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Orthosteric vs Allosteric Interactions— and the pHSense Shift in Internalization
Each edition highlights the decisions that move GPCR projects forward—from pharmacology essentials to ligand binding site strategies, bench-ready tools, and industry momentum shaping GPCR pipelines. Read fast, apply faster, and stay ahead in GPCR drug discovery with evidence-based insights—no hype, just strategies you can use.

Dr. GPCR News
Oct 25 min read


GPCR Allosteric Modulation: Why Allostery is the Engine of Drug Discovery
Explore how GPCRs function as dynamic allosteric machines in this expert-level breakdown from Dr. Terry Kenakin. Learn how probe dependence, cryptic binding sites, and conformational changes impact drug discovery and therapeutic design.

Terry's Desk
Jul 293 min read
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