (March

🎇 This Week’s Highlights: Congrats to: Remi Janicot , and Mikel Garcia-Marcos for their excellent

Cardarelli's research: Burixafor Hydrobromide (GPC-100) effects on hematopoietic cells in mice and humans Mark , 2023) Structure, Mechanism, and Drug Interactions of GPCRs, Ion Channels, and Transport Proteins (March

.; Farce, A.; Chavatte, P.; Poupaert, J. H.; Lambert, D. M.; Depreux, P.; Hénichart, J.-P.

Sir James Whyte Black OM. 14 June 192422 March 2010.