GPCR NewsOct 1, 20221 minStructural and Molecular InsightsMechanistic basis of GPCR activation explored by ensemble refinement of crystallographic structuresOctober 2022 "G protein-coupled receptors (GPCRs) are important drug targets characterized by a canonical seven transmembrane (TM) helix...
GPCR NewsOct 1, 20221 minStructural and Molecular InsightsMechanism of enhanced sensitivity of mutated β-adrenergic-like octopamine receptor to amitraz in...October 2022 Mechanism of enhanced sensitivity of mutated β-adrenergic-like octopamine receptor to amitraz in honeybee Apis mellifera: An...
GPCR NewsSep 1, 20221 minStructural and Molecular InsightsIsoforms of GPR35 have distinct extracellular N-termini that allosterically modify...September 2022 Isoforms of GPR35 have distinct extracellular N-termini that allosterically modify receptor-transducer coupling and...