Insights That Move the GPCR Field Forward

Read the latest analyses, interviews, and discoveries shaping the GPCR ecosystem — from research breakthroughs to biotech strategy.

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GPCR Articles

📰 GPCR Weekly News, February 6 to 12, 2023

Hello Readers👋, We're excited to share our weekly newsletter with you. Keep up-to-date with the latest research and advancements in the...

GPCR News

Feb 16, 20232 min read

New role of β-arrestins in MOR signaling

With around 187 people dying every day from an opioid overdose in the U.S., combatting the opioid overdose epidemic has become a mean...

Monserrat Avila-Zozaya

Feb 13, 20233 min read

📰 GPCR Weekly News, January 30 to February 5, 2023

Hello Readers👋, We're excited to share our weekly newsletter with you. Keep up-to-date with the latest research and advancements in the...

GPCR News

Feb 9, 20233 min read

📰 GPCR Weekly News, January 23 to 29, 2023

Hello Readers👋, We're excited to share our weekly newsletter with you. Keep up-to-date with the latest research and advancements in the...

GPCR News

Feb 2, 20232 min read

Unlocking the Therapeutic Potential of Previously Undruggable GPCRs

Executive Summary This whitepaper will provide an overview of G Protein-Coupled Receptors (GPCRs) and discuss current trends in GPCR drug...

Orion Biotechnology

Feb 1, 202310 min read

📰 GPCR Weekly News, January 16 to 22, 2023

Hello Readers👋, We're excited to share our weekly newsletter with you. Keep up-to-date with the latest research and advancements in the...

GPCR News

Jan 26, 20232 min read

📰 GPCR Weekly News - January 9 to 15, 2023

Hello Readers👋, We're excited to share our weekly newsletter with you. Keep up-to-date with the latest research and advancements in the...

GPCR News

Jan 19, 20232 min read

Odorant receptors – a bit of smell for drug discovery

Odorant receptors function and expression landscape Odorant receptors (ORs) belong to the G protein-coupled receptor (GPCR) family and...

Inês Pinheiro

Jan 13, 20234 min read

📰 GPCR Weekly News - January 2 to 8, 2023

Hello Readers👋, We're excited to share our weekly newsletter with you. Keep up-to-date with the latest research and advancements in the...

GPCR News

Jan 12, 20232 min read

📰 GPCR Weekly News

Hello Readers👋, Happy New Year! We're excited to be back and share our weekly newsletter! We'll be sending it directly to your inbox...

GPCR News

Jan 5, 20233 min read

📰 GPCR Weekly News

Hello Readers👋, We are working on bringing your the latest GPCR News more frequently directly in your inbox and in the Ecosystem. Below...

GPCR News

Dec 22, 20222 min read

Overview of adhesion GPCRs self-activation

Among the different families of G-protein-coupled receptors (GPCRs), adhesion GPCRs (aGPCRs) represent the second most abundant in humans....

Monserrat Avila-Zozaya

Dec 18, 20224 min read

📰 GPCR Weekly News

Hello Readers👋, Get the latest GPCR News more frequently directly in your inbox and in the Ecosystem. Below is your Classified GPCR News...

GPCR News

Dec 15, 20222 min read

📰 GPCR Weekly News

Hello Readers👋, We are working on bringing your the latest GPCR News more frequently directly in your inbox and in the Ecosystem. Below...

GPCR News

Dec 9, 20223 min read

Transmembrane domains of GPCR dimers – a novel hot spot for drug discovery

Transmembrane domains of GPCR dimers – a novel hot spot for drug discovery G-protein-coupled receptors (GPCRs) can form biologically...

Inês Pinheiro

Dec 6, 20223 min read

Ode to GPCRs

Every year, with the month of October, comes the excitement of the Nobel session to the global scientific community. In the first few...

Nipuna Weerasinghe

Nov 14, 20228 min read

Emerging approaches for decoding neuropeptide transmission

November 2022 "Neuropeptides produce robust effects on behavior across species, and recent research has benefited from advances in...

GPCR Papers

GPCR News

Nov 1, 20221 min read

Location bias contributes to functionally selective responses of biased CXCR3 agonists

November 2022 "Some G protein-coupled receptor (GPCR) ligands act as "biased agonists" that preferentially activate specific signaling...

GPCR Papers

GPCR News

Nov 1, 20221 min read

Deciphering the signaling mechanisms of β-arrestin1 and β-arrestin2 in regulation of cancer cell...

November 2022 Deciphering the signaling mechanisms of β-arrestin1 and β-arrestin2 in regulation of cancer cell cycle and metastasis...

GPCR Papers

GPCR News

Nov 1, 20221 min read

Structure-Based Discovery of Negative Allosteric Modulators of the Metabotropic Glutamate Receptor 5

November 2022 "Recently determined structures of class C G protein-coupled receptors (GPCRs) revealed the location of allosteric binding...

GPCR Papers

GPCR News

Nov 1, 20221 min read

Structural insights into adhesion GPCR ADGRL3 activation and Gq, Gs, Gi, and G12 coupling

November 2022 "Adhesion G-protein-coupled receptors (aGPCRs) play key roles in a diversity of physiologies. A hallmark of aGPCR...

GPCR Papers

GPCR News

Nov 1, 20221 min read

Conservation of Allosteric Ligand Binding Sites in G-Protein Coupled Receptors

November 2022 "Despite the growing number of G protein-coupled receptor (GPCR) structures, only 39 structures have been cocrystallized...

GPCR Papers

GPCR News

Nov 1, 20221 min read

Dimerization of β2-adrenergic receptor is responsible for the constitutive activity subjected to inv

November 2022 "Dimerization of beta 2-adrenergic receptor (β2-AR) has been observed across various physiologies. However, the function of...

GPCR Papers

GPCR News

Nov 1, 20221 min read

High hedgehog signaling is transduced by a multikinase-dependent switch controlling the...

October 2022 High hedgehog signaling is transduced by a multikinase-dependent switch controlling the apico-basal distribution of the GPCR...

GPCR Papers

GPCR News

Oct 1, 20221 min read

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