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The program of the Dr. GPCR Summit from October 10th to the 16th is taking shape. Check it out today but first become a Dr. GPCR...
Dr. GPCR News
Sep 3, 20221 min read
🎧Episode 85 of the Dr. GPCR podcast is here!
Episode 85 of the Dr. GPCR podcast is here! 🎧Hear Dr. Nicholas Holliday and how he has combined his university role with his leadership...
Dr. GPCR News
Sep 2, 20221 min read
Immerse yourself in the Dr. GPCR Ecosystem!
Immerse yourself in the Dr. GPCR Ecosystem with a paid membership for extra benefits. Catch up with the latest #GPCR news, our monthly...
Dr. GPCR News
Sep 2, 20221 min read
Join the #GPCR movement today!
Did you know that you can enjoy a Dr. GPCR Ecosystem paid membership with extra benefits? Create your own group, watch the latest podcast...
Dr. GPCR News
Sep 1, 20221 min read
Join Dr. GPCR Summit 2022 in 3 simple steps!
🌟The Dr. GPCR event of the year is the 3rd edition of the Summit. Come join us from October 10 to 16 to hear about exciting #GPCR...
Dr. GPCR News
Sep 1, 20221 min read
Signaling pathways activated by sea bass gonadotropin-inhibitory hormone peptides in COS-7 cells...
September 2022 Signaling pathways activated by sea bass gonadotropin-inhibitory hormone peptides in COS-7 cells transfected with their...
GPCR News
Sep 1, 20221 min read
Expression pattern and clinical significance of beta 2-adrenergic receptor in oral squamous cell...
September 2022 Expression pattern and clinical significance of beta 2-adrenergic receptor in oral squamous cell carcinoma: an emerging...
GPCR News
Aug 31, 20221 min read
Upregulation of Phospholipase C Gene Expression Due to Norepinephrine-Induced Hypertrophic Response
September 2022 "The activation of phospholipase C (PLC) is thought to have a key role in the cardiomyocyte response to several different...
GPCR News
Aug 31, 20221 min read
Fentanyl activates ovarian cancer and alleviates chemotherapy-induced toxicity via opioid...
September 2022 Fentanyl activates ovarian cancer and alleviates chemotherapy-induced toxicity via opioid receptor-dependent activation of...
GPCR News
Aug 31, 20221 min read
Chemerin Forms: Their Generation and Activity
September 2022 "Chemerin is the product of the RARRES2 gene which is secreted as a precursor of 143 amino acids. That precursor is...
GPCR News
Aug 31, 20221 min read
PI(4,5)P 2-stimulated positive feedback drives the recruitment of Dishevelled to Frizzled in Wnt-β-c
September 2022 "In the Wnt-β-catenin pathway, Wnt binding to Frizzled (Fzd) and LRP5 or LRP6 (LRP5/6) co-receptors inhibits the...
GPCR News
Aug 31, 20221 min read
CCL25/CCR9 interaction promotes the malignant behavior of salivary adenoid cystic carcinoma via...
September 2022 CCL25/CCR9 interaction promotes the malignant behavior of salivary adenoid cystic carcinoma via the PI3K/AKT signaling...
GPCR News
Aug 31, 20221 min read
G protein coupling and activation of the metabotropic GABAB heterodimer
September 2022 "Metabotropic γ-aminobutyric acid receptor (GABABR), a class C G protein-coupled receptor (GPCR) heterodimer, plays a...
GPCR News
Aug 31, 20221 min read
GRK3 is a poor prognosticator and serves as a therapeutic target in advanced gastric adenocarcinoma
September 2022 "Background G protein-coupled receptor (GPCR) is the most targeted protein family by the FDA-approved drugs. GPCR-kinase 3...
GPCR News
Aug 31, 20221 min read
Neurotransmitters: Potential Targets in Glioblastoma
September 2022 "For decades, glioblastoma multiforme (GBM), a type of the most lethal brain tumor, has remained a formidable challenge in...
GPCR News
Aug 31, 20221 min read
GPCR/endocytosis/ERK signaling/S2R is involved in the regulation of the internalization...
September 2022 GPCR/endocytosis/ERK signaling/S2R is involved in the regulation of the internalization, mitochondria-targeting and...
GPCR News
Aug 31, 20221 min read
Structure of the human galanin receptor 2 bound to galanin and Gq reveals the basis of ligand...
September 2022 Structure of the human galanin receptor 2 bound to galanin and Gq reveals the basis of ligand specificity and how binding...
GPCR News
Aug 31, 20221 min read
Platelets in the NETworks interweaving inflammation and thrombosis
September 2022 "Platelets are well characterized for their indispensable role in primary hemostasis to control hemorrhage. Research over...
GPCR News
Aug 31, 20222 min read
Structure of Mycobacterium tuberculosis Cya, an evolutionary ancestor of the mammalian membrane...
September 2022 Structure of Mycobacterium tuberculosis Cya, an evolutionary ancestor of the mammalian membrane adenylyl cyclases...
GPCR News
Aug 31, 20221 min read
Ginsenoside Rg5 allosterically interacts with P2RY12 and ameliorates deep venous thrombosis by...
September 2022 Ginsenoside Rg5 allosterically interacts with P2RY12 and ameliorates deep venous thrombosis by counteracting neutrophil...
GPCR News
Aug 31, 20221 min read
C5aR2 receptor: The genomic twin of the flamboyant C5aR1
September 2022 "The complement fragment C5a is one of the most potent proinflammatory glycoproteins liberated by the activation of the...
GPCR News
Aug 31, 20221 min read
C1-inhibitor influence on platelet activation by thrombin receptors agonists
September 2022 "Introduction Protease activated receptors 1 (PAR1) and 4 (PAR4) agonists are used to study platelet activation. Data on...
GPCR News
Aug 31, 20221 min read
Residency time of agonists does not affect the stability of GPCR-arrestin complexes
September 2022 "Background and purpose: The interaction of arrestins with G-protein coupled receptors (GPCRs) desensitizes...
GPCR News
Aug 31, 20221 min read
Cell-Type-Specific Effects of the Ovarian Cancer G-Protein Coupled Receptor (OGR1) on Inflammation..
September 2022 Cell-Type-Specific Effects of the Ovarian Cancer G-Protein Coupled Receptor (OGR1) on Inflammation and Fibrosis; Potential...
GPCR News
Aug 31, 20221 min read
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