top of page
Insights That Move the GPCR Field Forward
Read the latest analyses, interviews, and discoveries shaping the GPCR ecosystem — from research breakthroughs to biotech strategy.
GPCR News powered by our Strategic Partners
Blog: Blog2
Search
GPR108 is required for gambogic acid inhibiting NF-κB signaling in cancer
September 2022 "GPCRs are the most potential targets for drug discovery, however, their role in oncology is underappreciated and...
GPCR News
Aug 31, 20221 min read
Dynamics of tumor-associated macrophages in a quantitative systems pharmacology model of...
September 2022 Dynamics of tumor-associated macrophages in a quantitative systems pharmacology model of immunotherapy in triple-negative...
GPCR News
Aug 31, 20221 min read
GPCR kinase phosphorylation of distal C-tail sites specifies βarrestin1-mediated signaling by...
September 2022 "G protein-coupled receptor (GPCR) kinases (GRKs) and arrestins mediate GPCR desensitization, internalization, and...
GPCR News
Aug 31, 20221 min read
The Impact of CB1 Receptor on Nuclear Receptors in Skeletal Muscle Cells
September 2021 "Cannabinoids are abundant signaling compounds; their influence predominantly arises via engagement with the principal two...
GPCR News
Aug 31, 20222 min read
Biased GPCR signaling by the native parathyroid hormone-related protein 1 to 141 relative to its...
September 2022 Biased GPCR signaling by the native parathyroid hormone-related protein 1 to 141 relative to its N-terminal fragment 1 to...
GPCR News
Aug 31, 20221 min read
Opposite Effects of Src Family Kinases on YAP and ERK Activation in Pancreatic Cancer Cells...
September 2022 Opposite Effects of Src Family Kinases on YAP and ERK Activation in Pancreatic Cancer Cells: Implications for Targeted...
GPCR News
Aug 31, 20221 min read
Sign Up Now!
🌐 🤝 We want to bring closer the #GPCR community! Join the Dr. GPCR Ecosystem as a site member today for FREE and start exploring! Sign...
Dr. GPCR News
Aug 31, 20221 min read
Dr. GPCR Summit 2022 is coming!
The 3rd edition of the Dr. GPCR Summit is between October 10th to the 16th! 💡Trainees are invited to participate by presenting a trainee...
Dr. GPCR News
Aug 30, 20221 min read
Join Us Today!
🌐Dr. GPCR Ecosystem is under construction and dozens of your colleagues are enjoying its benefits! Catch up with the latest #GPCR news,...
Dr. GPCR News
Aug 29, 20221 min read
Trainees, this is for you...
🔎 Are you a trainee? Would you like to develop your presentation skills? Give a talk or present a poster at the Dr. GPCR Summit 2022....
Dr. GPCR News
Aug 27, 20221 min read
Dr. Rosie Dawaliby Podcast!
We're very excited to announce the next episode of the Dr. GPCR podcast! 🥁 Drum rolls, please! Our guest is the wonderful Dr. Rosie...
Dr. GPCR News
Aug 26, 20221 min read
Join Us Now!
🌟 We're so excited about our upcoming Dr. GPCR Summit 2022. This is a great opportunity for us to come together and talk GPCRs. Do you...
Dr. GPCR News
Aug 25, 20221 min read
Learn about Dr. GPCR Ecosystem!
💻Did you know that Dr. GPCR is much more than a podcast? Come check out the brand new Dr. GPCR Ecosystem and explore its benefits! We...
Dr. GPCR News
Aug 24, 20221 min read
Dr. GPCR Summit is FREE for Ecosystem site members!
📢 Did you know that this 3rd Edition of the Dr. GPCR Summit is totally FREE for our Ecosystem site members? Join us and become a site...
Dr. GPCR News
Aug 23, 20221 min read
Opioid Ligands Addressing Unconventional Binding Sites and More Than One Opioid Receptor Subtype
August 2022 "Opioid receptors (ORs) represent one of the most significant groups of G-protein coupled receptor (GPCR) drug targets and...
GPCR News
Aug 1, 20221 min read
In vitro assays for the functional characterization of (psychedelic) substances at the serotonin...
August 2022 In vitro assays for the functional characterization of (psychedelic) substances at the serotonin receptor 5-HT2A R...
GPCR News
Aug 1, 20221 min read
Activation of the human chemokine receptor CX3CR1 regulated by cholesterol
August 2022 "As the only member of the CX3C chemokine receptor subfamily, CX3CR1 binds to its sole endogenous ligand CX3CL1, which shows...
GPCR News
Jul 31, 20221 min read
Murine bone marrow macrophages and human monocytes do not express atypical chemokine receptor 1
August 2022 "The atypical chemokine receptor 1 (ACKR1) was discovered on erythrocytes as the Duffy blood group antigen ( Cutbush et al.,...
GPCR News
Jul 31, 20221 min read
Dopamine D 1 receptor-mediated β-arrestin signaling: Insight from pharmacology, biology, behavior...
August 2022 Dopamine D 1 receptor-mediated β-arrestin signaling: Insight from pharmacology, biology, behavior, and neurophysiology "The...
GPCR News
Jul 31, 20221 min read
Production of human A2AAR in lipid nanodiscs for 19F-NMR and single-molecule fluorescence...
August 2022 Production of human A 2A AR in lipid nanodiscs for 19 F-NMR and single-molecule fluorescence spectroscopy "We describe...
GPCR News
Jul 31, 20221 min read
A correlation study of adhesion G protein-coupled receptors as potential therapeutic targets in...
August 2022 A correlation study of adhesion G protein-coupled receptors as potential therapeutic targets in Uterine Corpus Endometrial...
GPCR News
Jul 31, 20221 min read
8th RSC / SCI symposium on GPCRs in Medicinal Chemistry. October 5-7, 2022, Verona, Italy
August 2022 "GPCRs in Medicinal Chemistry Event 8th RSC / SCI symposium on GPCRs in Medicinal Chemistry Dates Wednesday-Friday, 5th-7th...
GPCR News
Jul 31, 20221 min read
Structure Therapeutics Extends Financing, Advances Diabetes and Obesity Clinical Program and...
August 2022 Structure Therapeutics Extends Financing, Advances Diabetes and Obesity Clinical Program and Changes Name from ShouTi "San...
GPCR News
Jul 31, 20221 min read
Therapeutic validation of an orphan G protein-coupled receptor: The case of GPR84
August 2022 "Despite the importance of members of the GPCR superfamily as targets of a broad range of effective medicines many GPCRs...
GPCR News
Jul 31, 20221 min read
bottom of page