GPCR NewsOct 1, 20221 minGPCR Activation and SignalingDimerization of β2-adrenergic receptor is responsible for the constitutive activity subjected to...October 2022 Dimerization of β2-adrenergic receptor is responsible for the constitutive activity subjected to inverse agonism...
GPCR NewsSep 1, 20221 minStructural and Molecular InsightsCholesterol occupies the lipid translocation pathway to block phospholipid scrambling by a GPCRSeptember 2022 "Class A (rhodopsin-like) G protein-coupled receptors (GPCRs) are constitutive phospholipid scramblases as evinced after...
GPCR NewsAug 1, 20221 minGPCR Activation and SignalingActivation of the human chemokine receptor CX3CR1 regulated by cholesterolAugust 2022 "As the only member of the CX3C chemokine receptor subfamily, CX3CR1 binds to its sole endogenous ligand CX3CL1, which shows...